Haider A

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PubMedSearch : Rong_2025_Acta.Pharm.Sin.B_15_6714
PubMedID: 41477323
Gene_locus related to this paper: human-MGLL

Title : Tritium-Labeled Compounds in PET Tracer Discovery? A Case Study from Roche's Internal Monoacylglycerol Lipase Program - Edelmann_2025_ACS.Chem.Neurosci__
Author(s) : Edelmann MR , Gobbi LC , Schmalzbauer S , Beck J , Muller MC , Hau JC , Huber S , Haider A , Wittwer MB , Pavlovic A , Collin L , Heer D , Topp A , Leibrock-Thielen L , Benz J , Hilbert M , Honer M , Grether U
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PubMedSearch : Edelmann_2025_ACS.Chem.Neurosci__
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Title : Expediting hit-to-lead progression in drug discovery through reaction prediction and multi-dimensional optimization - Nippa_2025_Nat.Commun__
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Title : Development of a novel (18)F-labeled reversible-binding radioligand for imaging monoacylglycerol lipase with positron emission tomography - Rong_2025_Acta.Pharm.Sin.B_15_6714
Author(s) : Rong J , Zhao C , Chaudhary AF , Ware T , Van RS , Li Y , Calderon Leon ER , Dang V , Chen J , Xiao Z , Zhou X , Zhang W , Bi C , Zhang K , Patel JS , Shao Y , Ran C , Collin L , Haider A , Cravatt BF , Liang SH
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PubMedSearch : Rong_2025_Acta.Pharm.Sin.B_15_6714
PubMedID: 41477323
Gene_locus related to this paper: human-MGLL

Title : Tritium-Labeled Compounds in PET Tracer Discovery? A Case Study from Roche's Internal Monoacylglycerol Lipase Program - Edelmann_2025_ACS.Chem.Neurosci__
Author(s) : Edelmann MR , Gobbi LC , Schmalzbauer S , Beck J , Muller MC , Hau JC , Huber S , Haider A , Wittwer MB , Pavlovic A , Collin L , Heer D , Topp A , Leibrock-Thielen L , Benz J , Hilbert M , Honer M , Grether U
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Title : Radiosynthesis and evaluation of novel (18)F labeled PET ligands for imaging monoacylglycerol lipase - Li_2025_Eur.J.Med.Chem_285_117246
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Gene_locus related to this paper: human-MGLL

Title : Expediting hit-to-lead progression in drug discovery through reaction prediction and multi-dimensional optimization - Nippa_2025_Nat.Commun__
Author(s) : Nippa DF , Atz K , Stenzhorn Y , Muller AT , Tosstorff A , Benz J , Binch H , Burkler M , Haider A , Heer D , Hochstrasser R , Kramer C , Reutlinger M , Schneider P , Shema T , Topp A , Walter A , Wittwer MB , Wolfard J , Kuhn B , van der Stelt M , Martin RE , Grether U , Schneider G
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Gene_locus related to this paper: human-MGLL

Title : Radiosynthesis and evaluation of novel (18)F labeled PET ligands for imaging monoacylglycerol lipase - Li_2025_Eur.J.Med.Chem_285_117246
Author(s) : Li Y , Mori W , Chaudhary A , Zhao C , Yamasaki T , Zhang Z , Feng S , Ware T , Rong J , Fujinaga M , Chen J , Kumata K , Zhang Y , Hu K , Xie L , Zhou X , Song Z , Gao Y , Sun Z , Patel JS , Zhai C , Yuan KY , Collier TL , Ran C , Collin L , Haider A , Grether U , Wittwer MB , Cravatt BF , Zhang MR , Liang SH
Ref : Eur Journal of Medicinal Chemistry , 285 :117246 , 2025
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PubMedSearch : Li_2025_Eur.J.Med.Chem_285_117246
PubMedID: 39793441
Gene_locus related to this paper: human-MGLL

