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Title : Carltonine-Derived Compounds for Targeted Butyrylcholinesterase Inhibition - Pidany_2024_RSC.Med.Chem__ |
Author(s) : Pidany F , Kroustkova J , Jenco J , Breiterova K , Muckovab L , Novakova L , Kunes J , Fibigar J , Kucera T , Novak M , Sorf A , Hrabinova M , Pulkrabkova L , Janousek J , Soukup O , Jun D , Korabecny J , Cahlikova L |
Ref : RSC Med Chem , : , 2024 |
Abstract : Pidany_2024_RSC.Med.Chem__ |
ESTHER : Pidany_2024_RSC.Med.Chem__ |
PubMedSearch : Pidany_2024_RSC.Med.Chem__ |
PubMedID: |
Title : Phenoxytacrine derivatives: Low-toxicity neuroprotectants exerting affinity to ifenprodil-binding site and cholinesterase inhibition - Misiachna_2024_Eur.J.Med.Chem_266_116130 |
Author(s) : Misiachna A , Svobodova B , Netolicky J , Chvojkova M , Kleteckova L , Prchal L , Novak M , Hrabinova M , Kucera T , Muckova L , Moravcova Z , Karasova JZ , Pejchal J , Blazek F , Malinak D , Hakenova K , Krausova BH , Kolcheva M , Ladislav M , Korabecny J , Pahnke J , Vales K , Horak M , Soukup O |
Ref : Eur Journal of Medicinal Chemistry , 266 :116130 , 2024 |
Abstract : Misiachna_2024_Eur.J.Med.Chem_266_116130 |
ESTHER : Misiachna_2024_Eur.J.Med.Chem_266_116130 |
PubMedSearch : Misiachna_2024_Eur.J.Med.Chem_266_116130 |
PubMedID: 38218127 |
Title : Differences in the Time Course of Recovery from Brain and Liver Dysfunction in Conventional Long-Term Treatment of Wilson Disease - Hefter_2023_J.Clin.Med_12_ |
Author(s) : Hefter H , Kruschel TS , Novak M , Rosenthal D , Luedde T , Meuth SG , Albrecht P , Hartmann CJ , Samadzadeh S |
Ref : J Clin Med , 12 : , 2023 |
Abstract : Hefter_2023_J.Clin.Med_12_ |
ESTHER : Hefter_2023_J.Clin.Med_12_ |
PubMedSearch : Hefter_2023_J.Clin.Med_12_ |
PubMedID: 37510976 |
Title : Sustainable ionic liquids-based molecular platforms for designing acetylcholinesterase reactivators - Kapitanov_2023_Chem.Biol.Interact_14ChEPon_110735 |
Author(s) : Kapitanov IV , Spulak M , Pour M , Soukup O , Marek J , Jun D , Novak M , Diz de Almeida JSF , Costa Franca TC , Gathergood N , Kuca K , Karpichev Y |
Ref : Chemico-Biological Interactions , :110735 , 2023 |
Abstract : Kapitanov_2023_Chem.Biol.Interact_14ChEPon_110735 |
ESTHER : Kapitanov_2023_Chem.Biol.Interact_14ChEPon_110735 |
PubMedSearch : Kapitanov_2023_Chem.Biol.Interact_14ChEPon_110735 |
PubMedID: 37802409 |
Title : Tacrine First-Phase Biotransformation and Associated Hepatotoxicity: A Possible Way to Avoid Quinone Methide Formation - Novak_2023_ACS.Chem.Biol_18_1993 |
Author(s) : Novak M , Vajrychova M , Koutsilieri S , Sismanoglou DC , Kobrlova T , Prchal L , Svobodova B , Korabecny J , Zarybnicky T , Raisova-Stuchlikova L , Skalova L , Lauschke VM , Kucera R , Soukup O |
Ref : ACS Chemical Biology , 18 :1993 , 2023 |
