Title : Phenoxytacrine derivatives: Low-toxicity neuroprotectants exerting affinity to ifenprodil-binding site and cholinesterase inhibition - Misiachna_2024_Eur.J.Med.Chem_266_116130 |
Author(s) : Misiachna A , Svobodova B , Netolicky J , Chvojkova M , Kleteckova L , Prchal L , Novak M , Hrabinova M , Kucera T , Muckova L , Moravcova Z , Karasova JZ , Pejchal J , Blazek F , Malinak D , Hakenova K , Krausova BH , Kolcheva M , Ladislav M , Korabecny J , Pahnke J , Vales K , Horak M , Soukup O |
Ref : Eur Journal of Medicinal Chemistry , 266 :116130 , 2024 |
Abstract : |
PubMedSearch : Misiachna_2024_Eur.J.Med.Chem_266_116130 |
PubMedID: 38218127 |
Title : Dizocilpine derivatives as neuroprotective NMDA receptor antagonists without psychomimetic side effects - Konecny_2024_Eur.J.Med.Chem_280_116981 |
Author(s) : Konecny J , Misiachna A , Chvojkova M , Kleteckova L , Kolcheva M , Novak M , Prchal L , Ladislav M , Hemelikova K , Netolicky J , Hrabinova M , Kobrlova T , Karasova JZ , Pejchal J , Fibigar J , Vecera Z , Kucera T , Jendelova P , Zahumenska P , Langore E , Doderovic J , Pang YP , Vales K , Korabecny J , Soukup O , Horak M |
Ref : Eur Journal of Medicinal Chemistry , 280 :116981 , 2024 |
Abstract : |
PubMedSearch : Konecny_2024_Eur.J.Med.Chem_280_116981 |
PubMedID: 39442339 |
Title : Pro-cognitive effects of dual tacrine derivatives acting as cholinesterase inhibitors and NMDA receptor antagonists - Chvojkova_2024_Biomed.Pharmacother_176_116821 |
Author(s) : Chvojkova M , Kolar D , Kovacova K , Cejkova L , Misiachna A , Hakenova K , Gorecki L , Horak M , Korabecny J , Soukup O , Vales K |
Ref : Biomed Pharmacother , 176 :116821 , 2024 |
Abstract : |
PubMedSearch : Chvojkova_2024_Biomed.Pharmacother_176_116821 |
PubMedID: 38823278 |
Title : Morphing cholinesterase inhibitor amiridine into multipotent drugs for the treatment of Alzheimer's disease - Mezeiova_2024_Biomed.Pharmacother_173_116399 |
Author(s) : Mezeiova E , Prchal L , Hrabinova M , Muckova L , Pulkrabkova L , Soukup O , Misiachna A , Janousek J , Fibigar J , Kucera T , Horak M , Makhaeva GF , Korabecny J |
Ref : Biomed Pharmacother , 173 :116399 , 2024 |
Abstract : |
PubMedSearch : Mezeiova_2024_Biomed.Pharmacother_173_116399 |
PubMedID: 38492439 |
Title : Structure-Guided Design of N-Methylpropargylamino-Quinazoline Derivatives as Multipotent Agents for the Treatment of Alzheimer's Disease - Svobodova_2023_Int.J.Mol.Sci_24_ |
Author(s) : Svobodova B , Pulkrabkova L , Panek D , Misiachna A , Kolcheva M , Andrys R , Handl J , Capek J , Nyvltova P , Rousar T , Prchal L , Hepnarova V , Hrabinova M , Muckova L , Tosnerova D , Karabanovich G , Finger V , Soukup O , Horak M , Korabecny J |
Ref : Int J Mol Sci , 24 : , 2023 |
Abstract : |
PubMedSearch : Svobodova_2023_Int.J.Mol.Sci_24_ |
PubMedID: 37298087 |
Title : Structure-activity relationships of dually-acting acetylcholinesterase inhibitors derived from tacrine on N-methyl-d-Aspartate receptors - Gorecki_2021_Eur.J.Med.Chem_219_113434 |
Author(s) : Gorecki L , Misiachna A , Damborsky J , Dolezal R , Korabecny J , Cejkova L , Hakenova K , Chvojkova M , Karasova JZ , Prchal L , Novak M , Kolcheva M , Kortus S , Vales K , Horak M , Soukup O |
Ref : Eur Journal of Medicinal Chemistry , 219 :113434 , 2021 |
Abstract : |
PubMedSearch : Gorecki_2021_Eur.J.Med.Chem_219_113434 |
PubMedID: 33892271 |
Title : Pursuing the Complexity of Alzheimer's Disease: Discovery of Fluoren-9-Amines as Selective Butyrylcholinesterase Inhibitors and N-Methyl-d-Aspartate Receptor Antagonists - Konecny_2020_Biomolecules_11_ |
Author(s) : Konecny J , Misiachna A , Hrabinova M , Pulkrabkova L , Benkova M , Prchal L , Kucera T , Kobrlova T , Finger V , Kolcheva M , Kortus S , Jun D , Valko M , Horak M , Soukup O , Korabecny J |
Ref : Biomolecules , 11 : , 2020 |
Abstract : |
PubMedSearch : Konecny_2020_Biomolecules_11_ |
PubMedID: 33375115 |