| Title : Discovery of reversible monoacylglycerol lipase (MAGL) inhibitors based on ortho-hydroxyanilide scaffold - Bononi_2025_Bioorg.Chem_163_108698 |
| Author(s) : Bononi G , Gado F , Masoni S , Scalabrini D , Vedova LD , Di Stefano M , Piazza L , Poles C , Lonzi C , Landucci E , Vagaggini C , Poggialini F , Brai A , Caligiuri I , Rizzolio F , Mohamed KA , Bertini S , De Lorenzi E , Dreassi E , Macchia M , Minutolo F , Laprairie RB , Granchi C , Tuccinardi T |
| Ref : Bioorg Chem , 163 :108698 , 2025 |
| Abstract : |
| PubMedSearch : Bononi_2025_Bioorg.Chem_163_108698 |
| PubMedID: 40554889 |
| Gene_locus related to this paper: human-MGLL |
| Title : Disease-Modifying Anti-Alzheimer's Drugs: Inhibitors of Human Cholinesterases Interfering with beta-Amyloid Aggregation - Brogi_2014_CNS.Neurosci.Ther_20_624 |
| Author(s) : Brogi S , Butini S , Maramai S , Colombo R , Verga L , Lanni C , De Lorenzi E , Lamponi S , Andreassi M , Bartolini M , Andrisano V , Novellino E , Campiani G , Brindisi M , Gemma S |
| Ref : CNS Neurosci Ther , 20 :624 , 2014 |
| Abstract : |
| PubMedSearch : Brogi_2014_CNS.Neurosci.Ther_20_624 |
| PubMedID: 24935788 |
| Title : Multifunctional cholinesterase and amyloid Beta fibrillization modulators. Synthesis and biological investigation - Butini_2013_ACS.Med.Chem.Lett_4_1178 |
| Author(s) : Butini S , Brindisi M , Brogi S , Maramai S , Guarino E , Panico A , Saxena A , Chauhan V , Colombo R , Verga L , De Lorenzi E , Bartolini M , Andrisano V , Novellino E , Campiani G , Gemma S |
| Ref : ACS Med Chem Lett , 4 :1178 , 2013 |
| Abstract : |
| PubMedSearch : Butini_2013_ACS.Med.Chem.Lett_4_1178 |
| PubMedID: 24900626 |