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Title : (+\/-)-BIGI-3h: Pentatarget-Directed Ligand combining Cholinesterase, Monoamine Oxidase, and Glycogen Synthase Kinase 3beta Inhibition with Calcium Channel Antagonism and Antiaggregating Properties for Alzheimer's Disease - Ismaili_2021_ACS.Chem.Neurosci__ |
Author(s) : Ismaili L , Monnin J , Etievant A , Arribas RL , Viejo L , Refouvelet B , Soukup O , Janockova J , Hepnarova V , Korabecny J , Kucera T , Jun D , Andrys R , Musilek K , Baguet A , Garcia-Frutos EM , De Simone A , Andrisano V , Bartolini M , de los Rios C , Marco-Contelles J , Haffen E |
Ref : ACS Chem Neurosci , : , 2021 |
Abstract : Ismaili_2021_ACS.Chem.Neurosci__ |
ESTHER : Ismaili_2021_ACS.Chem.Neurosci__ |
PubMedSearch : Ismaili_2021_ACS.Chem.Neurosci__ |
PubMedID: 33797877 |
Title : New Dual Small Molecules for Alzheimer's Disease Therapy Combining Histamine H3 Receptor (H3R) Antagonism and Calcium Channels Blockade with Additional Cholinesterase Inhibition - Malek_2019_J.Med.Chem_62_11416 |
Author(s) : Malek R , Arribas RL , Palomino-Antolin A , Totoson P , Demougeot C , Kobrlova T , Soukup O , Iriepa I , Moraleda I , Diez-Iriepa D , Godyn J , Panek D , Malawska B , Gluch-Lutwin M , Mordyl B , Siwek A , Chabchoub F , Marco-Contelles J , Kiec-Kononowicz K , Egea J , de los Rios C , Ismaili L |
Ref : Journal of Medicinal Chemistry , 62 :11416 , 2019 |
Abstract : Malek_2019_J.Med.Chem_62_11416 |
ESTHER : Malek_2019_J.Med.Chem_62_11416 |
PubMedSearch : Malek_2019_J.Med.Chem_62_11416 |
PubMedID: 31724859 |