Title : Derivatives of 9-phosphorylated acridine as butyrylcholinesterase inhibitors with antioxidant activity and the ability to inhibit beta-amyloid self-aggregation: potential therapeutic agents for Alzheimer's disease - Makhaeva_2023_Front.Pharmacol_14_1219980 |
Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Astakhova TY , Timokhina EN , Serebryakova OG , Shchepochkin AV , Averkov MA , Utepova IA , Demina NS , Radchenko EV , Palyulin VA , Fisenko VP , Bachurin SO , Chupakhin ON , Charushin VN , Richardson RJ |
Ref : Front Pharmacol , 14 :1219980 , 2023 |
Abstract : |
PubMedSearch : Makhaeva_2023_Front.Pharmacol_14_1219980 |
PubMedID: 37654616 |
Title : 9-Substituted acridine derivatives as acetylcholinesterase and butyrylcholinesterase inhibitors possessing antioxidant activity for Alzheimer's disease treatment - Makhaeva_2017_Bioorg.Med.Chem_25_5981 |
Author(s) : Makhaeva GF , Lushchekina SV , Boltneva NP , Serebryakova OG , Rudakova EV , Ustyugov AA , Bachurin SO , Shchepochkin AV , Chupakhin ON , Charushin VN , Richardson RJ |
Ref : Bioorganic & Medicinal Chemistry , 25 :5981 , 2017 |
Abstract : |
PubMedSearch : Makhaeva_2017_Bioorg.Med.Chem_25_5981 |
PubMedID: 28986116 |
Title : Synthesis, molecular docking, and biological activity of polyfluoroalkyl dihydroazolo[5,1-c][1,2,4]triazines as selective carboxylesterase inhibitors - Shchegol'kov_2017_Bioorg.Med.Chem_25_3997 |
Author(s) : Shchegol'kov EV , Makhaeva GF , Boltneva NP , Lushchekina SV , Serebryakova OG , Rudakova EV , Kovaleva NV , Burgart YV , Saloutin VI , Chupakhin ON , Bachurin SO , Richardson RJ |
Ref : Bioorganic & Medicinal Chemistry , 25 :3997 , 2017 |
Abstract : |
PubMedSearch : Shchegol'kov_2017_Bioorg.Med.Chem_25_3997 |
PubMedID: 28578994 |
Title : Alkyl 2-arylhydrazinylidene-3-oxo-3-polyfluoroalkylpropionates as new effective and selective inhibitors of carboxylesterase - Boltneva_2015_Dokl.Biochem.Biophys_465_381 |
Author(s) : Boltneva NP , Makhaeva GF , Kovaleva NV , Lushchekina SV , Burgart YV , Shchegol'kov EV , Saloutin VI , Chupakhin ON |
Ref : Dokl Biochem Biophys , 465 :381 , 2015 |
Abstract : |
PubMedSearch : Boltneva_2015_Dokl.Biochem.Biophys_465_381 |
PubMedID: 26728730 |