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Title : Conjugates of amiridine and thiouracil derivatives as effective inhibitors of butyrylcholinesterase with the potential to block beta-amyloid aggregation - Khudina_2023_Arch.Pharm.(Weinheim)__e2300447 |
Author(s) : Khudina OG , Grishchenko MV , Makhaeva GF , Kovaleva NV , Boltneva NP , Rudakova EV , Lushchekina SV , Shchegolkov EV , Borisevich SS , Burgart YV , Saloutin VI , Charushin VN |
Ref : Arch Pharm (Weinheim) , :e2300447 , 2023 |
Abstract : Khudina_2023_Arch.Pharm.(Weinheim)__e2300447 |
ESTHER : Khudina_2023_Arch.Pharm.(Weinheim)__e2300447 |
PubMedSearch : Khudina_2023_Arch.Pharm.(Weinheim)__e2300447 |
PubMedID: 38072670 |
Title : Derivatives of 9-phosphorylated acridine as butyrylcholinesterase inhibitors with antioxidant activity and the ability to inhibit beta-amyloid self-aggregation: potential therapeutic agents for Alzheimer's disease - Makhaeva_2023_Front.Pharmacol_14_1219980 |
Author(s) : Makhaeva GF , Kovaleva NV , Rudakova EV , Boltneva NP , Lushchekina SV , Astakhova TY , Timokhina EN , Serebryakova OG , Shchepochkin AV , Averkov MA , Utepova IA , Demina NS , Radchenko EV , Palyulin VA , Fisenko VP , Bachurin SO , Chupakhin ON , Charushin VN , Richardson RJ |
Ref : Front Pharmacol , 14 :1219980 , 2023 |
Abstract : Makhaeva_2023_Front.Pharmacol_14_1219980 |
ESTHER : Makhaeva_2023_Front.Pharmacol_14_1219980 |
PubMedSearch : Makhaeva_2023_Front.Pharmacol_14_1219980 |
PubMedID: 37654616 |
Title : 9-Substituted acridine derivatives as acetylcholinesterase and butyrylcholinesterase inhibitors possessing antioxidant activity for Alzheimer's disease treatment - Makhaeva_2017_Bioorg.Med.Chem_25_5981 |
Author(s) : Makhaeva GF , Lushchekina SV , Boltneva NP , Serebryakova OG , Rudakova EV , Ustyugov AA , Bachurin SO , Shchepochkin AV , Chupakhin ON , Charushin VN , Richardson RJ |
Ref : Bioorganic & Medicinal Chemistry , 25 :5981 , 2017 |
Abstract : Makhaeva_2017_Bioorg.Med.Chem_25_5981 |
ESTHER : Makhaeva_2017_Bioorg.Med.Chem_25_5981 |
PubMedSearch : Makhaeva_2017_Bioorg.Med.Chem_25_5981 |
PubMedID: 28986116 |