Full name : Bosak Anita
First name : Anita
Mail : Institute for Medical Research and Occupational Health\; Ksaverska cesta 2\; HR-10000 Zagreb
Zip Code :
City :
Country : Croatia
Email : abosak@imi.hr
Phone : +38514673188 +38514682551
Fax :
Website :
Directory :
Comment
| Title : Synthesis and biological evaluation of novel aminoquinolines with an n-octyl linker: Impact of halogen substituents on C(7) or a terminal amino group on anticholinesterase and BACE1 activity - Matosevic_2024_Bioorg.Med.Chem.Lett__129928 |
| Author(s) : Matosevic A , Bartolic M , Marakovic N , Zandona A , Petric R , Opsenica D , Bosak A |
| Ref : Bioorganic & Medicinal Chemistry Lett , :129928 , 2024 |
| Abstract : |
| PubMedSearch : Matosevic_2024_Bioorg.Med.Chem.Lett__129928 |
| PubMedID: 39151660 |
| Title : Evaluation of 4-aminoquinoline derivatives with an n-octylamino spacer as potential multi-targeting ligands for the treatment of Alzheimer's disease - Matosevic_2023_Chem.Biol.Interact_14ChEPon_382_110620 |
| Author(s) : Matosevic A , Opsenica DM , Spasic M , Marakovic N , Zandona A , Zunec S , Bartolic M , Kovarik Z , Bosak A |
| Ref : Chemico-Biological Interactions , 382 :110620 , 2023 |
| Abstract : |
| PubMedSearch : Matosevic_2023_Chem.Biol.Interact_14ChEPon_382_110620 |
| PubMedID: 37406982 |
| Title : Design, Synthesis and Biological Evaluation of Biscarbamates as Potential Selective Butyrylcholinesterase Inhibitors for the Treatment of Alzheimer's Disease - Matosevic_2022_Pharmaceuticals.(Basel)_15_ |
| Author(s) : Matosevic A , Knezevic A , Zandona A , Marakovic N , Kovarik Z , Bosak A |
| Ref : Pharmaceuticals (Basel) , 15 : , 2022 |
| Abstract : |
| PubMedSearch : Matosevic_2022_Pharmaceuticals.(Basel)_15_ |
| PubMedID: 36297332 |
| Title : Synthesis, Biological Evaluation and Machine Learning Prediction Model for Fluorinated Cinchona Alkaloid-Based Derivatives as Cholinesterase Inhibitors - Ramic_2022_Pharmaceuticals.(Basel)_15_ |
| Author(s) : Ramic A , Matosevic A , Debanic B , Mikelic A , Primozic I , Bosak A , Hrenar T |
| Ref : Pharmaceuticals (Basel) , 15 : , 2022 |
| Abstract : |
| PubMedSearch : Ramic_2022_Pharmaceuticals.(Basel)_15_ |
| PubMedID: 36297327 |
| Title : 4-Aminoquinoline-Based Adamantanes as Potential Anticholinesterase Agents in Symptomatic Treatment of Alzheimer's Disease - Komatovic_2022_Pharmaceutics_14_ |
| Author(s) : Komatovic K , Matosevic A , Terzic-Jovanovic N , Zunec S , Segan S , Zlatovic M , Marakovic N , Bosak A , Opsenica DM |
| Ref : Pharmaceutics , 14 : , 2022 |
| Abstract : |
| PubMedSearch : Komatovic_2022_Pharmaceutics_14_ |
| PubMedID: 35745878 |
| Title : Quinuclidine-Based Carbamates as Potential CNS Active Compounds - Matosevic_2021_Pharmaceutics_13_ |
| Author(s) : Matosevic A , Radman Kastelic A , Mikelic A , Zandona A , Katalinic M , Primozic I , Bosak A , Hrenar T |
| Ref : Pharmaceutics , 13 : , 2021 |
| Abstract : |
| PubMedSearch : Matosevic_2021_Pharmaceutics_13_ |
| PubMedID: 33804719 |
| Title : Structural isomers of saligenin-based beta2-agonists: synthesis and insight into the reaction mechanism - Knezevic_2020_Org.Biomol.Chem_18_9675 |
| Author(s) : Knezevic A , Novak J , Bosak A , Vinkovic M |
| Ref : Org Biomol Chem , 18 :9675 , 2020 |
| Abstract : |
| PubMedSearch : Knezevic_2020_Org.Biomol.Chem_18_9675 |
| PubMedID: 33220672 |
| Title : Carbamate group as structural motif in drugs: a review of carbamate derivatives used as therapeutic agents - Matosevic_2020_Arh.Hig.Rada.Toksikol_71_285 |
| Author(s) : Matosevic A , Bosak A |
| Ref : Arh Hig Rada Toksikol , 71 :285 , 2020 |
| Abstract : |
| PubMedSearch : Matosevic_2020_Arh.Hig.Rada.Toksikol_71_285 |
| PubMedID: 33410773 |
| Title : Interactions of Paraoxonase-1 with Pharmacologically Relevant Carbamates - Bosak_2020_Molecules_25_ |
