| Title : Discovery of Trifluoromethyl Glycol Carbamates as Potent and Selective Covalent Monoacylglycerol Lipase (MAGL) Inhibitors for Treatment of Neuroinflammation - McAllister_2018_J.Med.Chem_61_3008 |
| Author(s) : McAllister LA , Butler CR , Mente S , O'Neil SV , Fonseca KR , Piro JR , Cianfrogna JA , Foley TL , Gilbert AM , Harris AR , Helal CJ , Johnson DS , Montgomery JI , Nason DM , Noell S , Pandit J , Rogers BN , Samad TA , Shaffer CL , da Silva RG , Uccello DP , Webb D , Brodney MA |
| Ref : Journal of Medicinal Chemistry , 61 :3008 , 2018 |
| Abstract : |
| PubMedSearch : McAllister_2018_J.Med.Chem_61_3008 |
| PubMedID: 29498843 |
| Gene_locus related to this paper: human-MGLL |
| Title : Azetidine and Piperidine Carbamates as Efficient, Covalent Inhibitors of Monoacylglycerol Lipase - Butler_2017_J.Med.Chem_60_9860 |
| Author(s) : Butler CR , Beck EM , Harris A , Huang Z , McAllister LA , Am Ende CW , Fennell K , Foley TL , Fonseca K , Hawrylik SJ , Johnson DS , Knafels JD , Mente S , Noell GS , Pandit J , Phillips TB , Piro JR , Rogers BN , Samad TA , Wang J , Wan S , Brodney MA |
| Ref : Journal of Medicinal Chemistry , 60 :9860 , 2017 |
| Abstract : |
| PubMedSearch : Butler_2017_J.Med.Chem_60_9860 |
| PubMedID: 29148769 |
| Gene_locus related to this paper: human-MGLL |
| Title : Molecular medicine and neurodegenerative diseases - |
| Author(s) : Chang CJ , Cravatt BF , Johnson DS , Lim MH |
| Ref : Chem Soc Rev , 43 :6668 , 2014 |
| PubMedID: 25105517 |
| Title : O-hydroxyacetamide carbamates as a highly potent and selective class of endocannabinoid hydrolase inhibitors - Niphakis_2012_ACS.Chem.Neurosci_3_418 |
| Author(s) : Niphakis MJ , Johnson DS , Ballard TE , Stiff C , Cravatt BF |
| Ref : ACS Chem Neurosci , 3 :418 , 2012 |
| Abstract : |
| PubMedSearch : Niphakis_2012_ACS.Chem.Neurosci_3_418 |
| PubMedID: 22860211 |
| Gene_locus related to this paper: human-MGLL |
| Title : Discovery of PF-04457845: A Highly Potent, Orally Bioavailable, and Selective Urea FAAH Inhibitor - Johnson_2011_ACS.Med.Chem.Lett_2_91 |
| Author(s) : Johnson DS , Stiff C , Lazerwith SE , Kesten SR , Fay LK , Morris M , Beidler D , Liimatta MB , Smith SE , Dudley DT , Sadagopan N , Bhattachar SN , Kesten SJ , Nomanbhoy TK , Cravatt BF , Ahn K |
| Ref : ACS Med Chem Lett , 2 :91 , 2011 |
| Abstract : |
| PubMedSearch : Johnson_2011_ACS.Med.Chem.Lett_2_91 |
| PubMedID: 21666860 |
| Title : alpha-Conotoxin ImI exhibits subtype-specific nicotinic acetylcholine receptor blockade: preferential inhibition of homomeric alpha 7 and alpha 9 receptors - Johnson_1995_Mol.Pharmacol_48_194 |
| Author(s) : Johnson DS , Martinez J , Elgoyhen AB , Heinemann SF , McIntosh JM |
| Ref : Molecular Pharmacology , 48 :194 , 1995 |
| Abstract : |
| PubMedSearch : Johnson_1995_Mol.Pharmacol_48_194 |
| PubMedID: 7651351 |
| Title : Alpha 9: an acetylcholine receptor with novel pharmacological properties expressed in rat cochlear hair cells - Elgoyhen_1994_Cell_79_705 |
| Author(s) : Elgoyhen AB , Johnson DS , Boulter J , Vetter DE , Heinemann S |
| Ref : Cell , 79 :705 , 1994 |
| Abstract : |
| PubMedSearch : Elgoyhen_1994_Cell_79_705 |
| PubMedID: 7954834 |