| Title : Synthesis and evaluation of lipoic acid - donepezil hybrids for Alzheimer's disease using a straightforward strategy - Luzet_2024_Bioorg.Med.Chem.Lett__129938 |
| Author(s) : Luzet V , Allemand F , Richet C , Dehecq B , Bonet A , Harakat D , Refouvelet B , Martin H , Cardey B , Pudlo M |
| Ref : Bioorganic & Medicinal Chemistry Lett , :129938 , 2024 |
| Abstract : |
| PubMedSearch : Luzet_2024_Bioorg.Med.Chem.Lett__129938 |
| PubMedID: 39222891 |
| Title : Discovery of New Highly Potent Histamine H(3) Receptor Antagonists, Calcium Channel Blockers, and Acetylcholinesterase Inhibitors - Malek_2024_ACS.Chem.Neurosci__ |
| Author(s) : Malek R , Salat K , Totoson P , Karcz T , Refouvelet B , Skrzypczak-Wiercioch A , Maj M , Simakov A , Martin H , Siwek A , Szalaj N , Godyn J , Panek D , Wieckowska A , Jozwiak K , Demougeot C , Kiec-Kononowicz K , Chabchoub F , Iriepa I , Marco-Contelles J , Ismaili L |
| Ref : ACS Chem Neurosci , : , 2024 |
| Abstract : |
| PubMedSearch : Malek_2024_ACS.Chem.Neurosci__ |
| PubMedID: 39208251 |
| Title : Exploring the Potential of Sulfonamide-Dihydropyridine Hybrids as Multitargeted Ligands for Alzheimer's Disease Treatment - Dakhlaoui_2023_Int.J.Mol.Sci_24_ |
| Author(s) : Dakhlaoui I , Bernard PJ , Pietrzak D , Simakov A , Maj M , Refouvelet B , Beduneau A , Cornu R , Jozwiak K , Chabchoub F , Iriepa I , Martin H , Marco-Contelles J , Ismaili L |
| Ref : Int J Mol Sci , 24 : , 2023 |
| Abstract : |
| PubMedSearch : Dakhlaoui_2023_Int.J.Mol.Sci_24_ |
| PubMedID: 37298693 |
| Title : Biginelli Reaction Synthesis of Novel Multitarget-Directed Ligands with Ca(2+) Channel Blocking Ability, Cholinesterase Inhibition, Antioxidant Capacity, and Nrf2 Activation - Malek_2022_Molecules_28_ |
| Author(s) : Malek R , Simakov A , Davis A , Maj M , Bernard PJ , Wnorowski A , Martin H , Marco-Contelles J , Chabchoub F , Dallemagne P , Rochais C , Jozwiak K , Ismaili L |
| Ref : Molecules , 28 : , 2022 |
| Abstract : |
| PubMedSearch : Malek_2022_Molecules_28_ |
| PubMedID: 36615267 |
| Title : Synthesis of new Hantzsch adducts showing Ca(2+) channel blockade capacity, cholinesterase inhibition and antioxidant power - Pachon-Angona_2021_Future.Med.Chem__ |
| Author(s) : Pachon-Angona I , Maj M , Wnorowski A , Martin H , Jozwiak K , Ismaili L |
| Ref : Future Med Chem , : , 2021 |
| Abstract : |
| PubMedSearch : Pachon-Angona_2021_Future.Med.Chem__ |
| PubMedID: 34402661 |
| Title : Synthesis of Hantzsch Adducts as Cholinesterases and Calcium Flux inhibitors, Antioxidants and Neuroprotectives - Pachon_2020_Int.J.Mol.Sci_21_ |
| Author(s) : Pachon Angona I , Martin H , Daniel S , Moraleda I , Bonet A , Wnorowski A , Maj M , Jozwiak K , Iriepa I , Refouvelet B , Marco-Contelles J , Ismaili L |
| Ref : Int J Mol Sci , 21 : , 2020 |
| Abstract : |
| PubMedSearch : Pachon_2020_Int.J.Mol.Sci_21_ |
| PubMedID: 33081112 |
