Timokhina EN

References (21)

Title : 1-Azinyl-1'-Alkenylferrocenes with Anticholinesterase, Antioxidant, and Antiaggregating Activities as Multifunctional Agents for Potential Treatment of Alzheimer's Disease - Makhaeva_2025_Pharmaceuticals.(Basel)_18_
Author(s) : Makhaeva GF , Utepova IA , Rudakova EV , Kovaleva NV , Boltneva NP , Zyryanova EY , Musikhina AA , Lazarev VF , Vladimirova SA , Guzhova IV , Ganebnykh IN , Astakhova TY , Timokhina EN , Chupakhin ON , Charushin VN , Richardson RJ
Ref : Pharmaceuticals (Basel) , 18 : , 2025
Abstract :
PubMedSearch : Makhaeva_2025_Pharmaceuticals.(Basel)_18_
PubMedID: 41471351

Title : Synthesis, biological evaluation, and in silico studies of pyridoxal-amiridine hybrids as multitargeting anti-Alzheimer's disease agents - Makhaeva_2025_Eur.J.Med.Chem_303_118397
Author(s) : Makhaeva GF , Grishchenko MV , Rudakova EV , Kovaleva NV , Boltneva NP , Skornyakova TS , Khudina OG , Shchegolkov EV , Zhilina EF , Astakhova TY , Pronkin PG , Timokhina EN , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ
Ref : Eur Journal of Medicinal Chemistry , 303 :118397 , 2025
Abstract :
PubMedSearch : Makhaeva_2025_Eur.J.Med.Chem_303_118397
PubMedID: 41338134

Title : 1-Azinyl-1'-Alkenylferrocenes with Anticholinesterase, Antioxidant, and Antiaggregating Activities as Multifunctional Agents for Potential Treatment of Alzheimer's Disease - Makhaeva_2025_Pharmaceuticals.(Basel)_18_
Author(s) : Makhaeva GF , Utepova IA , Rudakova EV , Kovaleva NV , Boltneva NP , Zyryanova EY , Musikhina AA , Lazarev VF , Vladimirova SA , Guzhova IV , Ganebnykh IN , Astakhova TY , Timokhina EN , Chupakhin ON , Charushin VN , Richardson RJ
Ref : Pharmaceuticals (Basel) , 18 : , 2025
Abstract :
PubMedSearch : Makhaeva_2025_Pharmaceuticals.(Basel)_18_
PubMedID: 41471351

Title : Synthesis, biological evaluation, and in silico studies of pyridoxal-amiridine hybrids as multitargeting anti-Alzheimer's disease agents - Makhaeva_2025_Eur.J.Med.Chem_303_118397
Author(s) : Makhaeva GF , Grishchenko MV , Rudakova EV , Kovaleva NV , Boltneva NP , Skornyakova TS , Khudina OG , Shchegolkov EV , Zhilina EF , Astakhova TY , Pronkin PG , Timokhina EN , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ
Ref : Eur Journal of Medicinal Chemistry , 303 :118397 , 2025
Abstract :
PubMedSearch : Makhaeva_2025_Eur.J.Med.Chem_303_118397
PubMedID: 41338134

Title : Conjugates of amiridine and salicylic derivatives as promising multifunctional CNS agents for potential treatment of Alzheimer's disease - Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819
Author(s) : Makhaeva GF , Grishchenko MV , Kovaleva NV , Boltneva NP , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Lushchekina SV , Khudina OG , Zhilina EF , Shchegolkov EV , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ
Ref : Arch Pharm (Weinheim) , 358 :e2400819 , 2025
Abstract :
PubMedSearch : Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819
PubMedID: 39686878

Title : Conjugates of amiridine and salicylic derivatives as promising multifunctional CNS agents for potential treatment of Alzheimer's disease - Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819
Author(s) : Makhaeva GF , Grishchenko MV , Kovaleva NV , Boltneva NP , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Lushchekina SV , Khudina OG , Zhilina EF , Shchegolkov EV , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ
Ref : Arch Pharm (Weinheim) , 358 :e2400819 , 2025
Abstract :
PubMedSearch : Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819
PubMedID: 39686878

Title : Synthesis of Tacrine\/Amiridine Conjugates with Aminomethylidene Derivatives of Trifluoroacetoacetic Ester and their Biological Potential for the Therapy of Alzheimer's Disease - Grishchenko_2025_ChemMedChem__e202500723
Author(s) : Grishchenko MV , Makhaeva GF , Burgart YV , Kovaleva NV , Boltneva NP , Skornyakova TS , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Shchegolkov EV , Saloutin V , Charushin VN
Ref : ChemMedChem , :e202500723 , 2025
Abstract :
PubMedSearch : Grishchenko_2025_ChemMedChem__e202500723
PubMedID: 41047157