Title : Development of a novel (18)F-labeled reversible-binding radioligand for imaging monoacylglycerol lipase with positron emission tomography - Rong_2025_Acta.Pharm.Sin.B_15_6714
Author(s) : Rong J , Zhao C , Chaudhary AF , Ware T , Van RS , Li Y , Calderon Leon ER , Dang V , Chen J , Xiao Z , Zhou X , Zhang W , Bi C , Zhang K , Patel JS , Shao Y , Ran C , Collin L , Haider A , Cravatt BF , Liang SH
Ref : Acta Pharm Sin B , 15 :6714 , 2025
Abstract :
PubMedSearch : Rong_2025_Acta.Pharm.Sin.B_15_6714
PubMedID: 41477323
Gene_locus related to this paper: human-MGLL

Title : Tritium-Labeled Compounds in PET Tracer Discovery? A Case Study from Roche's Internal Monoacylglycerol Lipase Program - Edelmann_2025_ACS.Chem.Neurosci__
Author(s) : Edelmann MR , Gobbi LC , Schmalzbauer S , Beck J , Muller MC , Hau JC , Huber S , Haider A , Wittwer MB , Pavlovic A , Collin L , Heer D , Topp A , Leibrock-Thielen L , Benz J , Hilbert M , Honer M , Grether U
Ref : ACS Chem Neurosci , : , 2025
Abstract :
PubMedSearch : Edelmann_2025_ACS.Chem.Neurosci__
PubMedID: 40968094

Title : Expediting hit-to-lead progression in drug discovery through reaction prediction and multi-dimensional optimization - Nippa_2025_Nat.Commun__
Author(s) : Nippa DF , Atz K , Stenzhorn Y , Muller AT , Tosstorff A , Benz J , Binch H , Burkler M , Haider A , Heer D , Hochstrasser R , Kramer C , Reutlinger M , Schneider P , Shema T , Topp A , Walter A , Wittwer MB , Wolfard J , Kuhn B , van der Stelt M , Martin RE , Grether U , Schneider G
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Abstract :
PubMedSearch : Nippa_2025_Nat.Commun__
PubMedID: 41290653
Gene_locus related to this paper: human-MGLL

Title : Radiosynthesis and evaluation of novel (18)F labeled PET ligands for imaging monoacylglycerol lipase - Li_2025_Eur.J.Med.Chem_285_117246
Author(s) : Li Y , Mori W , Chaudhary A , Zhao C , Yamasaki T , Zhang Z , Feng S , Ware T , Rong J , Fujinaga M , Chen J , Kumata K , Zhang Y , Hu K , Xie L , Zhou X , Song Z , Gao Y , Sun Z , Patel JS , Zhai C , Yuan KY , Collier TL , Ran C , Collin L , Haider A , Grether U , Wittwer MB , Cravatt BF , Zhang MR , Liang SH
Ref : Eur Journal of Medicinal Chemistry , 285 :117246 , 2025
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PubMedSearch : Li_2025_Eur.J.Med.Chem_285_117246
PubMedID: 39793441
Gene_locus related to this paper: human-MGLL

Title : Enhancing Drug Discovery and Development through the Integration of Medicinal Chemistry, Chemical Biology, and Academia-Industry Partnerships: Insights from Roche's Endocannabinoid System Projects - Aebi_2024_Chimia.(Aarau)_78_499
Author(s) : Aebi J , Atz K , Ametamey SM , Benz J , Blaising J , Butini S , Campiani G , Carreira EM , Collin L , De Lago E , Gazzi T , Gertsch J , Gobbi L , Guba W , Fernandez-Ruiz J , Fingerle J , Haider A , He Y , Heitman LH , Honer M , Hunziker D , Kuhn B , Maccarrone M , Marki HP , Martin RE , Mohr P , Mu L , Nazare M , Nippa DF , Oddi S , O'Hara F , Pacher P , Romero J , Rover S , Rufer AC , Schibli R , Schneider G , Stepan AF , Sykes DA , Ullmer C , van der Stelt M , Veprintsev DB , Wittwer MB , Grether U
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PubMedSearch : Aebi_2024_Chimia.(Aarau)_78_499
PubMedID: 39221845

