Title : Radiosynthesis and evaluation of novel (18)F labeled PET ligands for imaging monoacylglycerol lipase - Li_2025_Eur.J.Med.Chem_285_117246 |
Author(s) : Li Y , Mori W , Chaudhary A , Zhao C , Yamasaki T , Zhang Z , Feng S , Ware T , Rong J , Fujinaga M , Chen J , Kumata K , Zhang Y , Hu K , Xie L , Zhou X , Song Z , Gao Y , Sun Z , Patel JS , Zhai C , Yuan KY , Collier TL , Ran C , Collin L , Haider A , Grether U , Wittwer MB , Cravatt BF , Zhang MR , Liang SH |
Ref : Eur Journal of Medicinal Chemistry , 285 :117246 , 2025 |
Abstract : |
PubMedSearch : Li_2025_Eur.J.Med.Chem_285_117246 |
PubMedID: 39793441 |
Gene_locus related to this paper: human-MGLL |
Title : A novel monoacylglycerol lipase-targeted (18)F-labeled probe for positron emission tomography imaging of brown adipose tissue in the energy network - Cheng_2022_Acta.Pharmacol.Sin__ |
Author(s) : Cheng R , Fujinaga M , Yang J , Rong J , Haider A , Ogasawara D , Van RS , Shao T , Chen Z , Zhang X , Calderon Leon ER , Zhang Y , Mori W , Kumata K , Yamasaki T , Xie L , Sun S , Wang L , Ran C , Shao Y , Cravatt B , Josephson L , Zhang MR , Liang SH |
Ref : Acta Pharmacol Sin , : , 2022 |
Abstract : |
PubMedSearch : Cheng_2022_Acta.Pharmacol.Sin__ |
PubMedID: 35513432 |
Gene_locus related to this paper: human-MGLL |
Title : Novel Reversible-Binding PET Ligands for Imaging Monoacylglycerol Lipase Based on the Piperazinyl Azetidine Scaffold - Rong_2021_J.Med.Chem__ |
Author(s) : Rong J , Mori W , Xia X , Schafroth MA , Zhao C , Van RS , Yamasaki T , Chen J , Xiao Z , Haider A , Ogasawara D , Hiraishi A , Shao T , Zhang Y , Chen Z , Pang F , Hu K , Xie L , Fujinaga M , Kumata K , Gou Y , Fang Y , Gu S , Wei H , Bao L , Xu H , Collier TL , Shao Y , Carson RE , Cravatt BF , Wang L , Zhang MR , Liang SH |
Ref : Journal of Medicinal Chemistry , : , 2021 |
Abstract : |
PubMedSearch : Rong_2021_J.Med.Chem__ |
PubMedID: 34569803 |
Gene_locus related to this paper: human-MGLL |
Title : Design, Synthesis, and Evaluation of Reversible and Irreversible Monoacylglycerol Lipase Positron Emission Tomography (PET) Tracers Using a Tail Switching Strategy on a Piperazinyl Azetidine Skeleton - Chen_2019_J.Med.Chem_62_3336 |
Author(s) : Chen Z , Mori W , Deng X , Cheng R , Ogasawara D , Zhang G , Schafroth MA , Dahl K , Fu H , Hatori A , Shao T , Zhang Y , Yamasaki T , Zhang X , Rong J , Yu Q , Hu K , Fujinaga M , Xie L , Kumata K , Gou Y , Chen J , Gu S , Bao L , Wang L , Collier TL , Vasdev N , Shao Y , Ma JA , Cravatt BF , Fowler C , Josephson L , Zhang MR , Liang SH |
Ref : Journal of Medicinal Chemistry , 62 :3336 , 2019 |
Abstract : |
PubMedSearch : Chen_2019_J.Med.Chem_62_3336 |
PubMedID: 30829483 |
Gene_locus related to this paper: human-MGLL |
Title : Radiosynthesis and evaluation of a novel monoacylglycerol lipase radiotracer: 1,1,1,3,3,3-hexafluoropropan-2-yl-3-(1-benzyl-1H-pyrazol-3-yl)azetidine-1-[(11)C]carboxylate - Mori_2019_Bioorg.Med.Chem_27_3568 |
Author(s) : Mori W , Hatori A , Zhang Y , Kurihara Y , Yamasaki T , Xie L , Kumata K , Hu K , Fujinaga M , Zhang MR |
Ref : Bioorganic & Medicinal Chemistry , 27 :3568 , 2019 |
Abstract : |
PubMedSearch : Mori_2019_Bioorg.Med.Chem_27_3568 |
PubMedID: 31278005 |
Title : In Vitro and in Vivo Evaluation of (11)C-Labeled Azetidinecarboxylates for Imaging Monoacylglycerol Lipase by PET Imaging Studies - Cheng_2018_J.Med.Chem_61_2278 |
Author(s) : Cheng R , Mori W , Ma L , Alhouayek M , Hatori A , Zhang Y , Ogasawara D , Yuan G , Chen Z , Zhang X , Shi H , Yamasaki T , Xie L , Kumata K , Fujinaga M , Nagai Y , Minamimoto T , Svensson M , Wang L , Du Y , Ondrechen MJ , Vasdev N , Cravatt BF , Fowler C , Zhang MR , Liang SH |
Ref : Journal of Medicinal Chemistry , 61 :2278 , 2018 |
Abstract : |
PubMedSearch : Cheng_2018_J.Med.Chem_61_2278 |
PubMedID: 29481079 |