Full name : De la Mora Eugenio
First name : Eugenio
Mail : Institut de Biologie Structurale, Grenoble
Zip Code :
City :
Country : France
Email : eugenio.de-la-mora-lugo@ibs.fr
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Directory :
Title : Chiral Separation, X-ray Structure, and Biological Evaluation of a Potent and Reversible Dual Binding Site AChE Inhibitor - Catto_2020_ACS.Med.Chem.Lett_11_869 |
Author(s) : Catto M , Pisani L , De la Mora E , Belviso BD , Mangiatordi GF , Pinto A , Palma A , Denora N , Caliandro R , Colletier JP , Silman I , Nicolotti O , Altomare CD |
Ref : ACS Med Chem Lett , 11 :869 , 2020 |
Abstract : |
PubMedSearch : Catto_2020_ACS.Med.Chem.Lett_11_869 |
PubMedID: 32435398 |
Title : Rivastigmine and metabolite analogues with putative Alzheimer's disease-modifying properties in a Caenorhabditis elegans model. - Dighe_2019_Commun.Chem_2_35 |
Author(s) : Dighe SN , De la Mora E , Chan S , Kantham S , McColl G , Miles JA , Veliyath SK , Sreenivas BY , Nassar ZD , Silman I , Sussman JL , Weik M , McGeary RP , Parat MO , Brazzolotto X , Ross BP |
Ref : Communications chemistry , 2 :35 , 2019 |
Abstract : |
PubMedSearch : Dighe_2019_Commun.Chem_2_35 |
PubMedID: |
Gene_locus related to this paper: human-BCHE , torca-ACHE |
Title : Structure-Based Optimization of Nonquaternary Reactivators of Acetylcholinesterase Inhibited by Organophosphorus Nerve Agents - Santoni_2018_J.Med.Chem_61_7630 |
Author(s) : Santoni G , de Sousa J , De la Mora E , Dias J , Jean L , Sussman JL , Silman I , Renard PY , Brown RCD , Weik M , Baati R , Nachon F |
Ref : Journal of Medicinal Chemistry , 61 :7630 , 2018 |
Abstract : |
PubMedSearch : Santoni_2018_J.Med.Chem_61_7630 |
PubMedID: 30125110 |
Gene_locus related to this paper: torca-ACHE |
Title : Potent 3-Hydroxy-2-Pyridine Aldoxime Reactivators of Organophosphate-Inhibited Cholinesterases with Predicted Blood-Brain Barrier Penetration - Zorbaz_2018_Chemistry_24_9675 |
Author(s) : Zorbaz T , Braiki A , Marakovic N , Renou J , De la Mora E , Macek Hrvat N , Katalinic M , Silman I , Sussman JL , Mercey G , Gomez C , Mougeot R , Perez B , Baati R , Nachon F , Weik M , Jean L , Kovarik Z , Renard PY |
Ref : Chemistry , 24 :9675 , 2018 |
Abstract : |
PubMedSearch : Zorbaz_2018_Chemistry_24_9675 |
PubMedID: 29672968 |
Gene_locus related to this paper: torca-ACHE |
Title : Discovery and Structure-Activity Relationships of a Highly Selective Butyrylcholinesterase Inhibitor by Structure-Based Virtual Screening - Dighe_2016_J.Med.Chem_59_7683 |
Author(s) : Dighe SN , Deora GS , De la Mora E , Nachon F , Chan S , Parat MO , Brazzolotto X , Ross BP |
Ref : Journal of Medicinal Chemistry , 59 :7683 , 2016 |
Abstract : |
PubMedSearch : Dighe_2016_J.Med.Chem_59_7683 |
PubMedID: 27405689 |
Gene_locus related to this paper: human-BCHE |