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| Title : Novel 6-alkyl-bridged 4-arylalkylpiperazin-1-yl derivatives of azepino[4,3-b]indol-1(2H)-one as potent BChE-selective inhibitors showing protective effects against neurodegenerative insults - Samarelli_2024_Eur.J.Med.Chem_270_116353 |
| Author(s) : Samarelli F , Purgatorio R , Lopopolo G , Deruvo C , Catto M , Andresini M , Carrieri A , Nicolotti O , De Palma A , Miniero DV , de Candia M , Altomare CD |
| Ref : Eur Journal of Medicinal Chemistry , 270 :116353 , 2024 |
| Abstract : Samarelli_2024_Eur.J.Med.Chem_270_116353 |
| ESTHER : Samarelli_2024_Eur.J.Med.Chem_270_116353 |
| PubMedSearch : Samarelli_2024_Eur.J.Med.Chem_270_116353 |
| PubMedID: 38579622 |
| Title : Synthesis, computational and experimental pharmacological studies for (thio)ether-triazine 5-HT(6)R ligands with noticeable action on AChE\/BChE and chalcogen-dependent intrinsic activity in search for new class of drugs against Alzheimer's disease - Czarnota-Lydka_2023_Eur.J.Med.Chem_259_115695 |
| Author(s) : Czarnota-Lydka K , Sudol-Talaj S , Kucwaj-Brysz K , Kurczab R , Satala G , de Candia M , Samarelli F , Altomare CD , Carocci A , Barbarossa A , eslawska E , Gluch-Lutwin M , Mordyl B , Kubacka M , Wilczynska-Zawal N , Jastrzebska-Wiesek M , Partyka A , Khan N , Wiecek M , Nitek W , Honkisz-Orzechowska E , Latacz G , Wesolowska A , Carrieri A , Handzlik J |
| Ref : Eur Journal of Medicinal Chemistry , 259 :115695 , 2023 |
| Abstract : Czarnota-Lydka_2023_Eur.J.Med.Chem_259_115695 |
| ESTHER : Czarnota-Lydka_2023_Eur.J.Med.Chem_259_115695 |
| PubMedSearch : Czarnota-Lydka_2023_Eur.J.Med.Chem_259_115695 |
| PubMedID: 37567058 |
| Title : A twenty-year journey exploring coumarin-based derivatives as bioactive molecules - Pisani_2022_Front.Chem_10_1002547 |
| Author(s) : Pisani L , Catto M , Muncipinto G , Nicolotti O , Carrieri A , Rullo M , Stefanachi A , Leonetti F , Altomare CD |
| Ref : Front Chem , 10 :1002547 , 2022 |
| Abstract : Pisani_2022_Front.Chem_10_1002547 |
| ESTHER : Pisani_2022_Front.Chem_10_1002547 |
| PubMedSearch : Pisani_2022_Front.Chem_10_1002547 |
| PubMedID: 36300022 |
| Title : Novel Phenothiazine\/Donepezil-like Hybrids Endowed with Antioxidant Activity for a Multi-Target Approach to the Therapy of Alzheimer's Disease - Carocci_2022_Antioxidants.(Basel)_11_ |
| Author(s) : Carocci A , Barbarossa A , Leuci R , Carrieri A , Brunetti L , Laghezza A , Catto M , Limongelli F , Chaves S , Tortorella P , Altomare CD , Santos MA , Loiodice F , Piemontese L |
| Ref : Antioxidants (Basel) , 11 : , 2022 |
| Abstract : Carocci_2022_Antioxidants.(Basel)_11_ |
| ESTHER : Carocci_2022_Antioxidants.(Basel)_11_ |
| PubMedSearch : Carocci_2022_Antioxidants.(Basel)_11_ |
| PubMedID: 36139705 |
| Title : Structure-based design of novel donepezil-like hybrids for a multi-target approach to the therapy of Alzheimer's disease - Brunetti_2022_Eur.J.Med.Chem_237_114358 |
| Author(s) : Brunetti L , Leuci R , Carrieri A , Catto M , Occhineri S , Vinci G , Gambacorta L , Baltrukevich H , Chaves S , Laghezza A , Altomare CD , Tortorella P , Santos MA , Loiodice F , Piemontese L |
| Ref : Eur Journal of Medicinal Chemistry , 237 :114358 , 2022 |
| Abstract : Brunetti_2022_Eur.J.Med.Chem_237_114358 |
| ESTHER : Brunetti_2022_Eur.J.Med.Chem_237_114358 |
