| Title : Synthesis, biological evaluation, and in silico studies of pyridoxal-amiridine hybrids as multitargeting anti-Alzheimer's disease agents - Makhaeva_2025_Eur.J.Med.Chem_303_118397 |
| Author(s) : Makhaeva GF , Grishchenko MV , Rudakova EV , Kovaleva NV , Boltneva NP , Skornyakova TS , Khudina OG , Shchegolkov EV , Zhilina EF , Astakhova TY , Pronkin PG , Timokhina EN , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ |
| Ref : Eur Journal of Medicinal Chemistry , 303 :118397 , 2025 |
| Abstract : |
| PubMedSearch : Makhaeva_2025_Eur.J.Med.Chem_303_118397 |
| PubMedID: 41338134 |
| Title : Conjugates of anticholinesterase drugs ipidacrine and tacrine with thiouracils: synthesis and biological properties - Grishchenko_2025_Russ.Chem.Bull_73_3399 |
| Author(s) : Grishchenko MV , Khudina OG , Makhaeva GF , Burgart YV , Kovaleva NV , Rudakova EV , Boltneva NP , Ulitko MV , Saloutin VI , Charushin VN |
| Ref : Russ Chem Bull , 73 :3399 , 2025 |
| Abstract : |
| PubMedSearch : Grishchenko_2025_Russ.Chem.Bull_73_3399 |
| PubMedID: |
| Title : Synthesis, biological evaluation, and in silico studies of pyridoxal-amiridine hybrids as multitargeting anti-Alzheimer's disease agents - Makhaeva_2025_Eur.J.Med.Chem_303_118397 |
| Author(s) : Makhaeva GF , Grishchenko MV , Rudakova EV , Kovaleva NV , Boltneva NP , Skornyakova TS , Khudina OG , Shchegolkov EV , Zhilina EF , Astakhova TY , Pronkin PG , Timokhina EN , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ |
| Ref : Eur Journal of Medicinal Chemistry , 303 :118397 , 2025 |
| Abstract : |
| PubMedSearch : Makhaeva_2025_Eur.J.Med.Chem_303_118397 |
| PubMedID: 41338134 |
| Title : Conjugates of amiridine and salicylic derivatives as promising multifunctional CNS agents for potential treatment of Alzheimer's disease - Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819 |
| Author(s) : Makhaeva GF , Grishchenko MV , Kovaleva NV , Boltneva NP , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Lushchekina SV , Khudina OG , Zhilina EF , Shchegolkov EV , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ |
| Ref : Arch Pharm (Weinheim) , 358 :e2400819 , 2025 |
| Abstract : |
| PubMedSearch : Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819 |
| PubMedID: 39686878 |
| Title : Conjugates of amiridine and salicylic derivatives as promising multifunctional CNS agents for potential treatment of Alzheimer's disease - Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819 |
| Author(s) : Makhaeva GF , Grishchenko MV , Kovaleva NV , Boltneva NP , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Lushchekina SV , Khudina OG , Zhilina EF , Shchegolkov EV , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ |
| Ref : Arch Pharm (Weinheim) , 358 :e2400819 , 2025 |
| Abstract : |
| PubMedSearch : Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819 |
| PubMedID: 39686878 |
| Title : Synthesis of Tacrine\/Amiridine Conjugates with Aminomethylidene Derivatives of Trifluoroacetoacetic Ester and their Biological Potential for the Therapy of Alzheimer's Disease - Grishchenko_2025_ChemMedChem__e202500723 |
| Author(s) : Grishchenko MV , Makhaeva GF , Burgart YV , Kovaleva NV , Boltneva NP , Skornyakova TS , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Shchegolkov EV , Saloutin V , Charushin VN |
