Report for Alptuzun V

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References (16)

Title : Novel multifunctional tacrine-donepezil hybrids against Alzheimer's disease: Design synthesis and bioactivity studies - Bayraktar_2024_Arch.Pharm.(Weinheim)__e2300575
Author(s) : Bayraktar G , Bartolini M , Bolognesi ML , Erdogan MA , Armagan G , Bayir E , Sendemir A , Bagetta D , Alcaro S , Alptuzun V
Ref : Arch Pharm (Weinheim) , :e2300575 , 2024
Abstract : Bayraktar_2024_Arch.Pharm.(Weinheim)__e2300575
ESTHER : Bayraktar_2024_Arch.Pharm.(Weinheim)__e2300575
PubMedSearch : Bayraktar_2024_Arch.Pharm.(Weinheim)__e2300575
PubMedID: 38593283

Title : N-Substituted piperidine-3-carbohydrazide-hydrazones against Alzheimer's disease: Synthesis and evaluation of cholinesterase, beta-amyloid inhibitory activity, and antioxidant capacity - Parlar_2022_Arch.Pharm.(Weinheim)__e2200519
Author(s) : Parlar S , Sayar G , Tarikogullari AH , Karadagli SS , Alan E , Sevin G , Erciyas E , Holzgrabe U , Alptuzun V
Ref : Arch Pharm (Weinheim) , :e2200519 , 2022
Abstract : Parlar_2022_Arch.Pharm.(Weinheim)__e2200519
ESTHER : Parlar_2022_Arch.Pharm.(Weinheim)__e2200519
PubMedSearch : Parlar_2022_Arch.Pharm.(Weinheim)__e2200519
PubMedID: 36461719

Title : Design, synthesis, acetylcholinesterase, butyrylcholinesterase, and amyloid-beta aggregation inhibition studies of substituted 4,4'-diimine\/4,4'-diazobiphenyl derivatives - Fidan_2022_Arch.Pharm.(Weinheim)__e2200152
Author(s) : Fidan GS , Parlar S , Tarikogullari AH , Alptuzun V , Alpan AS
Ref : Arch Pharm (Weinheim) , :e2200152 , 2022
Abstract : Fidan_2022_Arch.Pharm.(Weinheim)__e2200152
ESTHER : Fidan_2022_Arch.Pharm.(Weinheim)__e2200152
PubMedSearch : Fidan_2022_Arch.Pharm.(Weinheim)__e2200152
PubMedID: 35976708

Title : Synthesis, bioactivity and molecular modeling studies on potential anti-Alzheimer piperidinehydrazide-hydrazones - Parlar_2019_Bioorg.Chem_87_888
Author(s) : Parlar S , Sayar G , Tarikogullari AH , Karadagli SS , Alptuzun V , Erciyas E , Holzgrabe U
Ref : Bioorg Chem , 87 :888 , 2019
Abstract : Parlar_2019_Bioorg.Chem_87_888
ESTHER : Parlar_2019_Bioorg.Chem_87_888
PubMedSearch : Parlar_2019_Bioorg.Chem_87_888
PubMedID: 30538051

Title : Synthesis, biological evaluation, and docking studies of some 5-chloro-2(3H)-benzoxazolone Mannich bases derivatives as cholinesterase inhibitors - Uysal_2018_Arch.Pharm.(Weinheim)_351_e1700273
Author(s) : Uysal S , Parlar S , Tarikogullari AH , Aydin Kose F , Alptuzun V , Soyer Z
Ref : Arch Pharm (Weinheim) , 351 :e1700273 , 2018
Abstract : Uysal_2018_Arch.Pharm.(Weinheim)_351_e1700273
ESTHER : Uysal_2018_Arch.Pharm.(Weinheim)_351_e1700273
PubMedSearch : Uysal_2018_Arch.Pharm.(Weinheim)_351_e1700273
PubMedID: 29527733

