BBB endogenous transporters

General

Choline transporter and the L-type amino acid transporter 1 (LAT1)

Inhibitor	Main targeted enzyme families	Type	Structure
Tacrine-amino-propyl-carbamoyl-phenyl-propanoate-CpdL3	ACHE BCHE	Multitarget BBB endogenous transporters Derivative of Tacrine Acridine Propionate Carboxamide
Tacrine-hexyl-pyridinium-CpdC4	ACHE BCHE	Multitarget Pyridine Alkyl linked bis-ligand BBB endogenous transporters Pyridinium Derivative of Tacrine Acridine