| Title : Novel tacrine-based multi-target directed Ligands: Enhancing cholinesterase inhibition, NMDA receptor antagonism, and CNS bioavailability for Alzheimer's disease treatment - Svobodova_2025_Eur.J.Med.Chem_292_117678 |
| Author(s) : Svobodova B , Moravcova Z , Misiachna A , Novakova G , Marek A , Finger V , Odvarkova J , Pejchal J , Karasova JZ , Netolicky J , Ladislav M , Hrabinova M , Sorf A , Muckova L , Fikejzlova L , Benkova M , Novak M , Prchal L , Capek J , Handl J , Rousar T , Greber KE , Ciura K , Horak M , Soukup O , Korabecny J |
| Ref : Eur Journal of Medicinal Chemistry , 292 :117678 , 2025 |
| Abstract : |
| PubMedSearch : Svobodova_2025_Eur.J.Med.Chem_292_117678 |
| PubMedID: 40288120 |
| Title : Phenoxytacrine derivatives: Low-toxicity neuroprotectants exerting affinity to ifenprodil-binding site and cholinesterase inhibition - Misiachna_2024_Eur.J.Med.Chem_266_116130 |
| Author(s) : Misiachna A , Svobodova B , Netolicky J , Chvojkova M , Kleteckova L , Prchal L , Novak M , Hrabinova M , Kucera T , Muckova L , Moravcova Z , Karasova JZ , Pejchal J , Blazek F , Malinak D , Hakenova K , Krausova BH , Kolcheva M , Ladislav M , Korabecny J , Pahnke J , Vales K , Horak M , Soukup O |
| Ref : Eur Journal of Medicinal Chemistry , 266 :116130 , 2024 |
| Abstract : |
| PubMedSearch : Misiachna_2024_Eur.J.Med.Chem_266_116130 |
| PubMedID: 38218127 |
| Title : Dizocilpine derivatives as neuroprotective NMDA receptor antagonists without psychomimetic side effects - Konecny_2024_Eur.J.Med.Chem_280_116981 |
| Author(s) : Konecny J , Misiachna A , Chvojkova M , Kleteckova L , Kolcheva M , Novak M , Prchal L , Ladislav M , Hemelikova K , Netolicky J , Hrabinova M , Kobrlova T , Karasova JZ , Pejchal J , Fibigar J , Vecera Z , Kucera T , Jendelova P , Zahumenska P , Langore E , Doderovic J , Pang YP , Vales K , Korabecny J , Soukup O , Horak M |
| Ref : Eur Journal of Medicinal Chemistry , 280 :116981 , 2024 |
| Abstract : |
| PubMedSearch : Konecny_2024_Eur.J.Med.Chem_280_116981 |
| PubMedID: 39442339 |
| Title : Palmitoylation Controls NMDA Receptor Function and Steroid Sensitivity - Hubalkova_2021_J.Neurosci_41_2119 |
| Author(s) : Hubalkova P , Ladislav M , Vyklicky V , Smejkalova T , Hrcka Krausova B , Kysilov B , Krusek J , Naimova Z , Korinek M , Chodounska H , Kudova E , Cerny J , Vyklicky L, Jr. |
| Ref : Journal of Neuroscience , 41 :2119 , 2021 |
| Abstract : |
| PubMedSearch : Hubalkova_2021_J.Neurosci_41_2119 |
| PubMedID: 33526476 |