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Title : Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions - Papa_2022_Eur.J.Med.Chem_246_114952 |
Author(s) : Papa A , Pasquini S , Galvani F , Cammarota M , Contri C , Carullo G , Gemma S , Ramunno A , Lamponi S , Gorelli B , Saponara S , Varani K , Mor M , Campiani G , Boscia F , Vincenzi F , Lodola A , Butini S |
Ref : Eur Journal of Medicinal Chemistry , 246 :114952 , 2022 |
Abstract : Papa_2022_Eur.J.Med.Chem_246_114952 |
ESTHER : Papa_2022_Eur.J.Med.Chem_246_114952 |
PubMedSearch : Papa_2022_Eur.J.Med.Chem_246_114952 |
PubMedID: 36462439 |
Title : Development and Pharmacological Characterization of Selective Blockers of 2-Arachidonoyl Glycerol Degradation with Efficacy in Rodent Models of Multiple Sclerosis and Pain - Brindisi_2016_J.Med.Chem_59_2612 |
Author(s) : Brindisi M , Maramai S , Gemma S , Brogi S , Grillo A , Di Cesare Mannelli L , Gabellieri E , Lamponi S , Saponara S , Gorelli B , Tedesco D , Bonfiglio T , Landry C , Jung KM , Armirotti A , Luongo L , Ligresti A , Piscitelli F , Bertucci C , Dehouck MP , Campiani G , Maione S , Ghelardini C , Pittaluga A , Piomelli D , Di Marzo V , Butini S |
Ref : Journal of Medicinal Chemistry , 59 :2612 , 2016 |
Abstract : Brindisi_2016_J.Med.Chem_59_2612 |
ESTHER : Brindisi_2016_J.Med.Chem_59_2612 |
PubMedSearch : Brindisi_2016_J.Med.Chem_59_2612 |
PubMedID: 26888301 |