Title : Multifunctional cholinesterase inhibitors for Alzheimer's disease: Synthesis, biological evaluations, and docking studies of o\/p-propoxyphenylsubstituted-1H-benzimidazole derivatives - Sarikaya_2018_Arch.Pharm.(Weinheim)__
Author(s) : Sarikaya G , Coban G , Parlar S , Tarikogullari AH , Armagan G , Erdogan MA , Alptuzun V , Alpan AS
Ref : Arch Pharm (Weinheim) , : , 2018
Abstract : Sarikaya_2018_Arch.Pharm.(Weinheim)__
ESTHER : Sarikaya_2018_Arch.Pharm.(Weinheim)__
PubMedSearch : Sarikaya_2018_Arch.Pharm.(Weinheim)__
PubMedID: 29984517

Title : Synthesis and molecular docking studies of some 4-phthalimidobenzenesulfonamide derivatives as acetylcholinesterase and butyrylcholinesterase inhibitors - Soyer_2017_J.Enzyme.Inhib.Med.Chem_32_13
Author(s) : Soyer Z , Uysal S , Parlar S , Tarikogullari Dogan AH , Alptuzun V
Ref : J Enzyme Inhib Med Chem , 32 :13 , 2017
Abstract : Soyer_2017_J.Enzyme.Inhib.Med.Chem_32_13
ESTHER : Soyer_2017_J.Enzyme.Inhib.Med.Chem_32_13
PubMedSearch : Soyer_2017_J.Enzyme.Inhib.Med.Chem_32_13
PubMedID: 27766908

Title : Mannich-Benzimidazole Derivatives as Antioxidant and Anticholinesterase Inhibitors: Synthesis, Biological Evaluations, and Molecular Docking Study - Alpan_2017_Arch.Pharm.(Weinheim)_350_
Author(s) : Alpan AS , Sarikaya G , Coban G , Parlar S , Armagan G , Alptuzun V
Ref : Arch Pharm (Weinheim) , 350 : , 2017
Abstract : Alpan_2017_Arch.Pharm.(Weinheim)_350_
ESTHER : Alpan_2017_Arch.Pharm.(Weinheim)_350_
PubMedSearch : Alpan_2017_Arch.Pharm.(Weinheim)_350_
PubMedID: 28379621

Title : Synthesis, Biological Evaluation and Molecular Docking Study of Hydrazone-Containing Pyridinium Salts as Cholinesterase Inhibitors - Parlar_2016_Chem.Pharm.Bull.(Tokyo)_64_1281
Author(s) : Parlar S , Bayraktar G , Tarikogullari AH , Alptuzun V , Erciyas E
Ref : Chem Pharm Bull (Tokyo) , 64 :1281 , 2016
Abstract : Parlar_2016_Chem.Pharm.Bull.(Tokyo)_64_1281
ESTHER : Parlar_2016_Chem.Pharm.Bull.(Tokyo)_64_1281
PubMedSearch : Parlar_2016_Chem.Pharm.Bull.(Tokyo)_64_1281
PubMedID: 27581632

Title : Synthesis, biological activity and molecular modeling studies on 1H-benzimidazole derivatives as acetylcholinesterase inhibitors - Alpan_2013_Bioorg.Med.Chem_21_4928
Author(s) : Alpan AS , Parlar S , Carlino L , Tarikogullari AH , Alptuzun V , Gunes HS
Ref : Bioorganic & Medicinal Chemistry , 21 :4928 , 2013
Abstract : Alpan_2013_Bioorg.Med.Chem_21_4928
ESTHER : Alpan_2013_Bioorg.Med.Chem_21_4928
PubMedSearch : Alpan_2013_Bioorg.Med.Chem_21_4928
PubMedID: 23891231

