Report for Janssen APA

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References (6)

Title : Chemical Proteomics Reveals Antibiotic Targets of Oxadiazolones in MRSA - Bakker_2023_J.Am.Chem.Soc_145_1136
Author(s) : Bakker AT , Kotsogianni I , Mirenda L , Straub VM , Avalos M , van den Berg R , Florea BI , van Wezel GP , Janssen APA , Martin NI , van der Stelt M
Ref : Journal of the American Chemical Society , 145 :1136 , 2023
Abstract : Bakker_2023_J.Am.Chem.Soc_145_1136
ESTHER : Bakker_2023_J.Am.Chem.Soc_145_1136
PubMedSearch : Bakker_2023_J.Am.Chem.Soc_145_1136
PubMedID: 36584241
Gene_locus related to this paper: staa3-q2fkj0 , staau-MW0741 , staau-MW2456 , staau-SA1143 , staau-SA2367 , staau-SAV0321 , staau-SAV0655

Title : A monoacylglycerol lipase inhibitor showing therapeutic efficacy in mice without central side effects or dependence - Jiang_2023_Nat.Commun_14_8039
Author(s) : Jiang M , Huizenga MCW , Wirt JL , Paloczi J , Amedi A , van den Berg R , Benz J , Collin L , Deng H , Di X , Driever WF , Florea BI , Grether U , Janssen APA , Hankemeier T , Heitman LH , Lam TW , Mohr F , Pavlovic A , Ruf I , van den Hurk H , Stevens AF , van der Vliet D , van der Wel T , Wittwer MB , van Boeckel CAA , Pacher P , Hohmann AG , van der Stelt M
Ref : Nat Commun , 14 :8039 , 2023
Abstract : Jiang_2023_Nat.Commun_14_8039
ESTHER : Jiang_2023_Nat.Commun_14_8039
PubMedSearch : Jiang_2023_Nat.Commun_14_8039
PubMedID: 38052772

Title : ABHD2 Inhibitor Identified by Activity-Based Protein Profiling Reduces Acrosome Reaction - Baggelaar_2019_ACS.Chem.Biol_14_2295
Author(s) : Baggelaar MP , den Dulk H , Florea BI , Fazio D , Perruzza D , Bernabo N , Raspa M , Janssen APA , Scavizzi F , Barboni B , Overkleeft HS , Maccarrone M , van der Stelt M
Ref : ACS Chemical Biology , 14 :2295 , 2019
Abstract : Baggelaar_2019_ACS.Chem.Biol_14_2295
ESTHER : Baggelaar_2019_ACS.Chem.Biol_14_2295
PubMedSearch : Baggelaar_2019_ACS.Chem.Biol_14_2295
PubMedID: 31525885
Gene_locus related to this paper: human-ABHD2 , human-ABHD3

Title : Development of a Multiplexed Activity-Based Protein Profiling Assay to Evaluate Activity of Endocannabinoid Hydrolase Inhibitors - Janssen_2018_ACS.Chem.Biol_13_2406
Author(s) : Janssen APA , van der Vliet D , Bakker AT , Jiang M , Grimm SH , Campiani G , Butini S , van der Stelt M
Ref : ACS Chemical Biology , 13 :2406 , 2018
Abstract : Janssen_2018_ACS.Chem.Biol_13_2406
ESTHER : Janssen_2018_ACS.Chem.Biol_13_2406
PubMedSearch : Janssen_2018_ACS.Chem.Biol_13_2406
PubMedID: 30199617

Title : Design and Synthesis of Quenched Activity-based Probes for Diacylglycerol Lipase and alpha,beta-Hydrolase Domain Containing Protein 6 - van Rooden_2018_Chem.Asian.J_13_3491
Author(s) : van Rooden EJ , Kohsiek M , Kreekel R , van Esbroeck ACM , van den Nieuwendijk A , Janssen APA , van den Berg R , Overkleeft HS , van der Stelt M
Ref : Chem Asian J , 13 :3491 , 2018
Abstract : van Rooden_2018_Chem.Asian.J_13_3491
ESTHER : van Rooden_2018_Chem.Asian.J_13_3491
PubMedSearch : van Rooden_2018_Chem.Asian.J_13_3491
PubMedID: 29901868

Title : Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474 - van Esbroeck_2017_Science_356_1084
Author(s) : van Esbroeck ACM , Janssen APA , Cognetta AB, 3rd , Ogasawara D , Shpak G , van der Kroeg M , Kantae V , Baggelaar MP , de Vrij FMS , Deng H , Allara M , Fezza F , Lin Z , van der Wel T , Soethoudt M , Mock ED , den Dulk H , Baak IL , Florea BI , Hendriks G , De Petrocellis L , Overkleeft HS , Hankemeier T , De Zeeuw CI , Di Marzo V , Maccarrone M , Cravatt BF , Kushner SA , van der Stelt M
Ref : Science , 356 :1084 , 2017
Abstract : van Esbroeck_2017_Science_356_1084
ESTHER : van Esbroeck_2017_Science_356_1084
PubMedSearch : van Esbroeck_2017_Science_356_1084
PubMedID: 28596366