1. Home
  2. Type Inhibitor
  3. Quinazoline

Quinazoline

General

Building block for many inhibitors of enzymes
Inhibitor Main targeted enzyme families Type Structure
CHEMBL5854413 Monoglyceridelipase_lysophospholip Quinazoline Piperazine Benzoxazol Pyridine
CHEMBL467760 BCHE ACHE Quinazoline Alkyl linked bis-ligand Derivative of Amiridine Organochlorine
CHEMBL213889 BCHE Quinazoline Alkyl linked bis-ligand Azocine
CHEMBL466338 BCHE ACHE Quinazoline Multitarget Antioxidant Sulfur Compound Alkyl linked bis-ligand Dithiolane Derivative of Amiridine Organochlorine
CHEMBL466339 BCHE Quinazoline Multitarget Antioxidant Sulfur Compound Alkyl linked bis-ligand Dithiolane Azocine
VAV-8 ACHE Monoamine-oxidase-inhibitor Multitarget Morpholine Quinazoline Piperidine Alkyne
VAV-19 ACHE Monoamine-oxidase-inhibitor Multitarget Quinazoline Piperazine Alkyne
Terazosin Monoglyceridelipase_lysophospholip Not AlphaBeta Hydrolase target Drug Quinazoline Piperazine Sulfur Compound Adrenergic-Receptor-ligand
KV-1131 ACHE Monoamine-oxidase-inhibitor Multitarget Quinazoline Sulfur Compound Morpholine
KV-1234 ACHE Monoamine-oxidase-inhibitor Multitarget Quinazoline Pyrrolidine
Cyanophenyl-quinazolinthioacetamide-Cpd3e ACHE Quinazoline Sulfur Compound Cyanide
3-(Dimethylamino)-N-propanamide-Tryptanthrin ACHE Derivative of Deoxyvasicinone Quinazoline Indole
CHEMBL4207101 BCHE ACHE Derivative of Deoxyvasicinone Quinazoline Metal ion chelator
Dihydroquinazoline-carboxamide-34 Epoxide_hydrolase Carboxamide Multitarget 5-Lipoxygenase inhibitor Sulfur Compound Quinazoline Organochlorine
3-(Quinazolin-4-ylthio)propanoic-acid Pectinacetylesterase-Notum Fragment inhibitor of Notum Sulfur Compound Quinazoline
CHEMBL2152538 Not AlphaBeta Hydrolase target Isoquinoline Quinazoline Leaving group
Tetracyclic-carbamate-cp8 BCHE PET probe Carbamate Natural_modified Derivative of Evodiamine Isoquinoline Quinazoline
Tetracyclic-carbamate-melatonine-3c BCHE Carbamate Natural_modified Derivative of Evodiamine Isoquinoline Quinazoline Derivative of Tryptamine Indole Alkyl linked bis-ligand
Tetracyclic-carbamate-ferulicacid-4a BCHE Carbamate Natural_modified Derivative of Evodiamine Isoquinoline Quinazoline Feruloyl Antioxidant Alkyl linked bis-ligand
Tetracyclic-carbamate-UW-MD-95 BCHE Carbamate Natural_modified Derivative of Evodiamine Isoquinoline Quinazoline
CHEMBL4454960 BCHE Morpholine Isoquinoline Carbamate Quinazoline
75M-5T4F DPP4N_Peptidase_S9 Piperidine Quinazoline Cyanide Purine Alkyne
75L-5T4E DPP4N_Peptidase_S9 Piperidine Pyrimidine Quinazoline Purine Alkyne
75N-5T4B DPP4N_Peptidase_S9 Piperidine Quinazoline Purine Alkyne
UW-MD-71 ACHE BCHE Cholinesterase Piperidine Quinazoline Multitarget Histamine-Receptor3-H3-Antagonist
QADD2 RsbQ-like Quinazoline
Tetracyclic-carbamate-photoswitch-azo BCHE Carbamate Natural_modified Derivative of Evodiamine Isoquinoline Quinazoline Photoswitch
5ALR-8TM Epoxide_hydrolase Sulfur Compound Trifluoro Quinazoline
Linagliptin DPP4N_Peptidase_S9 Drug Purine Gliptin Quinazoline Alkyne
Quinazolin-carbamate-2p BCHE Quinazoline Carbamate Sulfur Compound Thiophen
CI-1002 ACHE Derivative of Tacrine Acridine Muscarinic antagonist Quinazoline Azepane Organochlorine