Title : Enhancing Drug Discovery and Development through the Integration of Medicinal Chemistry, Chemical Biology, and Academia-Industry Partnerships: Insights from Roche's Endocannabinoid System Projects - Aebi_2024_Chimia.(Aarau)_78_499
Author(s) : Aebi J , Atz K , Ametamey SM , Benz J , Blaising J , Butini S , Campiani G , Carreira EM , Collin L , De Lago E , Gazzi T , Gertsch J , Gobbi L , Guba W , Fernandez-Ruiz J , Fingerle J , Haider A , He Y , Heitman LH , Honer M , Hunziker D , Kuhn B , Maccarrone M , Marki HP , Martin RE , Mohr P , Mu L , Nazare M , Nippa DF , Oddi S , O'Hara F , Pacher P , Romero J , Rover S , Rufer AC , Schibli R , Schneider G , Stepan AF , Sykes DA , Ullmer C , van der Stelt M , Veprintsev DB , Wittwer MB , Grether U
Ref : Chimia (Aarau) , 78 :499 , 2024
Abstract :
PubMedSearch : Aebi_2024_Chimia.(Aarau)_78_499
PubMedID: 39221845

Title : Enhancing Drug Discovery and Development through the Integration of Medicinal Chemistry, Chemical Biology, and Academia-Industry Partnerships: Insights from Roche's Endocannabinoid System Projects - Aebi_2024_Chimia.(Aarau)_78_499
Author(s) : Aebi J , Atz K , Ametamey SM , Benz J , Blaising J , Butini S , Campiani G , Carreira EM , Collin L , De Lago E , Gazzi T , Gertsch J , Gobbi L , Guba W , Fernandez-Ruiz J , Fingerle J , Haider A , He Y , Heitman LH , Honer M , Hunziker D , Kuhn B , Maccarrone M , Marki HP , Martin RE , Mohr P , Mu L , Nazare M , Nippa DF , Oddi S , O'Hara F , Pacher P , Romero J , Rover S , Rufer AC , Schibli R , Schneider G , Stepan AF , Sykes DA , Ullmer C , van der Stelt M , Veprintsev DB , Wittwer MB , Grether U
Ref : Chimia (Aarau) , 78 :499 , 2024
Abstract :
PubMedSearch : Aebi_2024_Chimia.(Aarau)_78_499
PubMedID: 39221845

Title : Synthesis, Structural Elucidation and Pharmacological Applications of Cu(II) Heteroleptic Carboxylates - Ullah_2023_Pharmaceuticals.(Basel)_16_
Author(s) : Ullah S , Sirajuddin M , Ullah Z , Mushtaq A , Naz S , Zubair M , Haider A , Ali S , Kubicki M , Wani TA , Zargar S , Rehman MU
Ref : Pharmaceuticals (Basel) , 16 : , 2023
Abstract :
PubMedSearch : Ullah_2023_Pharmaceuticals.(Basel)_16_
PubMedID: 37242476

Title : Synthesis, Structural Elucidation and Pharmacological Applications of Cu(II) Heteroleptic Carboxylates - Ullah_2023_Pharmaceuticals.(Basel)_16_
Author(s) : Ullah S , Sirajuddin M , Ullah Z , Mushtaq A , Naz S , Zubair M , Haider A , Ali S , Kubicki M , Wani TA , Zargar S , Rehman MU
Ref : Pharmaceuticals (Basel) , 16 : , 2023
Abstract :
PubMedSearch : Ullah_2023_Pharmaceuticals.(Basel)_16_
PubMedID: 37242476

Title : Synthesis, Structural Elucidation and Pharmacological Applications of Cu(II) Heteroleptic Carboxylates - Ullah_2023_Pharmaceuticals.(Basel)_16_
Author(s) : Ullah S , Sirajuddin M , Ullah Z , Mushtaq A , Naz S , Zubair M , Haider A , Ali S , Kubicki M , Wani TA , Zargar S , Rehman MU
Ref : Pharmaceuticals (Basel) , 16 : , 2023
Abstract :
PubMedSearch : Ullah_2023_Pharmaceuticals.(Basel)_16_
PubMedID: 37242476

