| Title : Conjugates of anticholinesterase drugs ipidacrine and tacrine with thiouracils: synthesis and biological properties - Grishchenko_2025_Russ.Chem.Bull_73_3399 |
| Author(s) : Grishchenko MV , Khudina OG , Makhaeva GF , Burgart YV , Kovaleva NV , Rudakova EV , Boltneva NP , Ulitko MV , Saloutin VI , Charushin VN |
| Ref : Russ Chem Bull , 73 :3399 , 2025 |
| Abstract : |
| PubMedSearch : Grishchenko_2025_Russ.Chem.Bull_73_3399 |
| PubMedID: |
| Title : Conjugates of amiridine and salicylic derivatives as promising multifunctional CNS agents for potential treatment of Alzheimer's disease - Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819 |
| Author(s) : Makhaeva GF , Grishchenko MV , Kovaleva NV , Boltneva NP , Rudakova EV , Astakhova TY , Timokhina EN , Pronkin PG , Lushchekina SV , Khudina OG , Zhilina EF , Shchegolkov EV , Lapshina MA , Dubrovskaya ES , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Charushin VN , Richardson RJ |
| Ref : Arch Pharm (Weinheim) , 358 :e2400819 , 2025 |
| Abstract : |
| PubMedSearch : Makhaeva_2025_Arch.Pharm.(Weinheim)_358_e2400819 |
| PubMedID: 39686878 |
| Title : 2-Arylhydrazinylidene-3-oxo-3-polyfluoroalkylpropanoic acids as selective and effective carboxylesterase inhibitors with powerful antioxidant potential - Burgart_2024_Bioorg.Med.Chem_115_117938 |
| Author(s) : Burgart YV , Makhaeva GF , Khudina OG , Krasnykh OP , Kovaleva NV , Elkina NA , Boltneva NP , Rudakova EV , Lushchekina SV , Shchegolkov EV , Triandafilova GA , Malysheva KO , Serebryakova OG , Borisevich SS , Ilyina MG , Zhilina EF , Saloutin VI , Charushin VN , Richardson RJ |
| Ref : Bioorganic & Medicinal Chemistry , 115 :117938 , 2024 |
| Abstract : |
| PubMedSearch : Burgart_2024_Bioorg.Med.Chem_115_117938 |
| PubMedID: 39504592 |
| Title : Conjugates of amiridine and thiouracil derivatives as effective inhibitors of butyrylcholinesterase with the potential to block beta-amyloid aggregation - Khudina_2023_Arch.Pharm.(Weinheim)__e2300447 |
| Author(s) : Khudina OG , Grishchenko MV , Makhaeva GF , Kovaleva NV , Boltneva NP , Rudakova EV , Lushchekina SV , Shchegolkov EV , Borisevich SS , Burgart YV , Saloutin VI , Charushin VN |
| Ref : Arch Pharm (Weinheim) , :e2300447 , 2023 |
| Abstract : |
| PubMedSearch : Khudina_2023_Arch.Pharm.(Weinheim)__e2300447 |
| PubMedID: 38072670 |
| Title : Synthesis of 2-arylhydrazinylidene-3-oxo-4,4,4-trifluorobutanoic acids as new selective carboxylesterase inhibitors and radical scavengers - Khudina_2019_Bioorg.Med.Chem.Lett__126716 |
| Author(s) : Khudina OG , Makhaeva GF , Elkina NA , Boltneva NP , Serebryakova OG , Shchegolkov EV , Rudakova EV , Lushchekina SV , Burgart YV , Bachurin SO , Richardson RJ , Saloutin VI |
| Ref : Bioorganic & Medicinal Chemistry Lett , :126716 , 2019 |
| Abstract : |
| PubMedSearch : Khudina_2019_Bioorg.Med.Chem.Lett__126716 |
| PubMedID: 31640885 |