| Title : The first-in-class 1,3,5-triazine-derived dual 5-HT(6)R\/FAAH modulators in search for potential drug against neurodegenerative diseases with cognitive impairment - Czarnota-Lydka_2025_Eur.J.Med.Chem_298_118026 |
| Author(s) : Czarnota-Lydka K , Kucwaj-Brysz K , Mordyl B , Gluch-Lutwin M , Karcz T , Jastrzebska-Wiesek M , Partyka A , Dbrowska M , Satala G , Sudol-Talaj S , Brunetti L , de Candia M , Purgatorio R , Cerini M , Piemontese L , Podlewska S , Latacz G , Starek M , Wesolowska A , Carrieri A , Handzlik J |
| Ref : Eur Journal of Medicinal Chemistry , 298 :118026 , 2025 |
| Abstract : |
| PubMedSearch : Czarnota-Lydka_2025_Eur.J.Med.Chem_298_118026 |
| PubMedID: 40774068 |
| Title : Discovery of New Highly Potent Histamine H(3) Receptor Antagonists, Calcium Channel Blockers, and Acetylcholinesterase Inhibitors - Malek_2024_ACS.Chem.Neurosci__ |
| Author(s) : Malek R , Salat K , Totoson P , Karcz T , Refouvelet B , Skrzypczak-Wiercioch A , Maj M , Simakov A , Martin H , Siwek A , Szalaj N , Godyn J , Panek D , Wieckowska A , Jozwiak K , Demougeot C , Kiec-Kononowicz K , Chabchoub F , Iriepa I , Marco-Contelles J , Ismaili L |
| Ref : ACS Chem Neurosci , : , 2024 |
| Abstract : |
| PubMedSearch : Malek_2024_ACS.Chem.Neurosci__ |
| PubMedID: 39208251 |
| Title : 4-Oxypiperidine Ethers as Multiple Targeting Ligands at Histamine H(3) Receptors and Cholinesterases - Michalska_2024_ACS.Chem.Neurosci__ |
| Author(s) : Michalska B , Dziegielewski M , Godyn J , Werner T , Bajda M , Karcz T , Szczepanska K , Stark H , Wieckowska A , Walczynski K , Staszewski M |
| Ref : ACS Chem Neurosci , : , 2024 |
| Abstract : |
| PubMedSearch : Michalska_2024_ACS.Chem.Neurosci__ |
| PubMedID: 38440987 |