Title : A novel monoacylglycerol lipase-targeted (18)F-labeled probe for positron emission tomography imaging of brown adipose tissue in the energy network - Cheng_2022_Acta.Pharmacol.Sin__
Author(s) : Cheng R , Fujinaga M , Yang J , Rong J , Haider A , Ogasawara D , Van RS , Shao T , Chen Z , Zhang X , Calderon Leon ER , Zhang Y , Mori W , Kumata K , Yamasaki T , Xie L , Sun S , Wang L , Ran C , Shao Y , Cravatt B , Josephson L , Zhang MR , Liang SH
Ref : Acta Pharmacol Sin , : , 2022
Abstract :
PubMedSearch : Cheng_2022_Acta.Pharmacol.Sin__
PubMedID: 35513432
Gene_locus related to this paper: human-MGLL

Title : A novel monoacylglycerol lipase-targeted (18)F-labeled probe for positron emission tomography imaging of brown adipose tissue in the energy network - Cheng_2022_Acta.Pharmacol.Sin__
Author(s) : Cheng R , Fujinaga M , Yang J , Rong J , Haider A , Ogasawara D , Van RS , Shao T , Chen Z , Zhang X , Calderon Leon ER , Zhang Y , Mori W , Kumata K , Yamasaki T , Xie L , Sun S , Wang L , Ran C , Shao Y , Cravatt B , Josephson L , Zhang MR , Liang SH
Ref : Acta Pharmacol Sin , : , 2022
Abstract :
PubMedSearch : Cheng_2022_Acta.Pharmacol.Sin__
PubMedID: 35513432
Gene_locus related to this paper: human-MGLL

Title : A novel monoacylglycerol lipase-targeted (18)F-labeled probe for positron emission tomography imaging of brown adipose tissue in the energy network - Cheng_2022_Acta.Pharmacol.Sin__
Author(s) : Cheng R , Fujinaga M , Yang J , Rong J , Haider A , Ogasawara D , Van RS , Shao T , Chen Z , Zhang X , Calderon Leon ER , Zhang Y , Mori W , Kumata K , Yamasaki T , Xie L , Sun S , Wang L , Ran C , Shao Y , Cravatt B , Josephson L , Zhang MR , Liang SH
Ref : Acta Pharmacol Sin , : , 2022
Abstract :
PubMedSearch : Cheng_2022_Acta.Pharmacol.Sin__
PubMedID: 35513432
Gene_locus related to this paper: human-MGLL

Title : Novel Reversible-Binding PET Ligands for Imaging Monoacylglycerol Lipase Based on the Piperazinyl Azetidine Scaffold - Rong_2021_J.Med.Chem__
Author(s) : Rong J , Mori W , Xia X , Schafroth MA , Zhao C , Van RS , Yamasaki T , Chen J , Xiao Z , Haider A , Ogasawara D , Hiraishi A , Shao T , Zhang Y , Chen Z , Pang F , Hu K , Xie L , Fujinaga M , Kumata K , Gou Y , Fang Y , Gu S , Wei H , Bao L , Xu H , Collier TL , Shao Y , Carson RE , Cravatt BF , Wang L , Zhang MR , Liang SH
Ref : Journal of Medicinal Chemistry , : , 2021
Abstract :
PubMedSearch : Rong_2021_J.Med.Chem__
PubMedID: 34569803
Gene_locus related to this paper: human-MGLL

Title : Prospective Application of Two New Pyridine-Based Zinc (II) Amide Carboxylate in Management of Alzheimer's Disease: Synthesis, Characterization, Computational and in vitro Approaches - Zafar_2021_Drug.Des.Devel.Ther_15_2679
Author(s) : Zafar R , Naureen H , Zubair M , Shahid K , Saeed Jan M , Akhtar S , Ahmad H , Waseem W , Haider A , Ali S , Tariq M , Sadiq A
Ref : Drug Des Devel Ther , 15 :2679 , 2021
Abstract :
PubMedSearch : Zafar_2021_Drug.Des.Devel.Ther_15_2679
PubMedID: 34188447