| PubMedSearch : Brunetti_2022_Eur.J.Med.Chem_237_114358 |
| PubMedID: 35462163 |
| Title : A New Series of Aryloxyacetic Acids Endowed with Multi-Target Activity towards Peroxisome Proliferator-Activated Receptors (PPARs), Fatty Acid Amide Hydrolase (FAAH), and Acetylcholinesterase (AChE) - Leuci_2022_Molecules_27_ |
| Author(s) : Leuci R , Brunetti L , Laghezza A , Piemontese L , Carrieri A , Pisani L , Tortorella P , Catto M , Loiodice F |
| Ref : Molecules , 27 : , 2022 |
| Abstract : Leuci_2022_Molecules_27_ |
| ESTHER : Leuci_2022_Molecules_27_ |
| PubMedSearch : Leuci_2022_Molecules_27_ |
| PubMedID: 35164223 |
| Title : Derivatives of Tenuazonic Acid as Potential New Multi-Target Anti-Alzheimer's Disease Agents - Poliseno_2021_Biomolecules_11_ |
| Author(s) : Poliseno V , Chaves S , Brunetti L , Loiodice F , Carrieri A , Laghezza A , Tortorella P , Magalhaes JD , Cardoso SM , Santos MA , Piemontese L |
| Ref : Biomolecules , 11 : , 2021 |
| Abstract : Poliseno_2021_Biomolecules_11_ |
| ESTHER : Poliseno_2021_Biomolecules_11_ |
| PubMedSearch : Poliseno_2021_Biomolecules_11_ |
| PubMedID: 33467709 |
| Title : Evaluation of water-soluble Mannich base prodrugs of 2,3,4,5-tetrahydroazepino[4,3-b]indol-1(6H)-one as multitarget-directed agents for Alzheimer's disease - Purgatorio_2021_ChemMedChem_16_589 |
| Author(s) : Purgatorio R , de Candia M , Catto M , Rullo M , Pisani L , Denora N , Carrieri A , Nevskaya AA , Voskressensky LG , Altomare CD |
| Ref : ChemMedChem , 16 :589 , 2021 |
| Abstract : Purgatorio_2021_ChemMedChem_16_589 |
| ESTHER : Purgatorio_2021_ChemMedChem_16_589 |
| PubMedSearch : Purgatorio_2021_ChemMedChem_16_589 |
| PubMedID: 33156950 |
| Title : Scouting around 1,2,3,4-Tetrahydrochromeno[3,2-c]pyridin-10-ones for Single- and Multi-target Ligands Directed towards Relevant Alzheimer's Targets - Purgatorio_2020_ChemMedChem_15_1947 |
| Author(s) : Purgatorio R , Kulikova L , Pisani L , Catto M , de Candia M , Carrieri A , Cellamare S , De Palma A , Beloglazkin A , Raesi GR , Voskressensky L , Altomare CD |
| Ref : ChemMedChem , 15 :1947 , 2020 |
| Abstract : Purgatorio_2020_ChemMedChem_15_1947 |
| ESTHER : Purgatorio_2020_ChemMedChem_15_1947 |
| PubMedSearch : Purgatorio_2020_ChemMedChem_15_1947 |
| PubMedID: 32716595 |
| Title : Investigating 1,2,3,4,5,6-hexahydroazepino[4,3-b]indole as scaffold of butyrylcholinesterase-selective inhibitors with additional neuroprotective activities for Alzheimer's disease - Purgatorio_2019_Eur.J.Med.Chem_177_414 |
| Author(s) : Purgatorio R , de Candia M , Catto M , Carrieri A , Pisani L , De Palma A , Toma M , Ivanova OA , Voskressensky LG , Altomare CD |
| Ref : Eur Journal of Medicinal Chemistry , 177 :414 , 2019 |
| Abstract : Purgatorio_2019_Eur.J.Med.Chem_177_414 |
| ESTHER : Purgatorio_2019_Eur.J.Med.Chem_177_414 |
| PubMedSearch : Purgatorio_2019_Eur.J.Med.Chem_177_414 |
| PubMedID: 31158754 |
| Title : Chasing ChEs-MAO B Multi-Targeting 4-Aminomethyl-7-Benzyloxy-2H-Chromen-2-ones - Rullo_2019_Molecules_24_ |
| Author(s) : Rullo M , Catto M , Carrieri A , de Candia M , Altomare CD , Pisani L |
| Ref : Molecules , 24 : , 2019 |
| Abstract : Rullo_2019_Molecules_24_ |
| ESTHER : Rullo_2019_Molecules_24_ |
| PubMedSearch : Rullo_2019_Molecules_24_ |
| PubMedID: 31835376 |