Gutschow M

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Title : Aminoalkoxy-substituted coumarins: Synthesis and evaluation for reactivation of inhibited human acetylcholinesterase - Elsinghorst_2022_Arch.Pharm.(Weinheim)__e2200208
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Gene_locus related to this paper: human-MGLL

Title : omega-Phthalimidoalkyl Aryl Ureas as Potent and Selective Inhibitors of Cholesterol Esterase - Dato_2018_ChemMedChem_13_1833
Author(s) : Dato FM , Sheikh M , Uhl RZ , Schuller AW , Steinkruger M , Koch P , Neudorfl JM , Gutschow M , Goldfuss B , Pietsch M
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Title : A novel fluorogenic probe for the investigation of free thiols: Application to kinetic measurements of acetylcholinesterase activity - Mertens_2016_Toxicol.Lett_244_161
Author(s) : Mertens MD , Bierwisch A , Li T , Gutschow M , Thiermann H , Wille T , Elsinghorst PW
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Title : New cholesterol esterase inhibitors based on rhodanine and thiazolidinedione scaffolds - Heng_2011_Bioorg.Med.Chem_19_7453
Author(s) : Heng S , Tieu W , Hautmann S , Kuan K , Pedersen DS , Pietsch M , Gutschow M , Abell AD
Ref : Bioorganic & Medicinal Chemistry , 19 :7453 , 2011
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PubMedSearch : Heng_2011_Bioorg.Med.Chem_19_7453
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Title : Hyperbolic mixed-type inhibition of acetylcholinesterase by tetracyclic thienopyrimidines - Tanarro_2011_J.Enzyme.Inhib.Med.Chem_26_350
Author(s) : Tanarro CM , Gutschow M
Ref : J Enzyme Inhib Med Chem , 26 :350 , 2011
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PubMedSearch : Tanarro_2011_J.Enzyme.Inhib.Med.Chem_26_350
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Title : A hydrazide linker strategy for heterobivalent compounds as ortho- and allosteric ligands of acetylcholine-binding proteins - Elsinghorst_2011_Curr.Top.Med.Chem_11_2731
Author(s) : Elsinghorst PW , Hartig W , Gundisch D , Mohr K , Trankle C , Gutschow M
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Author(s) : Hartig W , Kacza J , Paulke BR , Grosche J , Bauer U , Hoffmann A , Elsinghorst PW , Gutschow M
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Title : A gorge-spanning, high-affinity cholinesterase inhibitor to explore beta-amyloid plaques - Elsinghorst_2009_Org.Biomol.Chem_7_3940
Author(s) : Elsinghorst PW , Hartig W , Goldhammer S , Grosche J , Gutschow M
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PubMedSearch : Elsinghorst_2009_Org.Biomol.Chem_7_3940
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Title : Kinetics of inhibition of acetylcholinesterase in the presence of acetonitrile - Pietsch_2009_FEBS.J_276_2292
Author(s) : Pietsch M , Christian L , Inhester T , Petzold S , Gutschow M
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PubMedSearch : Pietsch_2009_FEBS.J_276_2292
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Title : Synthesis and elastase-inhibiting activity of 2-pyridinyl-isothiazol-3(2H)-one 1,1-dioxides - Eilfeld_2008_Bioorg.Med.Chem_16_8127
Author(s) : Eilfeld A , Gonzalez Tanarro CM , Frizler M , Sieler J , Schulze B , Gutschow M
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PubMedSearch : Eilfeld_2008_Bioorg.Med.Chem_16_8127
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Title : First gallamine-tacrine hybrid: design and characterization at cholinesterases and the M2 muscarinic receptor - Elsinghorst_2007_J.Med.Chem_50_5685
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Title : Novel heterobivalent tacrine derivatives as cholinesterase inhibitors with notable selectivity toward butyrylcholinesterase - Elsinghorst_2006_J.Med.Chem_49_7540
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Title : Synthesis of tricyclic 1,3-oxazin-4-ones and kinetic analysis of cholesterol esterase and acetylcholinesterase inhibition - Pietsch_2005_J.Med.Chem_48_8270
Author(s) : Pietsch M , Gutschow M
Ref : Journal of Medicinal Chemistry , 48 :8270 , 2005
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PubMedSearch : Pietsch_2005_J.Med.Chem_48_8270
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Title : Alternate substrate inhibition of cholesterol esterase by thieno[2,3-d][1,3]oxazin-4-ones - Pietsch_2002_J.Biol.Chem_277_24006
Author(s) : Pietsch M , Gutschow M
Ref : Journal of Biological Chemistry , 277 :24006 , 2002
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PubMedSearch : Pietsch_2002_J.Biol.Chem_277_24006
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