| Title : Synthesis and biological assessment of KojoTacrines as new agents for Alzheimer's disease therapy - Dgachi_2019_J.Enzyme.Inhib.Med.Chem_34_163 |
| Author(s) : Dgachi Y , Martin H , Malek R , Jun D , Janockova J , Sepsova V , Soukup O , Iriepa I , Moraleda I , Maalej E , Carreiras MC , Refouvelet B , Chabchoub F , Marco-Contelles J , Ismaili L |
| Ref : J Enzyme Inhib Med Chem , 34 :163 , 2019 |
| Abstract : |
| PubMedSearch : Dgachi_2019_J.Enzyme.Inhib.Med.Chem_34_163 |
| PubMedID: 30482062 |
| Title : Donepezil + chromone + melatonin hybrids as promising agents for Alzheimer's disease therapy - Pachon-Angona_2019_J.Enzyme.Inhib.Med.Chem_34_479 |
| Author(s) : Pachon-Angona I , Refouvelet B , Andrys R , Martin H , Luzet V , Iriepa I , Moraleda I , Diez-Iriepa D , Oset-Gasque MJ , Marco-Contelles J , Musilek K , Ismaili L |
| Ref : J Enzyme Inhib Med Chem , 34 :479 , 2019 |
| Abstract : |
| PubMedSearch : Pachon-Angona_2019_J.Enzyme.Inhib.Med.Chem_34_479 |
| PubMedID: 30712420 |
| Title : New (benz)imidazolopyridino tacrines as nonhepatotoxic, cholinesterase inhibitors for Alzheimer disease - Boulebd_2017_Future.Med.Chem_9_723 |
| Author(s) : Boulebd H , Ismaili L , Martin H , Bonet A , Chioua M , Marco Contelles J , Belfaitah A |
| Ref : Future Med Chem , 9 :723 , 2017 |
| Abstract : |
| PubMedSearch : Boulebd_2017_Future.Med.Chem_9_723 |
| PubMedID: 28485637 |
| Title : Synthesis and biological assessment of racemic benzochromenopyrimidinetriones as promising agents for Alzheimer's disease therapy - Dgachi_2017_Future.Med.Chem_9_715 |
| Author(s) : Dgachi Y , Martin H , Bonet A , Chioua M , Iriepa I , Moraleda I , Chabchoub F , Marco-Contelles J , Ismaili L |
| Ref : Future Med Chem , 9 :715 , 2017 |
| Abstract : |
| PubMedSearch : Dgachi_2017_Future.Med.Chem_9_715 |
| PubMedID: 28504912 |
| Title : Synthesis and Biological Assessment of Racemic Benzochromenopyrimidinimines as Antioxidant, Cholinesterase, and Abeta1-42 Aggregation Inhibitors for Alzheimer's Disease Therapy - Dgachi_2016_ChemMedChem_11_1318 |
| Author(s) : Dgachi Y , Ismaili L , Knez D , Benchekroun M , Martin H , Szalaj N , Wehle S , Bautista-Aguilera OM , Luzet V , Bonnet A , Malawska B , Gobec S , Chioua M , Decker M , Chabchoub F , Marco-Contelles J |
| Ref : ChemMedChem , 11 :1318 , 2016 |
| Abstract : |
| PubMedSearch : Dgachi_2016_ChemMedChem_11_1318 |
| PubMedID: 26804623 |
| Title : Imidazopyranotacrines as Non-Hepatotoxic, Selective Acetylcholinesterase Inhibitors, and Antioxidant Agents for Alzheimer's Disease Therapy - Boulebd_2016_Molecules_21_ |
| Author(s) : Boulebd H , Ismaili L , Bartolini M , Bouraiou A , Andrisano V , Martin H , Bonet A , Moraleda I , Iriepa I , Chioua M , Belfaitah A , Marco-Contelles J |
| Ref : Molecules , 21 : , 2016 |
| Abstract : |
| PubMedSearch : Boulebd_2016_Molecules_21_ |
| PubMedID: 27023499 |