Desoxypeganine ACHE BCHE Not AlphaBeta Hydrolase target beta-carboline Natural Alkaloid Quinazoline
CHEMBL5854413 Monoglyceridelipase_lysophospholip Quinazoline Piperazine Benzoxazol Pyridine
CHEMBL467760 BCHE ACHE Quinazoline Alkyl linked bis-ligand Derivative of Amiridine Organochlorine
CHEMBL213889 BCHE Quinazoline Alkyl linked bis-ligand Azocine
CHEMBL466338 BCHE ACHE Quinazoline Multitarget Antioxidant Sulfur compound Alkyl linked bis-ligand Dithiolane Derivative of Amiridine Organochlorine
CHEMBL466339 BCHE Quinazoline Multitarget Antioxidant Sulfur compound Alkyl linked bis-ligand Dithiolane Azocine
VAV-8 ACHE Monoamine-oxidase-inhibitor Multitarget Morpholine Quinazoline Piperidine Alkyne
VAV-19 ACHE Monoamine-oxidase-inhibitor Multitarget Quinazoline Piperazine Alkyne
Terazosin Monoglyceridelipase_lysophospholip Not AlphaBeta Hydrolase target Drug Quinazoline Piperazine Sulfur compound Adrenergic-Receptor-ligand
KV-1131 ACHE Monoamine-oxidase-inhibitor Multitarget Quinazoline Sulfur compound Morpholine
KV-1234 ACHE Monoamine-oxidase-inhibitor Multitarget Quinazoline Pyrrolidine
Cyanophenyl-quinazolinthioacetamide-Cpd3e ACHE Quinazoline Sulfur compound Cyanide
3-(Dimethylamino)-N-propanamide-Tryptanthrin ACHE Derivative of Deoxyvasicinone Quinazoline Indole
CHEMBL4207101 BCHE ACHE Derivative of Deoxyvasicinone Quinazoline Metal ion chelator
Dihydroquinazoline-carboxamide-34 Epoxide_hydrolase Carboxamide Multitarget 5-Lipoxygenase inhibitor Sulfur compound Quinazoline Organochlorine
3-(Quinazolin-4-ylthio)propanoic-acid Pectinacetylesterase-Notum Fragment inhibitor of Notum Sulfur compound Quinazoline
CHEMBL2152538 Not AlphaBeta Hydrolase target Isoquinoline Quinazoline Leaving group
Tetracyclic-carbamate-cp8 BCHE PET probe Carbamate Natural_modified Derivative of Evodiamine Isoquinoline Quinazoline
Tetracyclic-carbamate-melatonine-3c BCHE Carbamate Natural_modified Derivative of Evodiamine Isoquinoline Quinazoline Derivative of Tryptamine Indole Alkyl linked bis-ligand
Tetracyclic-carbamate-ferulicacid-4a BCHE Carbamate Natural_modified Derivative of Evodiamine Isoquinoline Quinazoline Feruloyl Antioxidant Alkyl linked bis-ligand
Tetracyclic-carbamate-UW-MD-95 BCHE Carbamate Natural_modified Derivative of Evodiamine Isoquinoline Quinazoline
CHEMBL4454960 BCHE Morpholine Isoquinoline Carbamate Quinazoline
75M-5T4F DPP4N_Peptidase_S9 Piperidine Quinazoline Cyanide Purine Alkyne
75L-5T4E DPP4N_Peptidase_S9 Piperidine Pyrimidine Quinazoline Purine Alkyne
75N-5T4B DPP4N_Peptidase_S9 Piperidine Quinazoline Purine Alkyne
UW-MD-71 ACHE BCHE Cholinesterase Piperidine Quinazoline Multitarget Histamine-Receptor3-H3-Antagonist
QADD2 RsbQ-like Quinazoline
Tetracyclic-carbamate-photoswitch-azo BCHE Carbamate Natural_modified Derivative of Evodiamine Isoquinoline Quinazoline Photoswitch
5ALR-8TM Epoxide_hydrolase Sulfur compound Trifluoro Quinazoline
Linagliptin DPP4N_Peptidase_S9 Drug Purine Gliptin Quinazoline Alkyne
Quinazolin-carbamate-2p BCHE Quinazoline Carbamate Sulfur compound Thiophen
CI-1002 ACHE Derivative of Tacrine Acridine Muscarinic antagonist Quinazoline Azepane Organochlorine