Abstract : Novak_2023_ACS.Chem.Biol_18_1993 |
ESTHER : Novak_2023_ACS.Chem.Biol_18_1993 |
PubMedSearch : Novak_2023_ACS.Chem.Biol_18_1993 |
PubMedID: 37622522 |
Title : UHPLC-Orbitrap study of the first phase tacrine in vitro metabolites and related Alzheimer's drug candidates using human liver microsomes - Novak_2023_J.Pharm.Biomed.Anal_224_115154 |
Author(s) : Novak M , Svobodova B , Konecny J , Kuratkova A , Nevosadova L , Prchal L , Korabecny J , Lauschke VM , Soukup O , Kucera R |
Ref : J Pharm Biomed Anal , 224 :115154 , 2023 |
Abstract : Novak_2023_J.Pharm.Biomed.Anal_224_115154 |
ESTHER : Novak_2023_J.Pharm.Biomed.Anal_224_115154 |
PubMedSearch : Novak_2023_J.Pharm.Biomed.Anal_224_115154 |
PubMedID: 36442458 |
Title : Cholinesterase Deficiency Syndrome-A Pitfall in the Use of Butyrylcholinesterase as a Biomarker for Wilson's Disease - Arslan_2022_Biomolecules_12_ |
Author(s) : Arslan M , Novak M , Rosenthal D , Hartmann CJ , Albrecht P , Samadzadeh S , Hefter H |
Ref : Biomolecules , 12 : , 2022 |
Abstract : Arslan_2022_Biomolecules_12_ |
ESTHER : Arslan_2022_Biomolecules_12_ |
PubMedSearch : Arslan_2022_Biomolecules_12_ |
PubMedID: 36291607 |
Title : Pseudocholinesterase as a Biomarker for Untreated Wilson's Disease - Hefter_2022_Biomolecules_12_ |
Author(s) : Hefter H , Arslan M , Kruschel TS , Novak M , Rosenthal D , Meuth SG , Albrecht P , Hartmann CJ , Samadzadeh S |
Ref : Biomolecules , 12 : , 2022 |
Abstract : Hefter_2022_Biomolecules_12_ |
ESTHER : Hefter_2022_Biomolecules_12_ |
PubMedSearch : Hefter_2022_Biomolecules_12_ |
PubMedID: 36551217 |
Title : Structure-activity relationships of dually-acting acetylcholinesterase inhibitors derived from tacrine on N-methyl-d-Aspartate receptors - Gorecki_2021_Eur.J.Med.Chem_219_113434 |
Author(s) : Gorecki L , Misiachna A , Damborsky J , Dolezal R , Korabecny J , Cejkova L , Hakenova K , Chvojkova M , Karasova JZ , Prchal L , Novak M , Kolcheva M , Kortus S , Vales K , Horak M , Soukup O |
Ref : Eur Journal of Medicinal Chemistry , 219 :113434 , 2021 |
Abstract : Gorecki_2021_Eur.J.Med.Chem_219_113434 |
ESTHER : Gorecki_2021_Eur.J.Med.Chem_219_113434 |
PubMedSearch : Gorecki_2021_Eur.J.Med.Chem_219_113434 |
PubMedID: 33892271 |
Title : 7-phenoxytacrine is a dually acting drug with neuroprotective efficacy in vivo - Kaniakova_2021_Biochem.Pharmacol__114460 |
Author(s) : Kaniakova M , Korabecny J , Holubova K , Kleteckova L , Chvojkova M , Hakenova K , Prchal L , Novak M , Dolezal R , Hepnarova V , Svobodova B , Kucera T , Lichnerova K , Krausova B , Horak M , Vales K , Soukup O |
Ref : Biochemical Pharmacology , :114460 , 2021 |
Abstract : Kaniakova_2021_Biochem.Pharmacol__114460 |
ESTHER : Kaniakova_2021_Biochem.Pharmacol__114460 |
PubMedSearch : Kaniakova_2021_Biochem.Pharmacol__114460 |
PubMedID: 33571502 |