Full name : Fibigar Jakub
First name : Jakub
Mail : University of Defence, Military Faculty of Medicine, Department of Toxicology and Military Pharmacy, Trebesska 1575, 500 01, Hradec Krlove
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Country : Czech Republic
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Comment
| Title : Reactivation screening of A-234-inhibited human recombinant acetylcholinesterase in vitro - Opravil_2025_Chem.Biol.Interact_15ChEPon_423_111810 |
| Author(s) : Opravil J , Pejchal J , Hrabinova M , Muckova L , Prchal L , Korabecny J , Rozsypal T , Gorecki L , Fibigar J , Soukup O , Musilek K , Jun D |
| Ref : Chemico-Biological Interactions , 423 :111810 , 2025 |
| Abstract : |
| PubMedSearch : Opravil_2025_Chem.Biol.Interact_15ChEPon_423_111810 |
| PubMedID: 41197850 |
| Title : Reactivation screening of A-234-inhibited human recombinant acetylcholinesterase in vitro - Opravil_2025_Chem.Biol.Interact_15ChEPon_423_111810 |
| Author(s) : Opravil J , Pejchal J , Hrabinova M , Muckova L , Prchal L , Korabecny J , Rozsypal T , Gorecki L , Fibigar J , Soukup O , Musilek K , Jun D |
| Ref : Chemico-Biological Interactions , 423 :111810 , 2025 |
| Abstract : |
| PubMedSearch : Opravil_2025_Chem.Biol.Interact_15ChEPon_423_111810 |
| PubMedID: 41197850 |
| Title : Reactivation screening of A-234-inhibited human recombinant acetylcholinesterase in vitro - Opravil_2025_Chem.Biol.Interact_15ChEPon_423_111810 |
| Author(s) : Opravil J , Pejchal J , Hrabinova M , Muckova L , Prchal L , Korabecny J , Rozsypal T , Gorecki L , Fibigar J , Soukup O , Musilek K , Jun D |
| Ref : Chemico-Biological Interactions , 423 :111810 , 2025 |
| Abstract : |
| PubMedSearch : Opravil_2025_Chem.Biol.Interact_15ChEPon_423_111810 |
| PubMedID: 41197850 |
| Title : Dizocilpine derivatives as neuroprotective NMDA receptor antagonists without psychomimetic side effects - Konecny_2024_Eur.J.Med.Chem_280_116981 |
| Author(s) : Konecny J , Misiachna A , Chvojkova M , Kleteckova L , Kolcheva M , Novak M , Prchal L , Ladislav M , Hemelikova K , Netolicky J , Hrabinova M , Kobrlova T , Karasova JZ , Pejchal J , Fibigar J , Vecera Z , Kucera T , Jendelova P , Zahumenska P , Langore E , Doderovic J , Pang YP , Vales K , Korabecny J , Soukup O , Horak M |
| Ref : Eur Journal of Medicinal Chemistry , 280 :116981 , 2024 |
| Abstract : |
| PubMedSearch : Konecny_2024_Eur.J.Med.Chem_280_116981 |
| PubMedID: 39442339 |
| Title : Morphing cholinesterase inhibitor amiridine into multipotent drugs for the treatment of Alzheimer's disease - Mezeiova_2024_Biomed.Pharmacother_173_116399 |
| Author(s) : Mezeiova E , Prchal L , Hrabinova M , Muckova L , Pulkrabkova L , Soukup O , Misiachna A , Janousek J , Fibigar J , Kucera T , Horak M , Makhaeva GF , Korabecny J |
| Ref : Biomed Pharmacother , 173 :116399 , 2024 |
| Abstract : |
| PubMedSearch : Mezeiova_2024_Biomed.Pharmacother_173_116399 |
| PubMedID: 38492439 |
| Title : Morphing cholinesterase inhibitor amiridine into multipotent drugs for the treatment of Alzheimer's disease - Mezeiova_2024_Biomed.Pharmacother_173_116399 |
| Author(s) : Mezeiova E , Prchal L , Hrabinova M , Muckova L , Pulkrabkova L , Soukup O , Misiachna A , Janousek J , Fibigar J , Kucera T , Horak M , Makhaeva GF , Korabecny J |
| Ref : Biomed Pharmacother , 173 :116399 , 2024 |
| Abstract : |
| PubMedSearch : Mezeiova_2024_Biomed.Pharmacother_173_116399 |
| PubMedID: 38492439 |
