Title : Highly Specific Miniaturized Fluorescent Monoacylglycerol Lipase Probes Enable Translational Research - Hentsch_2025_J.Am.Chem.Soc__ |
Author(s) : Hentsch A , Guberman M , Radetzki S , Kaushik S , Huizenga M , He Y , Contzen J , Kuhn B , Benz J , Schippers M , Paul J , Leibrock L , Collin L , Wittwer M , Topp A , O'Hara F , Heer D , Hochstrasser R , Blaising J , von Kries JP , Mu L , van der Stelt M , Mergenthaler P , Lipstein N , Grether U , Nazare M |
Ref : Journal of the American Chemical Society , : , 2025 |
Abstract : |
PubMedSearch : Hentsch_2025_J.Am.Chem.Soc__ |
PubMedID: 40063733 |
Gene_locus related to this paper: human-MGLL |
Title : A Highly Selective and Versatile Probe Platform for Visualization of Monoacylglycerol Lipase - Hentsch_2025_Angew.Chem.Int.Ed.Engl__e202413405 |
Author(s) : Hentsch A , Guberman M , Radetzki S , Kaushik S , Huizenga M , Paul J , Schippers M , Benz J , Kuhn B , Heer D , Topp A , Esteves Gloria L , Walter A , Hochstrasser R , Wittwer MB , von Kries JP , Collin L , Blaising J , van der Stelt M , Lipstein N , Grether U , Nazare M |
Ref : Angew Chem Int Ed Engl , :e202413405 , 2025 |
Abstract : |
PubMedSearch : Hentsch_2025_Angew.Chem.Int.Ed.Engl__e202413405 |
PubMedID: 39916545 |
Gene_locus related to this paper: human-MGLL |
Title : Chemical Probes for Investigating the Endocannabinoid System - Hanske_2025_Curr.Top.Behav.Neurosci__ |
Author(s) : Hanske A , Nazare M , Grether U |
Ref : Curr Top Behavioral Neuroscience , : , 2025 |
Abstract : |
PubMedSearch : Hanske_2025_Curr.Top.Behav.Neurosci__ |
PubMedID: 39747798 |
Title : Development of a Highly Selective NanoBRET Probe to Assess MAGL Inhibition in Live Cells - Gazzi_2024_Chembiochem__e202400704 |
Author(s) : Gazzi T , Brennecke B , Olikauskas V , Hochstrasser R , Wang H , Keen Chao S , Atz K , Mostinski Y , Topp A , Heer D , Kaufmann I , Ritter M , Gobbi L , Hornsperger B , Wagner B , Richter H , O'Hara F , Wittwer MB , Jul Hansen D , Collin L , Kuhn B , Benz J , Grether U , Nazare M |
Ref : Chembiochem , :e202400704 , 2024 |
Abstract : |
PubMedSearch : Gazzi_2024_Chembiochem__e202400704 |
PubMedID: 39607084 |
Gene_locus related to this paper: human-MGLL |
Title : Enhancing Drug Discovery and Development through the Integration of Medicinal Chemistry, Chemical Biology, and Academia-Industry Partnerships: Insights from Roche's Endocannabinoid System Projects - Aebi_2024_Chimia.(Aarau)_78_499 |
Author(s) : Aebi J , Atz K , Ametamey SM , Benz J , Blaising J , Butini S , Campiani G , Carreira EM , Collin L , De Lago E , Gazzi T , Gertsch J , Gobbi L , Guba W , Fernandez-Ruiz J , Fingerle J , Haider A , He Y , Heitman LH , Honer M , Hunziker D , Kuhn B , Maccarrone M , Marki HP , Martin RE , Mohr P , Mu L , Nazare M , Nippa DF , Oddi S , O'Hara F , Pacher P , Romero J , Rover S , Rufer AC , Schibli R , Schneider G , Stepan AF , Sykes DA , Ullmer C , van der Stelt M , Veprintsev DB , Wittwer MB , Grether U |
Ref : Chimia (Aarau) , 78 :499 , 2024 |
Abstract : |
PubMedSearch : Aebi_2024_Chimia.(Aarau)_78_499 |
PubMedID: 39221845 |