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Title : Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors - Di Stefano_2023_Eur.J.Med.Chem_263_115916 |
Author(s) : Di Stefano M , Masoni S , Bononi G , Poli G , Galati S , Gado F , Manzi S , Vagaggini C , Brai A , Caligiuri I , Asif K , Rizzolio F , Macchia M , Chicca A , Sodi A , Di Bussolo V , Minutolo F , Meier P , Gertsch J , Granchi C , Dreassi E , Tuccinardi T |
Ref : Eur Journal of Medicinal Chemistry , 263 :115916 , 2023 |
Abstract : Di Stefano_2023_Eur.J.Med.Chem_263_115916 |
ESTHER : Di Stefano_2023_Eur.J.Med.Chem_263_115916 |
PubMedSearch : Di Stefano_2023_Eur.J.Med.Chem_263_115916 |
PubMedID: 37976705 |
Title : Modification on the 1,2-dihydro-2-oxo-pyridine-3-carboxamide core to obtain multi-target modulators of endocannabinoid system - Gado_2019_Bioorg.Chem__103353 |
Author(s) : Gado F , Arena C , Fauci C , Reynoso-Moreno I , Bertini S , Digiacomo M , Meini S , Poli G , Macchia M , Tuccinardi T , Gertsch J , Chicca A , Manera C |
Ref : Bioorg Chem , :103353 , 2019 |
Abstract : Gado_2019_Bioorg.Chem__103353 |
ESTHER : Gado_2019_Bioorg.Chem__103353 |
PubMedSearch : Gado_2019_Bioorg.Chem__103353 |
PubMedID: 31668465 |
Title : Polypharmacological profile of 1,2-dihydro-2-oxo-pyridine-3-carboxamides in the endocannabinoid system - Chicca_2018_Eur.J.Med.Chem_154_155 |
Author(s) : Chicca A , Arena C , Bertini S , Gado F , Ciaglia E , Abate M , Digiacomo M , Lapillo M , Poli G , Bifulco M , Macchia M , Tuccinardi T , Gertsch J , Manera C |
Ref : Eur Journal of Medicinal Chemistry , 154 :155 , 2018 |
Abstract : Chicca_2018_Eur.J.Med.Chem_154_155 |
ESTHER : Chicca_2018_Eur.J.Med.Chem_154_155 |
PubMedSearch : Chicca_2018_Eur.J.Med.Chem_154_155 |
PubMedID: 29793210 |