Title : Synthesis, biological evaluation, and in silico studies of pyridoxal-amiridine hybrids as multitargeting anti-Alzheimer's disease agents - Makhaeva_2025_Eur.J.Med.Chem_303_118397
Author(s) : Makhaeva GF , Grishchenko MV , Rudakova EV , Kovaleva NV , Boltneva NP , Skornyakova TS , Khudina OG , Shchegolkov EV , Zhilina EF , Astakhova TY , Pronkin PG , Timokhina EN , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ
Ref : Eur Journal of Medicinal Chemistry , 303 :118397 , 2025
Abstract :
PubMedSearch : Makhaeva_2025_Eur.J.Med.Chem_303_118397
PubMedID: 41338134

Title : Synthesis of Tacrine\/Amiridine Conjugates with Aminomethylidene Derivatives of Trifluoroacetoacetic Ester and their Biological Potential for the Therapy of Alzheimer's Disease - Grishchenko_2025_ChemMedChem__e202500723
Author(s) : Grishchenko MV , Makhaeva GF , Burgart YV , Kovaleva NV , Boltneva NP , Skornyakova TS , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Shchegolkov EV , Saloutin V , Charushin VN
Ref : ChemMedChem , :e202500723 , 2025
Abstract :
PubMedSearch : Grishchenko_2025_ChemMedChem__e202500723
PubMedID: 41047157

Title : 1-Azinyl-1'-Alkenylferrocenes with Anticholinesterase, Antioxidant, and Antiaggregating Activities as Multifunctional Agents for Potential Treatment of Alzheimer's Disease - Makhaeva_2025_Pharmaceuticals.(Basel)_18_
Author(s) : Makhaeva GF , Utepova IA , Rudakova EV , Kovaleva NV , Boltneva NP , Zyryanova EY , Musikhina AA , Lazarev VF , Vladimirova SA , Guzhova IV , Ganebnykh IN , Astakhova TY , Timokhina EN , Chupakhin ON , Charushin VN , Richardson RJ
Ref : Pharmaceuticals (Basel) , 18 : , 2025
Abstract :
PubMedSearch : Makhaeva_2025_Pharmaceuticals.(Basel)_18_
PubMedID: 41471351

Title : Conjugates of amiridine and salicylic derivatives as promising multifunctional CNS agents for potential treatment of Alzheimer's disease - Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819
Author(s) : Makhaeva GF , Grishchenko MV , Kovaleva NV , Boltneva NP , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Lushchekina SV , Khudina OG , Zhilina EF , Shchegolkov EV , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ
Ref : Arch Pharm (Weinheim) , 358 :e2400819 , 2025
Abstract :
PubMedSearch : Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819
PubMedID: 39686878

Title : Synthesis of Tacrine\/Amiridine Conjugates with Aminomethylidene Derivatives of Trifluoroacetoacetic Ester and their Biological Potential for the Therapy of Alzheimer's Disease - Grishchenko_2025_ChemMedChem__e202500723
Author(s) : Grishchenko MV , Makhaeva GF , Burgart YV , Kovaleva NV , Boltneva NP , Skornyakova TS , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Shchegolkov EV , Saloutin V , Charushin VN
Ref : ChemMedChem , :e202500723 , 2025
Abstract :
PubMedSearch : Grishchenko_2025_ChemMedChem__e202500723
PubMedID: 41047157

Title : Combining Experimental and Computational Methods to Produce Conjugates of Anticholinesterase and Antioxidant Pharmacophores with Linker Chemistries Affecting Biological Activities Related to Treatment of Alzheimer's Disease - Makhaeva_2024_Molecules_29_321
Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Astakhova TY , Timokhina EN , Serkov IV , Proshin AN , Soldatova YV , Poletaeva DA , Faingold, II , Mumyatova VA , Terentiev AA , Radchenko EV , Palyulin VA , Bachurin SO , Richardson RJ
Ref : Molecules , 29 :321 , 2024
Abstract :
PubMedSearch : Makhaeva_2024_Molecules_29_321
PubMedID: 38257233

Title : Combining Experimental and Computational Methods to Produce Conjugates of Anticholinesterase and Antioxidant Pharmacophores with Linker Chemistries Affecting Biological Activities Related to Treatment of Alzheimer's Disease - Makhaeva_2024_Molecules_29_321
Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Astakhova TY , Timokhina EN , Serkov IV , Proshin AN , Soldatova YV , Poletaeva DA , Faingold, II , Mumyatova VA , Terentiev AA , Radchenko EV , Palyulin VA , Bachurin SO , Richardson RJ
Ref : Molecules , 29 :321 , 2024
Abstract :
PubMedSearch : Makhaeva_2024_Molecules_29_321
PubMedID: 38257233

