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| Title : Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization - Butini_2024_J.Med.Chem__ |
| Author(s) : Butini S , Grether U , Jung KM , Ligresti A , Allara M , Postmus AGJ , Maramai S , Brogi S , Papa A , Carullo G , Sykes D , Veprintsev D , Federico S , Grillo A , Di Guglielmo B , Ramunno A , Stevens AF , Heer D , Lamponi S , Gemma S , Benz J , Di Marzo V , van der Stelt M , Piomelli D , Campiani G |
| Ref : Journal of Medicinal Chemistry , : , 2024 |
| Abstract : Butini_2024_J.Med.Chem__ |
| ESTHER : Butini_2024_J.Med.Chem__ |
| PubMedSearch : Butini_2024_J.Med.Chem__ |
| PubMedID: 38241614 |
| Gene_locus related to this paper: human-MGLL |
| Title : Assay of Monoacylglycerol Lipase Activity - Jung_2023_Methods.Mol.Biol_2576_285 |
| Author(s) : Jung KM , Piomelli D |
| Ref : Methods Mol Biol , 2576 :285 , 2023 |
| Abstract : Jung_2023_Methods.Mol.Biol_2576_285 |
| ESTHER : Jung_2023_Methods.Mol.Biol_2576_285 |
| PubMedSearch : Jung_2023_Methods.Mol.Biol_2576_285 |
| PubMedID: 36152196 |
| Title : Benzisothiazolinone derivatives as potent allosteric monoacylglycerol lipase inhibitors that functionally mimic sulfenylation of regulatory cysteines - Castelli_2020_J.Med.Chem_63_1261 |
| Author(s) : Castelli R , Scalvini L , Vacondio F , Lodola A , Anselmi M , Vezzosi S , Carmi C , Bassi M , Ferlenghi F , Rivara S , Moller IR , Rand KD , Daglian J , Wei D , Dotsey EY , Ahmed F , Jung KM , Stella N , Singh S , Mor M , Piomelli D |
| Ref : Journal of Medicinal Chemistry , 63 :1261 , 2020 |
| Abstract : Castelli_2020_J.Med.Chem_63_1261 |
| ESTHER : Castelli_2020_J.Med.Chem_63_1261 |
| PubMedSearch : Castelli_2020_J.Med.Chem_63_1261 |
| PubMedID: 31714779 |
| Title : Development and Pharmacological Characterization of Selective Blockers of 2-Arachidonoyl Glycerol Degradation with Efficacy in Rodent Models of Multiple Sclerosis and Pain - Brindisi_2016_J.Med.Chem_59_2612 |
| Author(s) : Brindisi M , Maramai S , Gemma S , Brogi S , Grillo A , Di Cesare Mannelli L , Gabellieri E , Lamponi S , Saponara S , Gorelli B , Tedesco D , Bonfiglio T , Landry C , Jung KM , Armirotti A , Luongo L , Ligresti A , Piscitelli F , Bertucci C , Dehouck MP , Campiani G , Maione S , Ghelardini C , Pittaluga A , Piomelli D , Di Marzo V , Butini S |
| Ref : Journal of Medicinal Chemistry , 59 :2612 , 2016 |
| Abstract : Brindisi_2016_J.Med.Chem_59_2612 |
| ESTHER : Brindisi_2016_J.Med.Chem_59_2612 |
| PubMedSearch : Brindisi_2016_J.Med.Chem_59_2612 |
| PubMedID: 26888301 |
| Title : Free-energy studies reveal a possible mechanism for oxidation-dependent inhibition of MGL - Scalvini_2016_Sci.Rep_6_31046 |
| Author(s) : Scalvini L , Vacondio F , Bassi M , Pala D , Lodola A , Rivara S , Jung KM , Piomelli D , Mor M |
| Ref : Sci Rep , 6 :31046 , 2016 |
| Abstract : Scalvini_2016_Sci.Rep_6_31046 |
| ESTHER : Scalvini_2016_Sci.Rep_6_31046 |
| PubMedSearch : Scalvini_2016_Sci.Rep_6_31046 |
| PubMedID: 27499063 |
| Title : Endocannabinoid Modulation of Predator Stress-Induced Long-Term Anxiety in Rats - Lim_2016_Neuropsychopharmacology_41_1329 |
| Author(s) : Lim J , Igarashi M , Jung KM , Butini S , Campiani G , Piomelli D |
| Ref : Neuropsychopharmacology , 41 :1329 , 2016 |
| Abstract : Lim_2016_Neuropsychopharmacology_41_1329 |
| ESTHER : Lim_2016_Neuropsychopharmacology_41_1329 |
| PubMedSearch : Lim_2016_Neuropsychopharmacology_41_1329 |
| PubMedID: 26361059 |
