Title : Dizocilpine derivatives as neuroprotective NMDA receptor antagonists without psychomimetic side effects - Konecny_2024_Eur.J.Med.Chem_280_116981 |
Author(s) : Konecny J , Misiachna A , Chvojkova M , Kleteckova L , Kolcheva M , Novak M , Prchal L , Ladislav M , Hemelikova K , Netolicky J , Hrabinova M , Kobrlova T , Karasova JZ , Pejchal J , Fibigar J , Vecera Z , Kucera T , Jendelova P , Zahumenska P , Langore E , Doderovic J , Pang YP , Vales K , Korabecny J , Soukup O , Horak M |
Ref : Eur Journal of Medicinal Chemistry , 280 :116981 , 2024 |
Abstract : |
PubMedSearch : Konecny_2024_Eur.J.Med.Chem_280_116981 |
PubMedID: 39442339 |
Title : Phenoxytacrine derivatives: Low-toxicity neuroprotectants exerting affinity to ifenprodil-binding site and cholinesterase inhibition - Misiachna_2024_Eur.J.Med.Chem_266_116130 |
Author(s) : Misiachna A , Svobodova B , Netolicky J , Chvojkova M , Kleteckova L , Prchal L , Novak M , Hrabinova M , Kucera T , Muckova L , Moravcova Z , Karasova JZ , Pejchal J , Blazek F , Malinak D , Hakenova K , Krausova BH , Kolcheva M , Ladislav M , Korabecny J , Pahnke J , Vales K , Horak M , Soukup O |
Ref : Eur Journal of Medicinal Chemistry , 266 :116130 , 2024 |
Abstract : |
PubMedSearch : Misiachna_2024_Eur.J.Med.Chem_266_116130 |
PubMedID: 38218127 |
Title : 7-phenoxytacrine is a dually acting drug with neuroprotective efficacy in vivo - Kaniakova_2021_Biochem.Pharmacol__114460 |
Author(s) : Kaniakova M , Korabecny J , Holubova K , Kleteckova L , Chvojkova M , Hakenova K , Prchal L , Novak M , Dolezal R , Hepnarova V , Svobodova B , Kucera T , Lichnerova K , Krausova B , Horak M , Vales K , Soukup O |
Ref : Biochemical Pharmacology , :114460 , 2021 |
Abstract : |
PubMedSearch : Kaniakova_2021_Biochem.Pharmacol__114460 |
PubMedID: 33571502 |
Title : Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease - Chalupova_2019_Eur.J.Med.Chem_168_491 |
Author(s) : Chalupova K , Korabecny J , Bartolini M , Monti B , Lamba D , Caliandro R , Pesaresi A , Brazzolotto X , Gastellier AJ , Nachon F , Pejchal J , Jarosova M , Hepnarova V , Jun D , Hrabinova M , Dolezal R , Karasova JZ , Mzik M , Kristofikova Z , Misik J , Muckova L , Jost P , Soukup O , Benkova M , Setnicka V , Habartova L , Chvojkova M , Kleteckova L , Vales K , Mezeiova E , Uliassi E , Valis M , Nepovimova E , Bolognesi ML , Kuca K |
Ref : Eur Journal of Medicinal Chemistry , 168 :491 , 2019 |
Abstract : |
PubMedSearch : Chalupova_2019_Eur.J.Med.Chem_168_491 |
PubMedID: 30851693 |
Gene_locus related to this paper: torca-ACHE |
Title : Combination of Memantine and 6-Chlorotacrine as Novel Multi-Target Compound against Alzheimer's Disease - Kaniakova_2019_Curr.Alzheimer.Res_16_821 |
Author(s) : Kaniakova M , Nepovimova E , Kleteckova L , Skrenkova K , Holubova K , Chrienova Z , Hepnarova V , Kucera T , Kobrlova T , Vales K , Korabecny J , Soukup O , Horak M |
Ref : Curr Alzheimer Res , 16 :821 , 2019 |
Abstract : |
PubMedSearch : Kaniakova_2019_Curr.Alzheimer.Res_16_821 |
PubMedID: 30819076 |