| Title : Discovery of reversible monoacylglycerol lipase (MAGL) inhibitors based on ortho-hydroxyanilide scaffold - Bononi_2025_Bioorg.Chem_163_108698 |
| Author(s) : Bononi G , Gado F , Masoni S , Scalabrini D , Vedova LD , Di Stefano M , Piazza L , Poles C , Lonzi C , Landucci E , Vagaggini C , Poggialini F , Brai A , Caligiuri I , Rizzolio F , Mohamed KA , Bertini S , De Lorenzi E , Dreassi E , Macchia M , Minutolo F , Laprairie RB , Granchi C , Tuccinardi T |
| Ref : Bioorg Chem , 163 :108698 , 2025 |
| Abstract : |
| PubMedSearch : Bononi_2025_Bioorg.Chem_163_108698 |
| PubMedID: 40554889 |
| Gene_locus related to this paper: human-MGLL |
| Title : Watermelon: setup and validation of an in silico fragment-based approach - Di Stefano_2024_J.Enzyme.Inhib.Med.Chem_39_2356179 |
| Author(s) : Di Stefano M , Galati S , Piazza L , Gado F , Granchi C , Macchia M , Giordano A , Tuccinardi T , Poli G |
| Ref : J Enzyme Inhib Med Chem , 39 :2356179 , 2024 |
| Abstract : |
| PubMedSearch : Di Stefano_2024_J.Enzyme.Inhib.Med.Chem_39_2356179 |
| PubMedID: 38864179 |
| Title : Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors - Di Stefano_2023_Eur.J.Med.Chem_263_115916 |
| Author(s) : Di Stefano M , Masoni S , Bononi G , Poli G , Galati S , Gado F , Manzi S , Vagaggini C , Brai A , Caligiuri I , Asif K , Rizzolio F , Macchia M , Chicca A , Sodi A , Di Bussolo V , Minutolo F , Meier P , Gertsch J , Granchi C , Dreassi E , Tuccinardi T |
| Ref : Eur Journal of Medicinal Chemistry , 263 :115916 , 2023 |
| Abstract : |
| PubMedSearch : Di Stefano_2023_Eur.J.Med.Chem_263_115916 |
| PubMedID: 37976705 |
| Gene_locus related to this paper: human-ABHD6 |
| Title : Modification on the 1,2-dihydro-2-oxo-pyridine-3-carboxamide core to obtain multi-target modulators of endocannabinoid system - Gado_2019_Bioorg.Chem__103353 |
| Author(s) : Gado F , Arena C , Fauci C , Reynoso-Moreno I , Bertini S , Digiacomo M , Meini S , Poli G , Macchia M , Tuccinardi T , Gertsch J , Chicca A , Manera C |
| Ref : Bioorg Chem , :103353 , 2019 |
| Abstract : |
| PubMedSearch : Gado_2019_Bioorg.Chem__103353 |
| PubMedID: 31668465 |
| Title : Polypharmacological profile of 1,2-dihydro-2-oxo-pyridine-3-carboxamides in the endocannabinoid system - Chicca_2018_Eur.J.Med.Chem_154_155 |
| Author(s) : Chicca A , Arena C , Bertini S , Gado F , Ciaglia E , Abate M , Digiacomo M , Lapillo M , Poli G , Bifulco M , Macchia M , Tuccinardi T , Gertsch J , Manera C |
| Ref : Eur Journal of Medicinal Chemistry , 154 :155 , 2018 |
| Abstract : |
| PubMedSearch : Chicca_2018_Eur.J.Med.Chem_154_155 |
| PubMedID: 29793210 |