Title : Search for multifunctional agents against Alzheimer's disease among non-imidazole histamine H3 receptor ligands. In vitro and in vivo pharmacological evaluation and computational studies of piperazine derivatives - Jonczyk_2019_Bioorg.Chem_90_103084 |
Author(s) : Jonczyk J , Lodarski K , Staszewski M , Godyn J , Zareba P , Soukup O , Janockova J , Korabecny J , Salat K , Malikowska-Racia N , Hebda M , Szalaj N , Filipek B , Walczynski K , Malawska B , Bajda M |
Ref : Bioorg Chem , 90 :103084 , 2019 |
Abstract : |
PubMedSearch : Jonczyk_2019_Bioorg.Chem_90_103084 |
PubMedID: 31271942 |
Title : Development of an in-vivo active reversible butyrylcholinesterase inhibitor - Kosak_2016_Sci.Rep_6_39495 |
Author(s) : Kosak U , Brus B , Knez D , Sink R , Zakelj S , Trontelj J , Pislar A , Slenc J , Gobec M , Zivin M , Tratnjek L , Perse M , Salat K , Podkowa A , Filipek B , Nachon F , Brazzolotto X , Wieckowska A , Malawska B , Stojan J , Rascan IM , Kos J , Coquelle N , Colletier JP , Gobec S |
Ref : Sci Rep , 6 :39495 , 2016 |
Abstract : |
PubMedSearch : Kosak_2016_Sci.Rep_6_39495 |
PubMedID: 28000737 |
Gene_locus related to this paper: human-BCHE |
Title : Synthesis of new N-benzylpiperidine derivatives as cholinesterase inhibitors with beta-amyloid anti-aggregation properties and beneficial effects on memory in vivo - Wieckowska_2015_Bioorg.Med.Chem_23_2445 |
Author(s) : Wieckowska A , Wieckowski K , Bajda M , Brus B , Salat K , Czerwinska P , Gobec S , Filipek B , Malawska B |
Ref : Bioorganic & Medicinal Chemistry , 23 :2445 , 2015 |
Abstract : |
PubMedSearch : Wieckowska_2015_Bioorg.Med.Chem_23_2445 |
PubMedID: 25868744 |