| Ref : ChemMedChem , :e202500723 , 2025 |
| Abstract : |
| PubMedSearch : Grishchenko_2025_ChemMedChem__e202500723 |
| PubMedID: 41047157 |
| Title : Conjugates of anticholinesterase drugs ipidacrine and tacrine with thiouracils: synthesis and biological properties - Grishchenko_2025_Russ.Chem.Bull_73_3399 |
| Author(s) : Grishchenko MV , Khudina OG , Makhaeva GF , Burgart YV , Kovaleva NV , Rudakova EV , Boltneva NP , Ulitko MV , Saloutin VI , Charushin VN |
| Ref : Russ Chem Bull , 73 :3399 , 2025 |
| Abstract : |
| PubMedSearch : Grishchenko_2025_Russ.Chem.Bull_73_3399 |
| PubMedID: |
| Title : Conjugates of anticholinesterase drugs ipidacrine and tacrine with thiouracils: synthesis and biological properties - Grishchenko_2025_Russ.Chem.Bull_73_3399 |
| Author(s) : Grishchenko MV , Khudina OG , Makhaeva GF , Burgart YV , Kovaleva NV , Rudakova EV , Boltneva NP , Ulitko MV , Saloutin VI , Charushin VN |
| Ref : Russ Chem Bull , 73 :3399 , 2025 |
| Abstract : |
| PubMedSearch : Grishchenko_2025_Russ.Chem.Bull_73_3399 |
| PubMedID: |
| Title : Synthesis, biological evaluation, and in silico studies of pyridoxal-amiridine hybrids as multitargeting anti-Alzheimer's disease agents - Makhaeva_2025_Eur.J.Med.Chem_303_118397 |
| Author(s) : Makhaeva GF , Grishchenko MV , Rudakova EV , Kovaleva NV , Boltneva NP , Skornyakova TS , Khudina OG , Shchegolkov EV , Zhilina EF , Astakhova TY , Pronkin PG , Timokhina EN , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ |
| Ref : Eur Journal of Medicinal Chemistry , 303 :118397 , 2025 |
| Abstract : |
| PubMedSearch : Makhaeva_2025_Eur.J.Med.Chem_303_118397 |
| PubMedID: 41338134 |
| Title : Synthesis of Tacrine\/Amiridine Conjugates with Aminomethylidene Derivatives of Trifluoroacetoacetic Ester and their Biological Potential for the Therapy of Alzheimer's Disease - Grishchenko_2025_ChemMedChem__e202500723 |
| Author(s) : Grishchenko MV , Makhaeva GF , Burgart YV , Kovaleva NV , Boltneva NP , Skornyakova TS , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Shchegolkov EV , Saloutin V , Charushin VN |
| Ref : ChemMedChem , :e202500723 , 2025 |
| Abstract : |
| PubMedSearch : Grishchenko_2025_ChemMedChem__e202500723 |
| PubMedID: 41047157 |
| Title : Conjugates of amiridine and salicylic derivatives as promising multifunctional CNS agents for potential treatment of Alzheimer's disease - Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819 |
| Author(s) : Makhaeva GF , Grishchenko MV , Kovaleva NV , Boltneva NP , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Lushchekina SV , Khudina OG , Zhilina EF , Shchegolkov EV , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ |
| Ref : Arch Pharm (Weinheim) , 358 :e2400819 , 2025 |
| Abstract : |
| PubMedSearch : Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819 |
| PubMedID: 39686878 |
| Title : Synthesis of Tacrine\/Amiridine Conjugates with Aminomethylidene Derivatives of Trifluoroacetoacetic Ester and their Biological Potential for the Therapy of Alzheimer's Disease - Grishchenko_2025_ChemMedChem__e202500723 |
| Author(s) : Grishchenko MV , Makhaeva GF , Burgart YV , Kovaleva NV , Boltneva NP , Skornyakova TS , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Shchegolkov EV , Saloutin V , Charushin VN |
| Ref : ChemMedChem , :e202500723 , 2025 |