Title : Combining Experimental and Computational Methods to Produce Conjugates of Anticholinesterase and Antioxidant Pharmacophores with Linker Chemistries Affecting Biological Activities Related to Treatment of Alzheimer's Disease - Makhaeva_2024_Molecules_29_321
Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Astakhova TY , Timokhina EN , Serkov IV , Proshin AN , Soldatova YV , Poletaeva DA , Faingold, II , Mumyatova VA , Terentiev AA , Radchenko EV , Palyulin VA , Bachurin SO , Richardson RJ
Ref : Molecules , 29 :321 , 2024
Abstract :
PubMedSearch : Makhaeva_2024_Molecules_29_321
PubMedID: 38257233

Title : Derivatives of 9-phosphorylated acridine as butyrylcholinesterase inhibitors with antioxidant activity and the ability to inhibit beta-amyloid self-aggregation: potential therapeutic agents for Alzheimer's disease - Makhaeva_2023_Front.Pharmacol_14_1219980
Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Astakhova TY , Timokhina EN , Serebryakova OG , Shchepochkin AV , Averkov MA , Utepova IA , Demina NS , Radchenko EV , Palyulin VA , Fisenko VP , Bachurin SO , Chupakhin ON , Charushin VN , Richardson RJ
Ref : Front Pharmacol , 14 :1219980 , 2023
Abstract :
PubMedSearch : Makhaeva_2023_Front.Pharmacol_14_1219980
PubMedID: 37654616

Title : Conjugates of Tacrine and Salicylic Acid Derivatives as New Promising Multitarget Agents for Alzheimer's Disease - Makhaeva_2023_Int.J.Mol.Sci_24_2285
Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Grishchenko MV , Lushchekina SV , Astakhova TY , Serebryakova OG , Timokhina EN , Zhilina EF , Shchegolkov EV , Ulitko MV , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Bachurin SO , Richardson RJ
Ref : Int J Mol Sci , 24 :2285 , 2023
Abstract :
PubMedSearch : Makhaeva_2023_Int.J.Mol.Sci_24_2285
PubMedID: 36768608

Title : Derivatives of 9-phosphorylated acridine as butyrylcholinesterase inhibitors with antioxidant activity and the ability to inhibit beta-amyloid self-aggregation: potential therapeutic agents for Alzheimer's disease - Makhaeva_2023_Front.Pharmacol_14_1219980
Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Astakhova TY , Timokhina EN , Serebryakova OG , Shchepochkin AV , Averkov MA , Utepova IA , Demina NS , Radchenko EV , Palyulin VA , Fisenko VP , Bachurin SO , Chupakhin ON , Charushin VN , Richardson RJ
Ref : Front Pharmacol , 14 :1219980 , 2023
Abstract :
PubMedSearch : Makhaeva_2023_Front.Pharmacol_14_1219980
PubMedID: 37654616

Title : Conjugates of Tacrine and Salicylic Acid Derivatives as New Promising Multitarget Agents for Alzheimer's Disease - Makhaeva_2023_Int.J.Mol.Sci_24_2285
Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Grishchenko MV , Lushchekina SV , Astakhova TY , Serebryakova OG , Timokhina EN , Zhilina EF , Shchegolkov EV , Ulitko MV , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Bachurin SO , Richardson RJ
Ref : Int J Mol Sci , 24 :2285 , 2023
Abstract :
PubMedSearch : Makhaeva_2023_Int.J.Mol.Sci_24_2285
PubMedID: 36768608

Title : Derivatives of 9-phosphorylated acridine as butyrylcholinesterase inhibitors with antioxidant activity and the ability to inhibit beta-amyloid self-aggregation: potential therapeutic agents for Alzheimer's disease - Makhaeva_2023_Front.Pharmacol_14_1219980
Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Astakhova TY , Timokhina EN , Serebryakova OG , Shchepochkin AV , Averkov MA , Utepova IA , Demina NS , Radchenko EV , Palyulin VA , Fisenko VP , Bachurin SO , Chupakhin ON , Charushin VN , Richardson RJ
Ref : Front Pharmacol , 14 :1219980 , 2023
Abstract :
PubMedSearch : Makhaeva_2023_Front.Pharmacol_14_1219980
PubMedID: 37654616

Title : Conjugates of Tacrine and Salicylic Acid Derivatives as New Promising Multitarget Agents for Alzheimer's Disease - Makhaeva_2023_Int.J.Mol.Sci_24_2285
Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Grishchenko MV , Lushchekina SV , Astakhova TY , Serebryakova OG , Timokhina EN , Zhilina EF , Shchegolkov EV , Ulitko MV , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Bachurin SO , Richardson RJ
Ref : Int J Mol Sci , 24 :2285 , 2023
Abstract :
PubMedSearch : Makhaeva_2023_Int.J.Mol.Sci_24_2285
PubMedID: 36768608