| Title : Discovery of reversible monoacylglycerol lipase (MAGL) inhibitors based on ortho-hydroxyanilide scaffold - Bononi_2025_Bioorg.Chem_163_108698 |
| Author(s) : Bononi G , Gado F , Masoni S , Scalabrini D , Vedova LD , Di Stefano M , Piazza L , Poles C , Lonzi C , Landucci E , Vagaggini C , Poggialini F , Brai A , Caligiuri I , Rizzolio F , Mohamed KA , Bertini S , De Lorenzi E , Dreassi E , Macchia M , Minutolo F , Laprairie RB , Granchi C , Tuccinardi T |
| Ref : Bioorg Chem , 163 :108698 , 2025 |
| Abstract : |
| PubMedSearch : Bononi_2025_Bioorg.Chem_163_108698 |
| PubMedID: 40554889 |
| Gene_locus related to this paper: human-MGLL |
| Title : Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors - Di Stefano_2023_Eur.J.Med.Chem_263_115916 |
| Author(s) : Di Stefano M , Masoni S , Bononi G , Poli G , Galati S , Gado F , Manzi S , Vagaggini C , Brai A , Caligiuri I , Asif K , Rizzolio F , Macchia M , Chicca A , Sodi A , Di Bussolo V , Minutolo F , Meier P , Gertsch J , Granchi C , Dreassi E , Tuccinardi T |
| Ref : Eur Journal of Medicinal Chemistry , 263 :115916 , 2023 |
| Abstract : |
| PubMedSearch : Di Stefano_2023_Eur.J.Med.Chem_263_115916 |
| PubMedID: 37976705 |
| Gene_locus related to this paper: human-ABHD6 |
| Title : Reversible Monoacylglycerol Lipase Inhibitors: Discovery of a New Class of Benzylpiperidine Derivatives - Bononi_2022_J.Med.Chem__ |
| Author(s) : Bononi G , Di Stefano M , Poli G , Ortore G , Meier P , Masetto F , Caligiuri I , Rizzolio F , Macchia M , Chicca A , Avan A , Giovannetti E , Vagaggini C , Brai A , Dreassi E , Valoti M , Minutolo F , Granchi C , Gertsch J , Tuccinardi T |
| Ref : Journal of Medicinal Chemistry , : , 2022 |
| Abstract : |
| PubMedSearch : Bononi_2022_J.Med.Chem__ |
| PubMedID: 35522977 |