Title : Discovery of 4-benzylpiperazinequinoline BChE inhibitor that suppresses neuroinflammation for the treatment of Alzheimer's disease - Chen_2024_Eur.J.Med.Chem_272_116463 |
Author(s) : Chen Y , Zhang W , Li Q , Xie H , Xing S , Lu X , Lyu W , Xiong B , Wang Y , Qu W , Liu W , Chi H , Zhang X , Feng F , Sun H |
Ref : Eur Journal of Medicinal Chemistry , 272 :116463 , 2024 |
Abstract : |
PubMedSearch : Chen_2024_Eur.J.Med.Chem_272_116463 |
PubMedID: 38704944 |
Title : Prognostic and Immunological Roles of CES2 in Breast Cancer and Potential Application of CES2-Targeted Fluorescent Probe DDAB in Breast Surgery - Qu_2023_Int.J.Gen.Med_16_1567 |
Author(s) : Qu W , Yao Y , Liu Y , Jo H , Zhang Q , Zhao H |
Ref : Int J Gen Med , 16 :1567 , 2023 |
Abstract : |
PubMedSearch : Qu_2023_Int.J.Gen.Med_16_1567 |
PubMedID: 37139258 |
Gene_locus related to this paper: human-CES2 |
Title : Design, synthesis and evaluation of fused hybrids with acetylcholinesterase inhibiting and Nrf2 activating functions for Alzheimer's disease - Wang_2022_Eur.J.Med.Chem_244_114806 |
Author(s) : Wang Y , Xiong B , Lin H , Li Q , Yang H , Qiao Y , Xu Z , Lyu W , Qu W , Liu W , Chen Y , Feng F , Sun H |
Ref : Eur Journal of Medicinal Chemistry , 244 :114806 , 2022 |
Abstract : |
PubMedSearch : Wang_2022_Eur.J.Med.Chem_244_114806 |
PubMedID: 36223681 |
Title : Design, synthesis and biological evaluation of novel carboline-cinnamic acid hybrids as multifunctional agents for treatment of Alzheimer's disease - Liao_2020_Bioorg.Chem_99_103844 |
Author(s) : Liao Q , Li Q , Zhao Y , Jiang P , Yan Y , Sun H , Liu W , Feng F , Qu W |
Ref : Bioorg Chem , 99 :103844 , 2020 |
Abstract : |
PubMedSearch : Liao_2020_Bioorg.Chem_99_103844 |
PubMedID: 32325336 |
Title : Rational design and biological evaluation of a new class of thiazolopyridyl tetrahydroacridines as cholinesterase and GSK-3 dual inhibitors for Alzheimer's disease - Jiang_2020_Eur.J.Med.Chem_207_112751 |
Author(s) : Jiang X , Zhou J , Wang Y , Chen L , Duan Y , Huang J , Liu C , Chen Y , Liu W , Sun H , Feng F , Qu W |
Ref : Eur Journal of Medicinal Chemistry , 207 :112751 , 2020 |
Abstract : |
PubMedSearch : Jiang_2020_Eur.J.Med.Chem_207_112751 |
PubMedID: 32950908 |
Title : Effects of Picrasma quassioides and its active constituents on Alzheimer's disease in vitro and in vivo - Guo_2019_Bioorg.Chem_92_103258 |
Author(s) : Guo E , Hu Y , Du T , Zhu H , Chen L , Qu W , Zhang J , Xie N , Liu W , Feng F , Xu J |
Ref : Bioorg Chem , 92 :103258 , 2019 |
Abstract : |
PubMedSearch : Guo_2019_Bioorg.Chem_92_103258 |
PubMedID: 31520892 |
Title : Design, synthesis, biological evaluation, and molecular modeling studies of quinoline-ferulic acid hybrids as cholinesterase inhibitors - Mo_2019_Bioorg.Chem_93_103310 |
Author(s) : Mo J , Yang H , Chen T , Li Q , Lin H , Feng F , Liu W , Qu W , Guo Q , Chi H , Chen Y , Sun H |
Ref : Bioorg Chem , 93 :103310 , 2019 |
Abstract : |
PubMedSearch : Mo_2019_Bioorg.Chem_93_103310 |
PubMedID: 31586704 |
Title : Investigation of multi-target-directed ligands (MTDLs) with butyrylcholinesterase (BuChE) and indoleamine 2,3-dioxygenase 1 (IDO1) inhibition: The design, synthesis of miconazole analogues targeting Alzheimer's disease - Lu_2018_Bioorg.Med.Chem_26_1665 |
Author(s) : Lu X , He SY , Li Q , Yang H , Jiang X , Lin H , Chen Y , Qu W , Feng F , Bian Y , Zhou Y , Sun H |
Ref : Bioorganic & Medicinal Chemistry , 26 :1665 , 2018 |
Abstract : |
PubMedSearch : Lu_2018_Bioorg.Med.Chem_26_1665 |
PubMedID: 29475581 |
Title : Dual GSK-3beta\/AChE Inhibitors as a New Strategy for Multitargeting Anti-Alzheimer's Disease Drug Discovery - Jiang_2018_ACS.Med.Chem.Lett_9_171 |
Author(s) : Jiang XY , Chen TK , Zhou JT , He SY , Yang HY , Chen Y , Qu W , Feng F , Sun HP |
Ref : ACS Med Chem Lett , 9 :171 , 2018 |
Abstract : |
PubMedSearch : Jiang_2018_ACS.Med.Chem.Lett_9_171 |
PubMedID: 29541355 |
Title : Donepezil-based multi-functional cholinesterase inhibitors for treatment of Alzheimer's disease - Li_2018_Eur.J.Med.Chem_158_463 |
Author(s) : Li Q , He S , Chen Y , Feng F , Qu W , Sun H |
Ref : Eur Journal of Medicinal Chemistry , 158 :463 , 2018 |
Abstract : |
PubMedSearch : Li_2018_Eur.J.Med.Chem_158_463 |
PubMedID: 30243151 |
Title : Exploring the binding interaction between copper ions and Candida rugosa lipase - Qu_2018_Toxicol.Res.(Camb)_7_1100 |
Author(s) : Qu W , Yuan D , Zhao L , Zong W , Liu R |
Ref : Toxicol Res (Camb) , 7 :1100 , 2018 |
Abstract : |
PubMedSearch : Qu_2018_Toxicol.Res.(Camb)_7_1100 |
PubMedID: 30542604 |
Title : Acute toxicity of the pesticide methomyl on the topmouth gudgeon (Pseudorasbora parva): mortality and effects on four biomarkers - Li_2008_Fish.Physiol.Biochem_34_209 |
Author(s) : Li H , Jiang H , Gao X , Wang X , Qu W , Lin R , Chen J |
Ref : Fish Physiol Biochem , 34 :209 , 2008 |
Abstract : |
PubMedSearch : Li_2008_Fish.Physiol.Biochem_34_209 |
PubMedID: 18665458 |