| Author(s) : Bosak A , Bavec A , Konte T , Sinko G , Kovarik Z , Golicnik M |
| Ref : Molecules , 25 : , 2020 |
| Abstract : |
| PubMedSearch : Bosak_2020_Molecules_25_ |
| PubMedID: 31947900 |
| Title : Structural aspects of 4-aminoquinolines as reversible inhibitors of human acetylcholinesterase and butyrylcholinesterase - Bosak_2019_Chem.Biol.Interact_13ChEPon_308_101 |
| Author(s) : Bosak A , Opsenica DM , Sinko G , Zlatar M , Kovarik Z |
| Ref : Chemico-Biological Interactions , 308 :101 , 2019 |
| Abstract : |
| PubMedSearch : Bosak_2019_Chem.Biol.Interact_13ChEPon_308_101 |
| PubMedID: 31100281 |
| Title : Design and evaluation of selective butyrylcholinesterase inhibitors based on Cinchona alkaloid scaffold - Bosak_2018_PLoS.One_13_e0205193 |
| Author(s) : Bosak A , Ramic A , Smidlehner T , Hrenar T , Primozic I , Kovarik Z |
| Ref : PLoS ONE , 13 :e0205193 , 2018 |
| Abstract : |
| PubMedSearch : Bosak_2018_PLoS.One_13_e0205193 |
| PubMedID: 30289893 |
| Title : Oxime-assisted reactivation of tabun-inhibited acetylcholinesterase analysed by active site mutations - Katalinic_2018_Toxicology_406-407_104 |
| Author(s) : Katalinic M , Sinko G , Macek Hrvat N , Zorbaz T , Bosak A , Kovarik Z |
| Ref : Toxicology , 406-407 :104 , 2018 |
| Abstract : |
| PubMedSearch : Katalinic_2018_Toxicology_406-407_104 |
| PubMedID: 29772260 |
| Title : Resorcinol-, catechol- and saligenin-based bronchodilating beta2-agonists as inhibitors of human cholinesterase activity - Bosak_2017_J.Enzyme.Inhib.Med.Chem_32_789 |
| Author(s) : Bosak A , Knezevic A , Gazic Smilovic I , Sinko G , Kovarik Z |
| Ref : J Enzyme Inhib Med Chem , 32 :789 , 2017 |
| Abstract : |
| PubMedSearch : Bosak_2017_J.Enzyme.Inhib.Med.Chem_32_789 |
| PubMedID: 28573890 |
| Title : Peripheral site and acyl pocket define selective inhibition of mouse butyrylcholinesterase by two biscarbamates - Bosak_2013_Arch.Biochem.Biophys_529_140 |
| Author(s) : Bosak A , Smilovic IG , Stimac A , Vinkovic V , Sinko G , Kovarik Z |
| Ref : Archives of Biochemistry & Biophysics , 529 :140 , 2013 |
| Abstract : |
| PubMedSearch : Bosak_2013_Arch.Biochem.Biophys_529_140 |
| PubMedID: 23219600 |
| Title : Metaproterenol, isoproterenol, and their bisdimethylcarbamate derivatives as human cholinesterase inhibitors - Bosak_2012_J.Med.Chem_55_6716 |
| Author(s) : Bosak A , Gazic Smilovic I , Sinko G , Vinkovic V , Kovarik Z |
| Ref : Journal of Medicinal Chemistry , 55 :6716 , 2012 |
| Abstract : |
| PubMedSearch : Bosak_2012_J.Med.Chem_55_6716 |
| PubMedID: 22817559 |
| Title : [Cholinesterases: structure, role, and inhibition] - Bosak_2011_Arh.Hig.Rada.Toksikol_62_175 |
| Author(s) : Bosak A , Katalinic M , Kovarik Z |
| Ref : Arh Hig Rada Toksikol , 62 :175 , 2011 |
| Abstract : |
| PubMedSearch : Bosak_2011_Arh.Hig.Rada.Toksikol_62_175 |
| PubMedID: 21705306 |
| Title : Preparative HPLC separation of bambuterol enantiomers and stereoselective inhibition of human cholinesterases - Gazic_2008_Anal.Bioanal.Chem_385_1513 |
| Author(s) : Gazic I , Bosak A , Sinko G , Vinkovic V , Kovarik Z |
| Ref : Anal Bioanal Chem , 385 :1513 , 2008 |
| Abstract : |
| PubMedSearch : Gazic_2008_Anal.Bioanal.Chem_385_1513 |
| PubMedID: 16865342 |
| Title : Stereoselective inhibition of human, mouse, and horse cholinesterases by bambuterol enantiomers - Bosak_2008_Chem.Biol.Interact_175_192 |
| Author(s) : Bosak A , Gazic I , Vinkovic V , Kovarik Z |
| Ref : Chemico-Biological Interactions , 175 :192 , 2008 |
| Abstract : |
| PubMedSearch : Bosak_2008_Chem.Biol.Interact_175_192 |
| PubMedID: 18582854 |
| Title : Differentiation of EDTA-sensitive from EDTA-insensitive human serum esterases hydrolysing phenylacetate - Bosak_2008_J.Enzyme.Inhib.Med.Chem_23_521 |
| Author(s) : Bosak A , Barlovic-Tusek B , Reiner E |