| Title : Carltonine-Derived Compounds for Targeted Butyrylcholinesterase Inhibition - Pidany_2024_RSC.Med.Chem_15_1601 |
| Author(s) : Pidany F , Kroustkova J , Jenco J , Breiterova K , Muckovab L , Novakova L , Kunes J , Fibigar J , Kucera T , Novak M , Sorf A , Hrabinova M , Pulkrabkova L , Janousek J , Soukup O , Jun D , Korabecny J , Cahlikova L |
| Ref : RSC Med Chem , 15 :1601 , 2024 |
| Abstract : |
| PubMedSearch : Pidany_2024_RSC.Med.Chem_15_1601 |
| PubMedID: 38784455 |
| Gene_locus related to this paper: human-BCHE |
| Title : Carltonine-Derived Compounds for Targeted Butyrylcholinesterase Inhibition - Pidany_2024_RSC.Med.Chem_15_1601 |
| Author(s) : Pidany F , Kroustkova J , Jenco J , Breiterova K , Muckovab L , Novakova L , Kunes J , Fibigar J , Kucera T , Novak M , Sorf A , Hrabinova M , Pulkrabkova L , Janousek J , Soukup O , Jun D , Korabecny J , Cahlikova L |
| Ref : RSC Med Chem , 15 :1601 , 2024 |
| Abstract : |
| PubMedSearch : Pidany_2024_RSC.Med.Chem_15_1601 |
| PubMedID: 38784455 |
| Gene_locus related to this paper: human-BCHE |
| Title : Dizocilpine derivatives as neuroprotective NMDA receptor antagonists without psychomimetic side effects - Konecny_2024_Eur.J.Med.Chem_280_116981 |
| Author(s) : Konecny J , Misiachna A , Chvojkova M , Kleteckova L , Kolcheva M , Novak M , Prchal L , Ladislav M , Hemelikova K , Netolicky J , Hrabinova M , Kobrlova T , Karasova JZ , Pejchal J , Fibigar J , Vecera Z , Kucera T , Jendelova P , Zahumenska P , Langore E , Doderovic J , Pang YP , Vales K , Korabecny J , Soukup O , Horak M |
| Ref : Eur Journal of Medicinal Chemistry , 280 :116981 , 2024 |
| Abstract : |
| PubMedSearch : Konecny_2024_Eur.J.Med.Chem_280_116981 |
| PubMedID: 39442339 |
| Title : Carltonine-Derived Compounds for Targeted Butyrylcholinesterase Inhibition - Pidany_2024_RSC.Med.Chem_15_1601 |
| Author(s) : Pidany F , Kroustkova J , Jenco J , Breiterova K , Muckovab L , Novakova L , Kunes J , Fibigar J , Kucera T , Novak M , Sorf A , Hrabinova M , Pulkrabkova L , Janousek J , Soukup O , Jun D , Korabecny J , Cahlikova L |
| Ref : RSC Med Chem , 15 :1601 , 2024 |
| Abstract : |
| PubMedSearch : Pidany_2024_RSC.Med.Chem_15_1601 |
| PubMedID: 38784455 |
| Gene_locus related to this paper: human-BCHE |
| Title : Morphing cholinesterase inhibitor amiridine into multipotent drugs for the treatment of Alzheimer's disease - Mezeiova_2024_Biomed.Pharmacother_173_116399 |
| Author(s) : Mezeiova E , Prchal L , Hrabinova M , Muckova L , Pulkrabkova L , Soukup O , Misiachna A , Janousek J , Fibigar J , Kucera T , Horak M , Makhaeva GF , Korabecny J |
| Ref : Biomed Pharmacother , 173 :116399 , 2024 |
| Abstract : |
| PubMedSearch : Mezeiova_2024_Biomed.Pharmacother_173_116399 |
| PubMedID: 38492439 |
| Title : Dizocilpine derivatives as neuroprotective NMDA receptor antagonists without psychomimetic side effects - Konecny_2024_Eur.J.Med.Chem_280_116981 |
| Author(s) : Konecny J , Misiachna A , Chvojkova M , Kleteckova L , Kolcheva M , Novak M , Prchal L , Ladislav M , Hemelikova K , Netolicky J , Hrabinova M , Kobrlova T , Karasova JZ , Pejchal J , Fibigar J , Vecera Z , Kucera T , Jendelova P , Zahumenska P , Langore E , Doderovic J , Pang YP , Vales K , Korabecny J , Soukup O , Horak M |
| Ref : Eur Journal of Medicinal Chemistry , 280 :116981 , 2024 |
| Abstract : |
| PubMedSearch : Konecny_2024_Eur.J.Med.Chem_280_116981 |
| PubMedID: 39442339 |