| Title : Novel Dual-Acting Hybrids Targeting Type-2 Cannabinoid Receptors and Cholinesterase Activity Show Neuroprotective Effects In Vitro and Amelioration of Cognitive Impairment In Vivo - Mugnaini_2024_ACS.Chem.Neurosci__ |
| Author(s) : Mugnaini C , Brizzi A , Paolino M , Scarselli E , Castelli R , de Candia M , Gambacorta N , Nicolotti O , Kostrzewa M , Kumar P , Mahmoud AM , Borgonetti V , Iannotta M , Morace A , Galeotti N , Maione S , Altomare CD , Ligresti A , Corelli F |
| Ref : ACS Chem Neurosci , : , 2024 |
| Abstract : |
| PubMedSearch : Mugnaini_2024_ACS.Chem.Neurosci__ |
| PubMedID: 38372253 |
| Title : Identification of Cannabidiolic and Cannabigerolic Acids as MTDL AChE, BuChE, and BACE-1 Inhibitors Against Alzheimer's Disease by In Silico, In Vitro, and In Vivo Studies - Vitale_2024_Phytother.Res__ |
| Author(s) : Vitale RM , Morace AM , D'Errico A , Ricciardi F , Fusco A , Boccella S , Guida F , Nasso R , Rading S , Karsak M , Caprioglio D , Iannotti FA , Arcone R , Luongo L , Masullo M , Maione S , Amodeo P |
| Ref : Phytother Res , : , 2024 |
| Abstract : |
| PubMedSearch : Vitale_2024_Phytother.Res__ |
| PubMedID: 39510547 |
| Title : Development and Pharmacological Characterization of Selective Blockers of 2-Arachidonoyl Glycerol Degradation with Efficacy in Rodent Models of Multiple Sclerosis and Pain - Brindisi_2016_J.Med.Chem_59_2612 |
| Author(s) : Brindisi M , Maramai S , Gemma S , Brogi S , Grillo A , Di Cesare Mannelli L , Gabellieri E , Lamponi S , Saponara S , Gorelli B , Tedesco D , Bonfiglio T , Landry C , Jung KM , Armirotti A , Luongo L , Ligresti A , Piscitelli F , Bertucci C , Dehouck MP , Campiani G , Maione S , Ghelardini C , Pittaluga A , Piomelli D , Di Marzo V , Butini S |
| Ref : Journal of Medicinal Chemistry , 59 :2612 , 2016 |
| Abstract : |
| PubMedSearch : Brindisi_2016_J.Med.Chem_59_2612 |
| PubMedID: 26888301 |
| Title : Genetic deletion of monoacylglycerol lipase leads to impaired cannabinoid receptor CB1 R signaling and anxiety-like behavior - Imperatore_2015_J.Neurochem_135_799 |
| Author(s) : Imperatore R , Morello G , Luongo L , Taschler U , Romano R , De Gregorio D , Belardo C , Maione S , Di Marzo V , Cristino L |
| Ref : Journal of Neurochemistry , 135 :799 , 2015 |
| Abstract : |
| PubMedSearch : Imperatore_2015_J.Neurochem_135_799 |
| PubMedID: 26223500 |
| Title : Development of a potent inhibitor of 2-arachidonoylglycerol hydrolysis with antinociceptive activity in vivo - Bisogno_2009_Biochim.Biophys.Acta_1791_53 |
| Author(s) : Bisogno T , Ortar G , Petrosino S , Morera E , Palazzo E , Nalli M , Maione S , Di Marzo V |
| Ref : Biochimica & Biophysica Acta , 1791 :53 , 2009 |
| Abstract : |
| PubMedSearch : Bisogno_2009_Biochim.Biophys.Acta_1791_53 |
| PubMedID: 19027877 |
| Gene_locus related to this paper: human-DAGLA , human-DAGLB |
| Title : Antinociceptive effects of tetrazole inhibitors of endocannabinoid inactivation: cannabinoid and non-cannabinoid receptor-mediated mechanisms - Maione_2008_Br.J.Pharmacol_155_775 |
| Author(s) : Maione S , Morera E , Marabese I , Ligresti A , Luongo L , Ortar G , Di Marzo V |
| Ref : British Journal of Pharmacology , 155 :775 , 2008 |
| Abstract : |
| PubMedSearch : Maione_2008_Br.J.Pharmacol_155_775 |
| PubMedID: 18660824 |