Title : Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors - Di Stefano_2023_Eur.J.Med.Chem_263_115916 |
Author(s) : Di Stefano M , Masoni S , Bononi G , Poli G , Galati S , Gado F , Manzi S , Vagaggini C , Brai A , Caligiuri I , Asif K , Rizzolio F , Macchia M , Chicca A , Sodi A , Di Bussolo V , Minutolo F , Meier P , Gertsch J , Granchi C , Dreassi E , Tuccinardi T |
Ref : Eur Journal of Medicinal Chemistry , 263 :115916 , 2023 |
Abstract : |
PubMedSearch : Di Stefano_2023_Eur.J.Med.Chem_263_115916 |
PubMedID: 37976705 |
Title : Reversible Monoacylglycerol Lipase Inhibitors: Discovery of a New Class of Benzylpiperidine Derivatives - Bononi_2022_J.Med.Chem__ |
Author(s) : Bononi G , Di Stefano M , Poli G , Ortore G , Meier P , Masetto F , Caligiuri I , Rizzolio F , Macchia M , Chicca A , Avan A , Giovannetti E , Vagaggini C , Brai A , Dreassi E , Valoti M , Minutolo F , Granchi C , Gertsch J , Tuccinardi T |
Ref : Journal of Medicinal Chemistry , : , 2022 |
Abstract : |
PubMedSearch : Bononi_2022_J.Med.Chem__ |
PubMedID: 35522977 |
Title : Single-Cell Approach to Monitor the Unfolded Protein Response During Biotechnological Processes With Pichia pastoris - Raschmanova_2019_Front.Microbiol_10_335 |
Author(s) : Raschmanova H , Zamora I , Borcinova M , Meier P , Weninger A , Machler D , Glieder A , Melzoch K , Knejzlik Z , Kovar K |
Ref : Front Microbiol , 10 :335 , 2019 |
Abstract : |
PubMedSearch : Raschmanova_2019_Front.Microbiol_10_335 |
PubMedID: 30873140 |
Title : Structure of lipoprotein lipase in complex with GPIHBP1 - Arora_2019_Proc.Natl.Acad.Sci.U.S.A_116_10360 |
Author(s) : Arora R , Nimonkar AV , Baird D , Wang C , Chiu CH , Horton PA , Hanrahan S , Cubbon R , Weldon S , Tschantz WR , Mueller S , Brunner R , Lehr P , Meier P , Ottl J , Voznesensky A , Pandey P , Smith TM , Stojanovic A , Flyer A , Benson TE , Romanowski MJ , Trauger JW |
Ref : Proc Natl Acad Sci U S A , 116 :10360 , 2019 |
Abstract : |
PubMedSearch : Arora_2019_Proc.Natl.Acad.Sci.U.S.A_116_10360 |
PubMedID: 31072929 |
Gene_locus related to this paper: human-LPL |