| Ref : J Enzyme Inhib Med Chem , 23 :521 , 2008 |
| Abstract : |
| PubMedSearch : Bosak_2008_J.Enzyme.Inhib.Med.Chem_23_521 |
| PubMedID: 18665999 |
| Title : Oximes: Reactivators of phosphorylated acetylcholinesterase and antidotes in therapy against tabun poisoning - Kovarik_2008_Chem.Biol.Interact_175_173 |
| Author(s) : Kovarik Z , Calic M , Sinko G , Bosak A , Zunec S , Vrdoljak AL , Radic B |
| Ref : Chemico-Biological Interactions , 175 :173 , 2008 |
| Abstract : |
| PubMedSearch : Kovarik_2008_Chem.Biol.Interact_175_173 |
| PubMedID: 18501341 |
| Title : Interactions of butane, but-2-ene or xylene-like linked bispyridinium para-aldoximes with native and tabun-inhibited human cholinesterases - Calic_2008_Chem.Biol.Interact_175_305 |
| Author(s) : Calic M , Bosak A , Kuca K , Kovarik Z |
| Ref : Chemico-Biological Interactions , 175 :305 , 2008 |
| Abstract : |
| PubMedSearch : Calic_2008_Chem.Biol.Interact_175_305 |
| PubMedID: 18501885 |
| Title : Amino acid residues involved in stereoselective inhibition of cholinesterases with bambuterol - Bosak_2008_Arch.Biochem.Biophys_471_72 |
| Author(s) : Bosak A , Gazic I , Vinkovic V , Kovarik Z |
| Ref : Archives of Biochemistry & Biophysics , 471 :72 , 2008 |
| Abstract : |
| PubMedSearch : Bosak_2008_Arch.Biochem.Biophys_471_72 |
| PubMedID: 18167304 |
| Title : Structure-activity approach in the reactivation of tabun-phosphorylated human acetylcholinesterase with bispyridinium para-aldoximes - Kovarik_2007_Arh.Hig.Rada.Toksikol_58_201 |
| Author(s) : Kovarik Z , Calic M , Sinko G , Bosak A |
| Ref : Arh Hig Rada Toksikol , 58 :201 , 2007 |
| Abstract : |
| PubMedSearch : Kovarik_2007_Arh.Hig.Rada.Toksikol_58_201 |
| PubMedID: 17562604 |
| Title : Limitation of the Ellman method: cholinesterase activity measurement in the presence of oximes - Sinko_2007_Anal.Biochem_370_223 |
| Author(s) : Sinko G , Calic M , Bosak A , Kovarik Z |
| Ref : Analytical Biochemistry , 370 :223 , 2007 |
| Abstract : |
| PubMedSearch : Sinko_2007_Anal.Biochem_370_223 |
| PubMedID: 17716616 |
| Title : [Organophosphorus compounds: classification and enzyme reactions] - Bosak_2006_Arh.Hig.Rada.Toksikol_57_445 |
| Author(s) : Bosak A |
| Ref : Arh Hig Rada Toksikol , 57 :445 , 2006 |
| Abstract : |
| PubMedSearch : Bosak_2006_Arh.Hig.Rada.Toksikol_57_445 |
| PubMedID: 17265684 |
| Title : Preparation of enantiomers of quinuclidin-3-Ol derivatives and their interactions with human cholinesterases - |
| Author(s) : Simeon-Rudolf V , Tomic S , Bosak A , Primozic I , Orsulic M |
| Ref : Chemico-Biological Interactions , 157-158 :420 , 2005 |
| PubMedID: 16429567 |
| Title : Structure-inhibition relationships in the interaction of butyrylcholinesterase with bambuterol, haloxon and their leaving groups - |
| Author(s) : Sinko G , Bosak A , Kovarik Z , Simeon-Rudolf V |
| Ref : Chemico-Biological Interactions , 157-158 :421 , 2005 |
| PubMedID: 16429568 |
| Title : Activity of cholinesterases in human whole blood measured with acetylthiocholine as substrate and ethopropazine as selective inhibitor of plasma butyrylcholinesterase - Reiner_2004_Arh.Hig.Rada.Toksikol_55_1 |
| Author(s) : Reiner E , Bosak A , Simeon-Rudolf V |
| Ref : Arh Hig Rada Toksikol , 55 :1 , 2004 |
| Abstract : |
| PubMedSearch : Reiner_2004_Arh.Hig.Rada.Toksikol_55_1 |
| PubMedID: 15137175 |
| Title : Kinetics of ethopropazine binding to butyrylcholinesterase in the absence and presence of acetylthiocholine - |
| Author(s) : Reiner E , Sinko G , Bosak A , Simeon-Rudolf V , Radic Z , Taylor P , Stojan J , Golicnik M |
| Ref : In: Cholinesterases in the Second Millennium: Biomolecular and Pathological Aspects , (Inestrosa NC, Campos EO) P. Universidad Catolica de Chile-FONDAP Biomedicina :187 , 2004 |
| PubMedID: |