Desoxypeganine ACHE BCHE Not AlphaBeta Hydrolase target beta-carboline Natural Alkaloid Quinazoline
CHEMBL5854413 Monoglyceridelipase_lysophospholip Quinazoline Piperazine Benzoxazol Pyridine
CHEMBL467760 BCHE ACHE Quinazoline Alkyl linked bis-ligand Derivative of Amiridine Organochlorine
CHEMBL213889 BCHE Quinazoline Alkyl linked bis-ligand Azocine
CHEMBL466338 BCHE ACHE Quinazoline Multitarget Antioxidant Sulfur compound Alkyl linked bis-ligand Dithiolane Derivative of Amiridine Organochlorine
CHEMBL466339 BCHE Quinazoline Multitarget Antioxidant Sulfur compound Alkyl linked bis-ligand Dithiolane Azocine
VAV-8 ACHE Monoamine-oxidase-inhibitor Multitarget Morpholine Quinazoline Piperidine Alkyne
VAV-19 ACHE Monoamine-oxidase-inhibitor Multitarget Quinazoline Piperazine Alkyne
Terazosin Monoglyceridelipase_lysophospholip Not AlphaBeta Hydrolase target Drug Quinazoline Piperazine Sulfur compound Adrenergic-Receptor-ligand
KV-1131 ACHE Monoamine-oxidase-inhibitor Multitarget Quinazoline Sulfur compound Morpholine
KV-1234 ACHE Monoamine-oxidase-inhibitor Multitarget Quinazoline Pyrrolidine
Cyanophenyl-quinazolinthioacetamide-Cpd3e ACHE Quinazoline Sulfur compound Cyanide
3-(Dimethylamino)-N-propanamide-Tryptanthrin ACHE Derivative of Deoxyvasicinone Quinazoline Indole
CHEMBL4207101 BCHE ACHE Derivative of Deoxyvasicinone Quinazoline Metal ion chelator
Dihydroquinazoline-carboxamide-34 Epoxide_hydrolase Carboxamide Multitarget 5-Lipoxygenase inhibitor Sulfur compound Quinazoline Organochlorine
3-(Quinazolin-4-ylthio)propanoic-acid Pectinacetylesterase-Notum Fragment inhibitor of Notum Sulfur compound Quinazoline
CHEMBL2152538 Not AlphaBeta Hydrolase target Isoquinoline Quinazoline Leaving group
Tetracyclic-carbamate-cp8 BCHE PET probe Carbamate Natural_modified Derivative of Evodiamine Isoquinoline Quinazoline
Tetracyclic-carbamate-melatonine-3c BCHE Carbamate Natural_modified Derivative of Evodiamine Isoquinoline Quinazoline Derivative of Tryptamine Indole Alkyl linked bis-ligand
Tetracyclic-carbamate-ferulicacid-4a BCHE Carbamate Natural_modified Derivative of Evodiamine Isoquinoline Quinazoline Feruloyl Antioxidant Alkyl linked bis-ligand
Tetracyclic-carbamate-UW-MD-95 BCHE Carbamate Natural_modified Derivative of Evodiamine Isoquinoline Quinazoline
CHEMBL4454960 BCHE Morpholine Isoquinoline Carbamate Quinazoline
75M-5T4F DPP4N_Peptidase_S9 Piperidine Quinazoline Cyanide Purine Alkyne
75L-5T4E DPP4N_Peptidase_S9 Piperidine Pyrimidine Quinazoline Purine Alkyne
75N-5T4B DPP4N_Peptidase_S9 Piperidine Quinazoline Purine Alkyne
UW-MD-71 ACHE BCHE Cholinesterase Piperidine Quinazoline Multitarget Histamine-Receptor3-H3-Antagonist
QADD2 RsbQ-like Quinazoline
Tetracyclic-carbamate-photoswitch-azo BCHE Carbamate Natural_modified Derivative of Evodiamine Isoquinoline Quinazoline Photoswitch
5ALR-8TM Epoxide_hydrolase Sulfur compound Trifluoro Quinazoline
Linagliptin DPP4N_Peptidase_S9 Drug Purine Gliptin Quinazoline Alkyne
Quinazolin-carbamate-2p BCHE Quinazoline Carbamate Sulfur compound Thiophen
CI-1002 ACHE Derivative of Tacrine Acridine Muscarinic antagonist Quinazoline Azepane Organochlorine
Desoxypeganine ACHE BCHE Not AlphaBeta Hydrolase target beta-carboline Natural Alkaloid Quinazoline