| Title : 2-Arylhydrazinylidene-3-oxo-3-polyfluoroalkylpropanoic acids as selective and effective carboxylesterase inhibitors with powerful antioxidant potential - Burgart_2024_Bioorg.Med.Chem_115_117938 |
| Author(s) : Burgart YV , Makhaeva GF , Khudina OG , Krasnykh OP , Kovaleva NV , Elkina NA , Boltneva NP , Rudakova EV , Lushchekina SV , Shchegolkov EV , Triandafilova GA , Malysheva KO , Serebryakova OG , Borisevich SS , Ilyina MG , Zhilina EF , Saloutin VI , Charushin VN , Richardson RJ |
| Ref : Bioorganic & Medicinal Chemistry , 115 :117938 , 2024 |
| Abstract : |
| PubMedSearch : Burgart_2024_Bioorg.Med.Chem_115_117938 |
| PubMedID: 39504592 |
| Title : New Multifunctional Agents for Potential Alzheimer's Disease Treatment Based on Tacrine Conjugates with 2-Arylhydrazinylidene-1,3-Diketones - Elkina_2022_Biomolecules_12_ |
| Author(s) : Elkina NA , Grishchenko MV , Shchegolkov EV , Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Astakhova TY , Radchenko EV , Palyulin VA , Zhilina EF , Perminova AN , Lapshin LS , Burgart YV , Saloutin VI , Richardson RJ |
| Ref : Biomolecules , 12 : , 2022 |
| Abstract : |
| PubMedSearch : Elkina_2022_Biomolecules_12_ |
| PubMedID: 36358901 |
| Title : Powerful Potential of Polyfluoroalkyl-Containing 4-Arylhydrazinylidenepyrazol-3-ones for Pharmaceuticals - Burgart_2022_Molecules_28_ |
| Author(s) : Burgart YV , Elkina NA , Shchegolkov EV , Krasnykh OP , Makhaeva GF , Triandafilova GA , Solodnikov SY , Boltneva NP , Rudakova EV , Kovaleva NV , Serebryakova OG , Ulitko MV , Borisevich SS , Gerasimova NA , Evstigneeva NP , Kozlov SA , Korolkova YV , Minin AS , Belousova AV , Mozhaitsev ES , Klabukov AM , Saloutin VI |
| Ref : Molecules , 28 : , 2022 |
| Abstract : |
| PubMedSearch : Burgart_2022_Molecules_28_ |
| PubMedID: 36615256 |
| Title : Novel potent bifunctional carboxylesterase inhibitors based on a polyfluoroalkyl-2-imino-1,3-dione scaffold - Makhaeva_2021_Eur.J.Med.Chem_218_113385 |
| Author(s) : Makhaeva GF , Lushchekina SV , Boltneva NP , Serebryakova OG , Kovaleva NV , Rudakova EV , Elkina NA , Shchegolkov EV , Burgart YV , Stupina TS , Terentiev AA , Radchenko EV , Palyulin VA , Saloutin VI , Bachurin SO , Richardson RJ |
| Ref : Eur Journal of Medicinal Chemistry , 218 :113385 , 2021 |
| Abstract : |
| PubMedSearch : Makhaeva_2021_Eur.J.Med.Chem_218_113385 |
| PubMedID: 33831780 |
| Title : Synthesis, molecular docking, and biological evaluation of 3-oxo-2-tolylhydrazinylidene-4,4,4-trifluorobutanoates bearing higher and natural alcohol moieties as new selective carboxylesterase inhibitors - Makhaeva_2019_Bioorg.Chem_91_103097 |
| Author(s) : Makhaeva GF , Elkina NA , Shchegolkov EV , Boltneva NP , Lushchekina SV , Serebryakova OG , Rudakova EV , Kovaleva NV , Radchenko EV , Palyulin VA , Burgart YV , Saloutin VI , Bachurin SO , Richardson RJ |
| Ref : Bioorg Chem , 91 :103097 , 2019 |
| Abstract : |
| PubMedSearch : Makhaeva_2019_Bioorg.Chem_91_103097 |
| PubMedID: 31323527 |
| Title : Synthesis of 2-arylhydrazinylidene-3-oxo-4,4,4-trifluorobutanoic acids as new selective carboxylesterase inhibitors and radical scavengers - Khudina_2019_Bioorg.Med.Chem.Lett__126716 |
| Author(s) : Khudina OG , Makhaeva GF , Elkina NA , Boltneva NP , Serebryakova OG , Shchegolkov EV , Rudakova EV , Lushchekina SV , Burgart YV , Bachurin SO , Richardson RJ , Saloutin VI |
| Ref : Bioorganic & Medicinal Chemistry Lett , :126716 , 2019 |
| Abstract : |
| PubMedSearch : Khudina_2019_Bioorg.Med.Chem.Lett__126716 |
| PubMedID: 31640885 |