Title : Positron Emission Tomography Imaging of the Endocannabinoid System: Opportunities and Challenges in Radiotracer Development - Hou_2021_J.Med.Chem_64_123
Author(s) : Hou L , Rong J , Haider A , Ogasawara D , Varlow C , Schafroth MA , Mu L , Gan J , Xu H , Fowler CJ , Zhang MR , Vasdev N , Ametamey S , Cravatt BF , Wang L , Liang SH
Ref : Journal of Medicinal Chemistry , 64 :123 , 2021
Abstract :
PubMedSearch : Hou_2021_J.Med.Chem_64_123
PubMedID: 33379862

Title : Positron Emission Tomography Imaging of the Endocannabinoid System: Opportunities and Challenges in Radiotracer Development - Hou_2021_J.Med.Chem_64_123
Author(s) : Hou L , Rong J , Haider A , Ogasawara D , Varlow C , Schafroth MA , Mu L , Gan J , Xu H , Fowler CJ , Zhang MR , Vasdev N , Ametamey S , Cravatt BF , Wang L , Liang SH
Ref : Journal of Medicinal Chemistry , 64 :123 , 2021
Abstract :
PubMedSearch : Hou_2021_J.Med.Chem_64_123
PubMedID: 33379862

Title : Prospective Application of Two New Pyridine-Based Zinc (II) Amide Carboxylate in Management of Alzheimer's Disease: Synthesis, Characterization, Computational and in vitro Approaches - Zafar_2021_Drug.Des.Devel.Ther_15_2679
Author(s) : Zafar R , Naureen H , Zubair M , Shahid K , Saeed Jan M , Akhtar S , Ahmad H , Waseem W , Haider A , Ali S , Tariq M , Sadiq A
Ref : Drug Des Devel Ther , 15 :2679 , 2021
Abstract :
PubMedSearch : Zafar_2021_Drug.Des.Devel.Ther_15_2679
PubMedID: 34188447

Title : Novel Reversible-Binding PET Ligands for Imaging Monoacylglycerol Lipase Based on the Piperazinyl Azetidine Scaffold - Rong_2021_J.Med.Chem__
Author(s) : Rong J , Mori W , Xia X , Schafroth MA , Zhao C , Van RS , Yamasaki T , Chen J , Xiao Z , Haider A , Ogasawara D , Hiraishi A , Shao T , Zhang Y , Chen Z , Pang F , Hu K , Xie L , Fujinaga M , Kumata K , Gou Y , Fang Y , Gu S , Wei H , Bao L , Xu H , Collier TL , Shao Y , Carson RE , Cravatt BF , Wang L , Zhang MR , Liang SH
Ref : Journal of Medicinal Chemistry , : , 2021
Abstract :
PubMedSearch : Rong_2021_J.Med.Chem__
PubMedID: 34569803
Gene_locus related to this paper: human-MGLL

Title : Positron Emission Tomography Imaging of the Endocannabinoid System: Opportunities and Challenges in Radiotracer Development - Hou_2021_J.Med.Chem_64_123
Author(s) : Hou L , Rong J , Haider A , Ogasawara D , Varlow C , Schafroth MA , Mu L , Gan J , Xu H , Fowler CJ , Zhang MR , Vasdev N , Ametamey S , Cravatt BF , Wang L , Liang SH
Ref : Journal of Medicinal Chemistry , 64 :123 , 2021
Abstract :
PubMedSearch : Hou_2021_J.Med.Chem_64_123
PubMedID: 33379862

Title : Novel Reversible-Binding PET Ligands for Imaging Monoacylglycerol Lipase Based on the Piperazinyl Azetidine Scaffold - Rong_2021_J.Med.Chem__
Author(s) : Rong J , Mori W , Xia X , Schafroth MA , Zhao C , Van RS , Yamasaki T , Chen J , Xiao Z , Haider A , Ogasawara D , Hiraishi A , Shao T , Zhang Y , Chen Z , Pang F , Hu K , Xie L , Fujinaga M , Kumata K , Gou Y , Fang Y , Gu S , Wei H , Bao L , Xu H , Collier TL , Shao Y , Carson RE , Cravatt BF , Wang L , Zhang MR , Liang SH
Ref : Journal of Medicinal Chemistry , : , 2021
Abstract :
PubMedSearch : Rong_2021_J.Med.Chem__
PubMedID: 34569803
Gene_locus related to this paper: human-MGLL

