Title : Galantamine-memantine hybrids for Alzheimer's disease: The influence of linker rigidity in biological activity and pharmacokinetic properties - Basagni_2023_Eur.J.Med.Chem_261_115803 |
Author(s) : Basagni F , Ortega JA , Bertozzi SM , Armirotti A , Summa M , Bertorelli R , Bartolini M , Mellor IR , Bedeschi M , Bottegoni G , Lembo V , Minarini A , Cavalli A , Rosini M |
Ref : Eur Journal of Medicinal Chemistry , 261 :115803 , 2023 |
Abstract : |
PubMedSearch : Basagni_2023_Eur.J.Med.Chem_261_115803 |
PubMedID: 37734258 |
Title : Lid domain plasticity and lipid flexibility modulate enzyme specificity in human monoacylglycerol lipase - Riccardi_2017_Biochim.Biophys.Acta_1862_441 |
Author(s) : Riccardi L , Arencibia JM , Bono L , Armirotti A , Girotto S , De Vivo M |
Ref : Biochimica & Biophysica Acta , 1862 :441 , 2017 |
Abstract : |
PubMedSearch : Riccardi_2017_Biochim.Biophys.Acta_1862_441 |
PubMedID: 28088576 |
Title : Development and Pharmacological Characterization of Selective Blockers of 2-Arachidonoyl Glycerol Degradation with Efficacy in Rodent Models of Multiple Sclerosis and Pain - Brindisi_2016_J.Med.Chem_59_2612 |
Author(s) : Brindisi M , Maramai S , Gemma S , Brogi S , Grillo A , Di Cesare Mannelli L , Gabellieri E , Lamponi S , Saponara S , Gorelli B , Tedesco D , Bonfiglio T , Landry C , Jung KM , Armirotti A , Luongo L , Ligresti A , Piscitelli F , Bertucci C , Dehouck MP , Campiani G , Maione S , Ghelardini C , Pittaluga A , Piomelli D , Di Marzo V , Butini S |
Ref : Journal of Medicinal Chemistry , 59 :2612 , 2016 |
Abstract : |
PubMedSearch : Brindisi_2016_J.Med.Chem_59_2612 |
PubMedID: 26888301 |
Title : Keys to Lipid Selection in Fatty Acid Amide Hydrolase Catalysis: Structural Flexibility, Gating Residues and Multiple Binding Pockets - Palermo_2015_PLoS.Comput.Biol_11_e1004231 |
Author(s) : Palermo G , Bauer I , Campomanes P , Cavalli A , Armirotti A , Girotto S , Rothlisberger U , De Vivo M |
Ref : PLoS Comput Biol , 11 :e1004231 , 2015 |
Abstract : |
PubMedSearch : Palermo_2015_PLoS.Comput.Biol_11_e1004231 |
PubMedID: 26111155 |