| Title : Comprehensive Screening of Eight Known Causative Genes in Congenital Hypothyroidism With Gland-in-Situ - Nicholas_2016_J.Clin.Endocrinol.Metab_101_4521 |
| Author(s) : Nicholas AK , Serra EG , Cangul H , Alyaarubi S , Ullah I , Schoenmakers E , Deeb A , Habeb AM , Almaghamsi M , Peters C , Nathwani N , Aycan Z , Saglam H , Bober E , Dattani M , Shenoy S , Murray PG , Babiker A , Willemsen R , Thankamony A , Lyons G , Irwin R , Padidela R , Tharian K , Davies JH , Puthi V , Park SM , Massoud AF , Gregory JW , Albanese A , Pease-Gevers E , Martin H , Brugger K , Maher ER , Chatterjee VK , Anderson CA , Schoenmakers N |
| Ref : J Clinical Endocrinology Metab , 101 :4521 , 2016 |
| Abstract : |
| PubMedSearch : Nicholas_2016_J.Clin.Endocrinol.Metab_101_4521 |
| PubMedID: 27525530 |
| Title : Synthesis and Biological Evaluation of Benzochromenopyrimidinones as Cholinesterase Inhibitors and Potent Antioxidant, Non-Hepatotoxic Agents for Alzheimer's Disease - Dgachi_2016_Molecules_21_ |
| Author(s) : Dgachi Y , Bautista-Aguilera OM , Benchekroun M , Martin H , Bonet A , Knez D , Godyn J , Malawska B , Gobec S , Chioua M , Janockova J , Soukup O , Chabchoub F , Marco-Contelles J , Ismaili L |
| Ref : Molecules , 21 : , 2016 |
| Abstract : |
| PubMedSearch : Dgachi_2016_Molecules_21_ |
| PubMedID: 27187348 |
| Title : Tetrahydropyranodiquinolin-8-amines as new, non hepatotoxic, antioxidant, and acetylcholinesterase inhibitors for Alzheimer's disease therapy - Dgachi_2016_Eur.J.Med.Chem_126_576 |
| Author(s) : Dgachi Y , Sokolov O , Luzet V , Godyn J , Panek D , Bonet A , Martin H , Iriepa I , Moraleda I , Garcia-Iriepa C , Janockova J , Richert L , Soukup O , Malawska B , Chabchoub F , Marco-Contelles J , Ismaili L |
| Ref : Eur Journal of Medicinal Chemistry , 126 :576 , 2016 |
| Abstract : |
| PubMedSearch : Dgachi_2016_Eur.J.Med.Chem_126_576 |
| PubMedID: 27918993 |
| Title : Genome Sequences of 228 Shiga Toxin-Producing Escherichia coli Isolates and 12 Isolates Representing Other Diarrheagenic E. coli Pathotypes - Trees_2014_Genome.Announc_2_e00718 |
| Author(s) : Trees E , Strockbine N , Changayil S , Ranganathan S , Zhao K , Weil R , Maccannell D , Sabol A , Schmidtke A , Martin H , Stripling D , Ribot EM , Gerner-Smidt P |
| Ref : Genome Announc , 2 : , 2014 |
| Abstract : |
| PubMedSearch : Trees_2014_Genome.Announc_2_e00718 |
| PubMedID: 25103754 |
| Gene_locus related to this paper: ecoli-fes , ecoli-MCMK , ecoli-ybff , ecoli-yiel , ecoli-ypt1 , ecoli-Z1930 , ecoli-YfhR |
| Title : Uncoupling of the endocannabinoid signalling complex in a mouse model of fragile X syndrome - Jung_2012_Nat.Commun_3_1080 |
| Author(s) : Jung KM , Sepers M , Henstridge CM , Lassalle O , Neuhofer D , Martin H , Ginger M , Frick A , DiPatrizio NV , Mackie K , Katona I , Piomelli D , Manzoni OJ |
| Ref : Nat Commun , 3 :1080 , 2012 |
| Abstract : |
| PubMedSearch : Jung_2012_Nat.Commun_3_1080 |
| PubMedID: 23011134 |