Title : Prospective Application of Two New Pyridine-Based Zinc (II) Amide Carboxylate in Management of Alzheimer's Disease: Synthesis, Characterization, Computational and in vitro Approaches - Zafar_2021_Drug.Des.Devel.Ther_15_2679
Author(s) : Zafar R , Naureen H , Zubair M , Shahid K , Saeed Jan M , Akhtar S , Ahmad H , Waseem W , Haider A , Ali S , Tariq M , Sadiq A
Ref : Drug Des Devel Ther , 15 :2679 , 2021
Abstract :
PubMedSearch : Zafar_2021_Drug.Des.Devel.Ther_15_2679
PubMedID: 34188447

Title : Zinc metal carboxylates as Potential anti-Alzheimer's candidate: In-vitro anticholinesterase, antioxidant and molecular docking studies - Zafar_2020_J.Biomol.Struct.Dyn__1
Author(s) : Zafar R , Zubair M , Ali S , Shahid K , Waseem W , Naureen H , Haider A , Saeed Jan M , Ullah F , Sirajuddin M , Sadiq A
Ref : J Biomol Struct Dyn , :1 , 2020
Abstract :
PubMedSearch : Zafar_2020_J.Biomol.Struct.Dyn__1
PubMedID: 32013770

Title : Zinc metal carboxylates as Potential anti-Alzheimer's candidate: In-vitro anticholinesterase, antioxidant and molecular docking studies - Zafar_2020_J.Biomol.Struct.Dyn__1
Author(s) : Zafar R , Zubair M , Ali S , Shahid K , Waseem W , Naureen H , Haider A , Saeed Jan M , Ullah F , Sirajuddin M , Sadiq A
Ref : J Biomol Struct Dyn , :1 , 2020
Abstract :
PubMedSearch : Zafar_2020_J.Biomol.Struct.Dyn__1
PubMedID: 32013770

Title : Zinc metal carboxylates as Potential anti-Alzheimer's candidate: In-vitro anticholinesterase, antioxidant and molecular docking studies - Zafar_2020_J.Biomol.Struct.Dyn__1
Author(s) : Zafar R , Zubair M , Ali S , Shahid K , Waseem W , Naureen H , Haider A , Saeed Jan M , Ullah F , Sirajuddin M , Sadiq A
Ref : J Biomol Struct Dyn , :1 , 2020
Abstract :
PubMedSearch : Zafar_2020_J.Biomol.Struct.Dyn__1
PubMedID: 32013770

Title : beta-glucan attenuated scopolamine induced cognitive impairment via hippocampal acetylcholinesterase inhibition in rats - Haider_2016_Brain.Res_1644_141
Author(s) : Haider A , Inam W , Khan SA , Hifza , Mahmood W , Abbas G
Ref : Brain Research , 1644 :141 , 2016
Abstract :
PubMedSearch : Haider_2016_Brain.Res_1644_141
PubMedID: 27180103

Title : beta-glucan attenuated scopolamine induced cognitive impairment via hippocampal acetylcholinesterase inhibition in rats - Haider_2016_Brain.Res_1644_141
Author(s) : Haider A , Inam W , Khan SA , Hifza , Mahmood W , Abbas G
Ref : Brain Research , 1644 :141 , 2016
Abstract :
PubMedSearch : Haider_2016_Brain.Res_1644_141
PubMedID: 27180103

Title : beta-glucan attenuated scopolamine induced cognitive impairment via hippocampal acetylcholinesterase inhibition in rats - Haider_2016_Brain.Res_1644_141
Author(s) : Haider A , Inam W , Khan SA , Hifza , Mahmood W , Abbas G
Ref : Brain Research , 1644 :141 , 2016
Abstract :
PubMedSearch : Haider_2016_Brain.Res_1644_141
PubMedID: 27180103