| Abstract : |
| PubMedSearch : Grishchenko_2025_ChemMedChem__e202500723 |
| PubMedID: 41047157 |
| Title : Conjugates of Tacrine and Salicylic Acid Derivatives as New Promising Multitarget Agents for Alzheimer's Disease - Makhaeva_2023_Int.J.Mol.Sci_24_2285 |
| Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Grishchenko MV , Lushchekina SV , Astakhova TY , Serebryakova OG , Timokhina EN , Zhilina EF , Shchegolkov EV , Ulitko MV , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Bachurin SO , Richardson RJ |
| Ref : Int J Mol Sci , 24 :2285 , 2023 |
| Abstract : |
| PubMedSearch : Makhaeva_2023_Int.J.Mol.Sci_24_2285 |
| PubMedID: 36768608 |
| Title : Conjugates of amiridine and thiouracil derivatives as effective inhibitors of butyrylcholinesterase with the potential to block beta-amyloid aggregation - Khudina_2023_Arch.Pharm.(Weinheim)__e2300447 |
| Author(s) : Khudina OG , Grishchenko MV , Makhaeva GF , Kovaleva NV , Boltneva NP , Rudakova EV , Lushchekina SV , Shchegolkov EV , Borisevich SS , Burgart YV , Saloutin VI , Charushin VN |
| Ref : Arch Pharm (Weinheim) , :e2300447 , 2023 |
| Abstract : |
| PubMedSearch : Khudina_2023_Arch.Pharm.(Weinheim)__e2300447 |
| PubMedID: 38072670 |
| Title : Conjugates of amiridine and thiouracil derivatives as effective inhibitors of butyrylcholinesterase with the potential to block beta-amyloid aggregation - Khudina_2023_Arch.Pharm.(Weinheim)__e2300447 |
| Author(s) : Khudina OG , Grishchenko MV , Makhaeva GF , Kovaleva NV , Boltneva NP , Rudakova EV , Lushchekina SV , Shchegolkov EV , Borisevich SS , Burgart YV , Saloutin VI , Charushin VN |
| Ref : Arch Pharm (Weinheim) , :e2300447 , 2023 |
| Abstract : |
| PubMedSearch : Khudina_2023_Arch.Pharm.(Weinheim)__e2300447 |
| PubMedID: 38072670 |
| Title : Conjugates of Tacrine and Salicylic Acid Derivatives as New Promising Multitarget Agents for Alzheimer's Disease - Makhaeva_2023_Int.J.Mol.Sci_24_2285 |
| Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Grishchenko MV , Lushchekina SV , Astakhova TY , Serebryakova OG , Timokhina EN , Zhilina EF , Shchegolkov EV , Ulitko MV , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Bachurin SO , Richardson RJ |
| Ref : Int J Mol Sci , 24 :2285 , 2023 |
| Abstract : |
| PubMedSearch : Makhaeva_2023_Int.J.Mol.Sci_24_2285 |
| PubMedID: 36768608 |
| Title : Conjugates of amiridine and thiouracil derivatives as effective inhibitors of butyrylcholinesterase with the potential to block beta-amyloid aggregation - Khudina_2023_Arch.Pharm.(Weinheim)__e2300447 |
| Author(s) : Khudina OG , Grishchenko MV , Makhaeva GF , Kovaleva NV , Boltneva NP , Rudakova EV , Lushchekina SV , Shchegolkov EV , Borisevich SS , Burgart YV , Saloutin VI , Charushin VN |
| Ref : Arch Pharm (Weinheim) , :e2300447 , 2023 |
| Abstract : |
| PubMedSearch : Khudina_2023_Arch.Pharm.(Weinheim)__e2300447 |
| PubMedID: 38072670 |
| Title : Conjugates of Tacrine and Salicylic Acid Derivatives as New Promising Multitarget Agents for Alzheimer's Disease - Makhaeva_2023_Int.J.Mol.Sci_24_2285 |
| Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Grishchenko MV , Lushchekina SV , Astakhova TY , Serebryakova OG , Timokhina EN , Zhilina EF , Shchegolkov EV , Ulitko MV , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Bachurin SO , Richardson RJ |
