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Title : Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors - Di Stefano_2023_Eur.J.Med.Chem_263_115916 |
Author(s) : Di Stefano M , Masoni S , Bononi G , Poli G , Galati S , Gado F , Manzi S , Vagaggini C , Brai A , Caligiuri I , Asif K , Rizzolio F , Macchia M , Chicca A , Sodi A , Di Bussolo V , Minutolo F , Meier P , Gertsch J , Granchi C , Dreassi E , Tuccinardi T |
Ref : Eur Journal of Medicinal Chemistry , 263 :115916 , 2023 |
Abstract : Di Stefano_2023_Eur.J.Med.Chem_263_115916 |
ESTHER : Di Stefano_2023_Eur.J.Med.Chem_263_115916 |
PubMedSearch : Di Stefano_2023_Eur.J.Med.Chem_263_115916 |
PubMedID: 37976705 |
Title : Reversible Monoacylglycerol Lipase Inhibitors: Discovery of a New Class of Benzylpiperidine Derivatives - Bononi_2022_J.Med.Chem__ |
Author(s) : Bononi G , Di Stefano M , Poli G , Ortore G , Meier P , Masetto F , Caligiuri I , Rizzolio F , Macchia M , Chicca A , Avan A , Giovannetti E , Vagaggini C , Brai A , Dreassi E , Valoti M , Minutolo F , Granchi C , Gertsch J , Tuccinardi T |
Ref : Journal of Medicinal Chemistry , : , 2022 |
Abstract : Bononi_2022_J.Med.Chem__ |
ESTHER : Bononi_2022_J.Med.Chem__ |
PubMedSearch : Bononi_2022_J.Med.Chem__ |
PubMedID: 35522977 |