| Title : Synthesis, biological evaluation, and in silico studies of pyridoxal-amiridine hybrids as multitargeting anti-Alzheimer's disease agents - Makhaeva_2025_Eur.J.Med.Chem_303_118397 |
| Author(s) : Makhaeva GF , Grishchenko MV , Rudakova EV , Kovaleva NV , Boltneva NP , Skornyakova TS , Khudina OG , Shchegolkov EV , Zhilina EF , Astakhova TY , Pronkin PG , Timokhina EN , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ |
| Ref : Eur Journal of Medicinal Chemistry , 303 :118397 , 2025 |
| Abstract : |
| PubMedSearch : Makhaeva_2025_Eur.J.Med.Chem_303_118397 |
| PubMedID: 41338134 |
| Title : Synthesis, biological evaluation, and in silico studies of pyridoxal-amiridine hybrids as multitargeting anti-Alzheimer's disease agents - Makhaeva_2025_Eur.J.Med.Chem_303_118397 |
| Author(s) : Makhaeva GF , Grishchenko MV , Rudakova EV , Kovaleva NV , Boltneva NP , Skornyakova TS , Khudina OG , Shchegolkov EV , Zhilina EF , Astakhova TY , Pronkin PG , Timokhina EN , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ |
| Ref : Eur Journal of Medicinal Chemistry , 303 :118397 , 2025 |
| Abstract : |
| PubMedSearch : Makhaeva_2025_Eur.J.Med.Chem_303_118397 |
| PubMedID: 41338134 |
| Title : Conjugates of amiridine and salicylic derivatives as promising multifunctional CNS agents for potential treatment of Alzheimer's disease - Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819 |
| Author(s) : Makhaeva GF , Grishchenko MV , Kovaleva NV , Boltneva NP , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Lushchekina SV , Khudina OG , Zhilina EF , Shchegolkov EV , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ |
| Ref : Arch Pharm (Weinheim) , 358 :e2400819 , 2025 |
| Abstract : |
| PubMedSearch : Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819 |
| PubMedID: 39686878 |
| Title : Conjugates of amiridine and salicylic derivatives as promising multifunctional CNS agents for potential treatment of Alzheimer's disease - Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819 |
| Author(s) : Makhaeva GF , Grishchenko MV , Kovaleva NV , Boltneva NP , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Lushchekina SV , Khudina OG , Zhilina EF , Shchegolkov EV , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ |
| Ref : Arch Pharm (Weinheim) , 358 :e2400819 , 2025 |
| Abstract : |
| PubMedSearch : Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819 |
| PubMedID: 39686878 |
| Title : Synthesis of Tacrine\/Amiridine Conjugates with Aminomethylidene Derivatives of Trifluoroacetoacetic Ester and their Biological Potential for the Therapy of Alzheimer's Disease - Grishchenko_2025_ChemMedChem__e202500723 |
| Author(s) : Grishchenko MV , Makhaeva GF , Burgart YV , Kovaleva NV , Boltneva NP , Skornyakova TS , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Shchegolkov EV , Saloutin V , Charushin VN |
| Ref : ChemMedChem , :e202500723 , 2025 |
| Abstract : |
| PubMedSearch : Grishchenko_2025_ChemMedChem__e202500723 |
| PubMedID: 41047157 |
| Title : Synthesis, biological evaluation, and in silico studies of pyridoxal-amiridine hybrids as multitargeting anti-Alzheimer's disease agents - Makhaeva_2025_Eur.J.Med.Chem_303_118397 |
| Author(s) : Makhaeva GF , Grishchenko MV , Rudakova EV , Kovaleva NV , Boltneva NP , Skornyakova TS , Khudina OG , Shchegolkov EV , Zhilina EF , Astakhova TY , Pronkin PG , Timokhina EN , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ |
| Ref : Eur Journal of Medicinal Chemistry , 303 :118397 , 2025 |
| Abstract : |
| PubMedSearch : Makhaeva_2025_Eur.J.Med.Chem_303_118397 |
| PubMedID: 41338134 |
| Title : Synthesis of Tacrine\/Amiridine Conjugates with Aminomethylidene Derivatives of Trifluoroacetoacetic Ester and their Biological Potential for the Therapy of Alzheimer's Disease - Grishchenko_2025_ChemMedChem__e202500723 |
| Author(s) : Grishchenko MV , Makhaeva GF , Burgart YV , Kovaleva NV , Boltneva NP , Skornyakova TS , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Shchegolkov EV , Saloutin V , Charushin VN |
| Ref : ChemMedChem , :e202500723 , 2025 |
| Abstract : |
| PubMedSearch : Grishchenko_2025_ChemMedChem__e202500723 |
| PubMedID: 41047157 |
| Title : Conjugates of amiridine and salicylic derivatives as promising multifunctional CNS agents for potential treatment of Alzheimer's disease - Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819 |
| Author(s) : Makhaeva GF , Grishchenko MV , Kovaleva NV , Boltneva NP , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Lushchekina SV , Khudina OG , Zhilina EF , Shchegolkov EV , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ |
| Ref : Arch Pharm (Weinheim) , 358 :e2400819 , 2025 |
| Abstract : |
| PubMedSearch : Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819 |
| PubMedID: 39686878 |
| Title : Synthesis of Tacrine\/Amiridine Conjugates with Aminomethylidene Derivatives of Trifluoroacetoacetic Ester and their Biological Potential for the Therapy of Alzheimer's Disease - Grishchenko_2025_ChemMedChem__e202500723 |
| Author(s) : Grishchenko MV , Makhaeva GF , Burgart YV , Kovaleva NV , Boltneva NP , Skornyakova TS , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Shchegolkov EV , Saloutin V , Charushin VN |
| Ref : ChemMedChem , :e202500723 , 2025 |
| Abstract : |
| PubMedSearch : Grishchenko_2025_ChemMedChem__e202500723 |
| PubMedID: 41047157 |