| Ref : Int J Mol Sci , 24 :2285 , 2023 |
| Abstract : |
| PubMedSearch : Makhaeva_2023_Int.J.Mol.Sci_24_2285 |
| PubMedID: 36768608 |
| Title : New Multifunctional Agents for Potential Alzheimer's Disease Treatment Based on Tacrine Conjugates with 2-Arylhydrazinylidene-1,3-Diketones - Elkina_2022_Biomolecules_12_ |
| Author(s) : Elkina NA , Grishchenko MV , Shchegolkov EV , Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Astakhova TY , Radchenko EV , Palyulin VA , Zhilina EF , Perminova AN , Lapshin LS , Burgart YV , Saloutin VI , Richardson RJ |
| Ref : Biomolecules , 12 : , 2022 |
| Abstract : |
| PubMedSearch : Elkina_2022_Biomolecules_12_ |
| PubMedID: 36358901 |
| Title : Conjugates of Tacrine with Salicylamide as Promising Multitarget Agents for Alzheimer's Disease - Grishchenko_2022_ChemMedChem__e202200080 |
| Author(s) : Grishchenko MV , Makhaeva GF , Burgart YV , Rudakova EV , Boltneva NP , Kovaleva NV , Serebryakova OG , Lushchekina SV , Astakhova TY , Zhilina EF , Shchegolkov EV , Richardson RJ , Saloutin VI |
| Ref : ChemMedChem , :e202200080 , 2022 |
| Abstract : |
| PubMedSearch : Grishchenko_2022_ChemMedChem__e202200080 |
| PubMedID: 35322571 |
| Title : New Multifunctional Agents for Potential Alzheimer's Disease Treatment Based on Tacrine Conjugates with 2-Arylhydrazinylidene-1,3-Diketones - Elkina_2022_Biomolecules_12_ |
| Author(s) : Elkina NA , Grishchenko MV , Shchegolkov EV , Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Astakhova TY , Radchenko EV , Palyulin VA , Zhilina EF , Perminova AN , Lapshin LS , Burgart YV , Saloutin VI , Richardson RJ |
| Ref : Biomolecules , 12 : , 2022 |
| Abstract : |
| PubMedSearch : Elkina_2022_Biomolecules_12_ |
| PubMedID: 36358901 |
| Title : Conjugates of Tacrine with Salicylamide as Promising Multitarget Agents for Alzheimer's Disease - Grishchenko_2022_ChemMedChem__e202200080 |
| Author(s) : Grishchenko MV , Makhaeva GF , Burgart YV , Rudakova EV , Boltneva NP , Kovaleva NV , Serebryakova OG , Lushchekina SV , Astakhova TY , Zhilina EF , Shchegolkov EV , Richardson RJ , Saloutin VI |
| Ref : ChemMedChem , :e202200080 , 2022 |
| Abstract : |
| PubMedSearch : Grishchenko_2022_ChemMedChem__e202200080 |
| PubMedID: 35322571 |
| Title : New Multifunctional Agents for Potential Alzheimer's Disease Treatment Based on Tacrine Conjugates with 2-Arylhydrazinylidene-1,3-Diketones - Elkina_2022_Biomolecules_12_ |
| Author(s) : Elkina NA , Grishchenko MV , Shchegolkov EV , Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Astakhova TY , Radchenko EV , Palyulin VA , Zhilina EF , Perminova AN , Lapshin LS , Burgart YV , Saloutin VI , Richardson RJ |
| Ref : Biomolecules , 12 : , 2022 |
| Abstract : |
| PubMedSearch : Elkina_2022_Biomolecules_12_ |
| PubMedID: 36358901 |
| Title : Conjugates of Tacrine with Salicylamide as Promising Multitarget Agents for Alzheimer's Disease - Grishchenko_2022_ChemMedChem__e202200080 |
| Author(s) : Grishchenko MV , Makhaeva GF , Burgart YV , Rudakova EV , Boltneva NP , Kovaleva NV , Serebryakova OG , Lushchekina SV , Astakhova TY , Zhilina EF , Shchegolkov EV , Richardson RJ , Saloutin VI |
| Ref : ChemMedChem , :e202200080 , 2022 |
| Abstract : |
| PubMedSearch : Grishchenko_2022_ChemMedChem__e202200080 |
| PubMedID: 35322571 |