| Title : Activation of type 5 metabotropic glutamate receptors and diacylglycerol lipase-alpha initiates 2-arachidonoylglycerol formation and endocannabinoid-mediated analgesia - Gregg_2012_J.Neurosci_32_9457 |
| Author(s) : Gregg LC , Jung KM , Spradley JM , Nyilas R , Suplita RL, 2nd , Zimmer A , Watanabe M , Mackie K , Katona I , Piomelli D , Hohmann AG |
| Ref : Journal of Neuroscience , 32 :9457 , 2012 |
| Abstract : Gregg_2012_J.Neurosci_32_9457 |
| ESTHER : Gregg_2012_J.Neurosci_32_9457 |
| PubMedSearch : Gregg_2012_J.Neurosci_32_9457 |
| PubMedID: 22787031 |
| Gene_locus related to this paper: human-DAGLA |
| Title : Uncoupling of the endocannabinoid signalling complex in a mouse model of fragile X syndrome - Jung_2012_Nat.Commun_3_1080 |
| Author(s) : Jung KM , Sepers M , Henstridge CM , Lassalle O , Neuhofer D , Martin H , Ginger M , Frick A , DiPatrizio NV , Mackie K , Katona I , Piomelli D , Manzoni OJ |
| Ref : Nat Commun , 3 :1080 , 2012 |
| Abstract : Jung_2012_Nat.Commun_3_1080 |
| ESTHER : Jung_2012_Nat.Commun_3_1080 |
| PubMedSearch : Jung_2012_Nat.Commun_3_1080 |
| PubMedID: 23011134 |
| Title : Diacylglycerol lipase-alpha and -beta control neurite outgrowth in neuro-2a cells through distinct molecular mechanisms - Jung_2011_Mol.Pharmacol_80_60 |
| Author(s) : Jung KM , Astarita G , Thongkham D , Piomelli D |
| Ref : Molecular Pharmacology , 80 :60 , 2011 |
| Abstract : Jung_2011_Mol.Pharmacol_80_60 |
| ESTHER : Jung_2011_Mol.Pharmacol_80_60 |
| PubMedSearch : Jung_2011_Mol.Pharmacol_80_60 |
| PubMedID: 21493725 |
| Title : Discovery of potent and reversible monoacylglycerol lipase inhibitors - King_2009_Chem.Biol_16_1045 |
| Author(s) : King AR , Dotsey EY , Lodola A , Jung KM , Ghomian A , Qiu Y , Fu J , Mor M , Piomelli D |
| Ref : Chemical Biology , 16 :1045 , 2009 |
| Abstract : King_2009_Chem.Biol_16_1045 |
| ESTHER : King_2009_Chem.Biol_16_1045 |
| PubMedSearch : King_2009_Chem.Biol_16_1045 |
| PubMedID: 19875078 |
| Title : A key role for diacylglycerol lipase-alpha in metabotropic glutamate receptor-dependent endocannabinoid mobilization - Jung_2007_Mol.Pharmacol_72_612 |
| Author(s) : Jung KM , Astarita G , Zhu C , Wallace M , Mackie K , Piomelli D |
| Ref : Molecular Pharmacology , 72 :612 , 2007 |
| Abstract : Jung_2007_Mol.Pharmacol_72_612 |
| ESTHER : Jung_2007_Mol.Pharmacol_72_612 |
| PubMedSearch : Jung_2007_Mol.Pharmacol_72_612 |
| PubMedID: 17584991 |
| Title : Molecular composition of the endocannabinoid system at glutamatergic synapses - Katona_2006_J.Neurosci_26_5628 |
| Author(s) : Katona I , Urban GM , Wallace M , Ledent C , Jung KM , Piomelli D , Mackie K , Freund TF |
| Ref : Journal of Neuroscience , 26 :5628 , 2006 |
| Abstract : Katona_2006_J.Neurosci_26_5628 |
| ESTHER : Katona_2006_J.Neurosci_26_5628 |
| PubMedSearch : Katona_2006_J.Neurosci_26_5628 |
| PubMedID: 16723519 |
| Gene_locus related to this paper: mouse-q6wqj1 |
| Title : Stimulation of endocannabinoid formation in brain slice cultures through activation of group I metabotropic glutamate receptors - Jung_2005_Mol.Pharmacol_68_1196 |
| Author(s) : Jung KM , Mangieri R , Stapleton C , Kim J , Fegley D , Wallace M , Mackie K , Piomelli D |
| Ref : Molecular Pharmacology , 68 :1196 , 2005 |
| Abstract : Jung_2005_Mol.Pharmacol_68_1196 |
| ESTHER : Jung_2005_Mol.Pharmacol_68_1196 |
| PubMedSearch : Jung_2005_Mol.Pharmacol_68_1196 |
| PubMedID: 16051747 |
| Gene_locus related to this paper: rat-dglb |