| Title : Carltonine B derivatives: Synthesis and structure-activity relationship insights for selective butyrylcholinesterase inhibition - Al Mamun_2026_Bioorg.Chem_177_109894 |
| Author(s) : Al Mamun A , Konecny J , Hrabinova M , Sorf A , Muckova L , Fibigar J , Kucera T , Pulkrabkova L , Jun D , Prchal L , Panek D , Finger V , Soukup O , Cailly T , Collot V , Novakova L , Cahlikova L , Korabecny J |
| Ref : Bioorg Chem , 177 :109894 , 2026 |
| Abstract : |
| PubMedSearch : Al Mamun_2026_Bioorg.Chem_177_109894 |
| PubMedID: 42060983 |
| Title : Novel tacrine-based multi-target directed Ligands: Enhancing cholinesterase inhibition, NMDA receptor antagonism, and CNS bioavailability for Alzheimer's disease treatment - Svobodova_2025_Eur.J.Med.Chem_292_117678 |
| Author(s) : Svobodova B , Moravcova Z , Misiachna A , Novakova G , Marek A , Finger V , Odvarkova J , Pejchal J , Karasova JZ , Netolicky J , Ladislav M , Hrabinova M , Sorf A , Muckova L , Fikejzlova L , Benkova M , Novak M , Prchal L , Capek J , Handl J , Rousar T , Greber KE , Ciura K , Horak M , Soukup O , Korabecny J |
| Ref : Eur Journal of Medicinal Chemistry , 292 :117678 , 2025 |
| Abstract : |
| PubMedSearch : Svobodova_2025_Eur.J.Med.Chem_292_117678 |
| PubMedID: 40288120 |
| Title : Carltonine-Derived Compounds for Targeted Butyrylcholinesterase Inhibition - Pidany_2024_RSC.Med.Chem_15_1601 |
| Author(s) : Pidany F , Kroustkova J , Jenco J , Breiterova K , Muckovab L , Novakova L , Kunes J , Fibigar J , Kucera T , Novak M , Sorf A , Hrabinova M , Pulkrabkova L , Janousek J , Soukup O , Jun D , Korabecny J , Cahlikova L |
| Ref : RSC Med Chem , 15 :1601 , 2024 |
| Abstract : |
| PubMedSearch : Pidany_2024_RSC.Med.Chem_15_1601 |
| PubMedID: 38784455 |
| Gene_locus related to this paper: human-BCHE |
| Title : Multifunctional, fluorene-based modulator of cholinergic and GABAergic neurotransmission as a novel drug candidate for palliative treatment of Alzheimer's disease - Panek_2024_Angew.Chem.Int.Ed.Engl__e202420510 |
| Author(s) : Panek D , Pasieka A , Jonczyk JJ , Gawlinska M , Zareba P , Siwek A , Wolak M , Mordyl B , Gluch-Lutwin M , Latacz G , Brazzolotto X , Chantegreil F , Nachon F , Karasova JZ , Pejchal J , Mzik M , Sestak V , Prchal L , Odvarkova J , Soukup O , Korabecny J , Sorf A , Hamsikova M , Zemanova L , Muckova L , Vanova N , Dryja P , Salat K , Hofner G , Wanner K , Wieckowska A , Malawska B |
| Ref : Angew Chem Int Ed Engl , :e202420510 , 2024 |
| Abstract : |
| PubMedSearch : Panek_2024_Angew.Chem.Int.Ed.Engl__e202420510 |
| PubMedID: 39523866 |
| Gene_locus related to this paper: human-BCHE |
| Title : Differentiated SH-SY5Y neuroblastoma cells as a model for evaluation of nerve agent-associated neurotoxicity - Pulkrabkova_2023_Arch.Toxicol__ |
| Author(s) : Pulkrabkova L , Muckova L , Hrabinova M , Sorf A , Kobrlova T , Jost P , Bezdekova D , Korabecny J , Jun D , Soukup O |
| Ref : Archives of Toxicology , : , 2023 |
| Abstract : |
| PubMedSearch : Pulkrabkova_2023_Arch.Toxicol__ |
| PubMedID: 37221426 |
| Title : In vitro and in silico Evaluation of Non-Quaternary Reactivators of AChE as Antidotes of Organophosphorus Poisoning - a New Hope or a Blind Alley? - Soukup_2018_Med.Chem_14_281 |
| Author(s) : Soukup O , Korabecny J , Malinak D , Nepovimova E , Pham NL , Musilek K , Hrabinova M , Hepnarova V , Dolezal R , Pavek P , Jost P , Kobrlova T , Jankockova J , Gorecki L , Psotka M , Nguyen TD , Box K , Outhwaite B , Ceckova M , Sorf A , Jun D , Kuca K |
| Ref : Med Chem , 14 :281 , 2018 |
| Abstract : |
| PubMedSearch : Soukup_2018_Med.Chem_14_281 |
| PubMedID: 29332594 |