Title : 1,4-Substituted 4-(1H)-pyridylene-hydrazone-type inhibitors of AChE, BCHE, and amyloid-beta aggregation crossing the blood-brain barrier - Prinz_2013_Eur.J.Pharm.Sci_49_603
Author(s) : Prinz M , Parlar S , Bayraktar G , Alptuzun V , Erciyas E , Fallarero A , Karlsson D , Vuorela P , Burek M , Forster C , Turunc E , Armagan G , Yalcin A , Schiller C , Leuner K , Krug M , Sotriffer CA , Holzgrabe U
Ref : Eur J Pharm Sci , 49 :603 , 2013
Abstract : Prinz_2013_Eur.J.Pharm.Sci_49_603
ESTHER : Prinz_2013_Eur.J.Pharm.Sci_49_603
PubMedSearch : Prinz_2013_Eur.J.Pharm.Sci_49_603
PubMedID: 23643737

Title : Interaction of (benzylidene-hydrazono)-1,4-dihydropyridines with beta-amyloid, acetylcholine, and butyrylcholine esterases - Alptuzun_2010_Bioorg.Med.Chem_18_2049
Author(s) : Alptuzun V , Prinz M , Horr V , Scheiber J , Radacki K , Fallarero A , Vuorela P , Engels B , Braunschweig H , Erciyas E , Holzgrabe U
Ref : Bioorganic & Medicinal Chemistry , 18 :2049 , 2010
Abstract : Alptuzun_2010_Bioorg.Med.Chem_18_2049
ESTHER : Alptuzun_2010_Bioorg.Med.Chem_18_2049
PubMedSearch : Alptuzun_2010_Bioorg.Med.Chem_18_2049
PubMedID: 20149667

Title : Targeting acetylcholinesterase to treat neurodegeneration - Holzgrabe_2007_Expert.Opin.Ther.Targets_11_161
Author(s) : Holzgrabe U , Kapkova P , Alptuzun V , Scheiber J , Kugelmann E
Ref : Expert Opin Ther Targets , 11 :161 , 2007
Abstract : Holzgrabe_2007_Expert.Opin.Ther.Targets_11_161
ESTHER : Holzgrabe_2007_Expert.Opin.Ther.Targets_11_161
PubMedSearch : Holzgrabe_2007_Expert.Opin.Ther.Targets_11_161
PubMedID: 17227232

Title : Search for dual function inhibitors for Alzheimer's disease: synthesis and biological activity of acetylcholinesterase inhibitors of pyridinium-type and their Abeta fibril formation inhibition capacity - Kapkova_2006_Bioorg.Med.Chem_14_472
Author(s) : Kapkova P , Alptuzun V , Frey P , Erciyas E , Holzgrabe U
Ref : Bioorganic & Medicinal Chemistry , 14 :472 , 2006
Abstract : Kapkova_2006_Bioorg.Med.Chem_14_472
ESTHER : Kapkova_2006_Bioorg.Med.Chem_14_472
PubMedSearch : Kapkova_2006_Bioorg.Med.Chem_14_472
PubMedID: 16198581

Title : Cooperative interactions at M2 muscarinic acetylcholine receptors: structure\/activity relationships in stepwise shortened bispyridinium- and bis(ammonio)alkane-type allosteric modulators - Gilsbach_2003_Neurochem.Res_28_667
Author(s) : Gilsbach R , Grossmuller M , Alptuzun V , Erciyas E , Trankle C , Holzgrabe U , Mohr K
Ref : Neurochem Res , 28 :667 , 2003
Abstract : Gilsbach_2003_Neurochem.Res_28_667
ESTHER : Gilsbach_2003_Neurochem.Res_28_667
PubMedSearch : Gilsbach_2003_Neurochem.Res_28_667
PubMedID: 12675159

Title : Synthesis and biological activity of pyridinium-type acetylcholinesterase inhibitors - Alptuzun_2003_J.Pharm.Pharmacol_55_1397
Author(s) : Alptuzun V , Kapkova P , Baumann K , Erciyas E , Holzgrabe U
Ref : J Pharm Pharmacol , 55 :1397 , 2003
Abstract : Alptuzun_2003_J.Pharm.Pharmacol_55_1397
ESTHER : Alptuzun_2003_J.Pharm.Pharmacol_55_1397
PubMedSearch : Alptuzun_2003_J.Pharm.Pharmacol_55_1397
PubMedID: 14607022