Histamine-Receptor3-H3-Antagonist

General

Not an alpha/beta hydrolase target but can be used as a building block for larger inhibitors of enzymes of the family designed as multitarget compounds

Inhibitor	Main targeted enzyme families	Type
Contilistat		Multitarget Histamine-Receptor3-H3-Antagonist Monoamine-oxidase-inhibitor Piperidine Indole HDAC inhibitor prop-2-yn-1-yl
ADS031	ACHE	Histamine-Receptor3-H3-Antagonist Multitarget Piperidine Naphthalen
CHEMBL459756	ACHE BCHE	Histamine-Receptor3-H3-Antagonist Multitarget Piperidine
FUB833	ACHE BCHE	Acridine Derivative of Tacrine Alkyl linked bis-ligand Histamine-Receptor3-H3-Antagonist Multitarget Piperidine
11a-quinoxaline	ACHE BCHE Cholinesterase	Multitarget Histamine-Receptor3-H3-Antagonist Quinoxaline
18-E100	ACHE BCHE Cholinesterase	Multitarget Azepane Histamine-Receptor3-H3-Antagonist
UW-MD-71	ACHE BCHE Cholinesterase	Piperidine Quinazoline Multitarget Histamine-Receptor3-H3-Antagonist
Contilisant	ACHE BCHE	Multitarget Histamine-Receptor3-H3-Antagonist Monoamine-oxidase-inhibitor Piperidine Indole prop-2-yn-1-yl