FAPI-04

Theranostic ligand for FAP. DOTA (Tetraxetan 2-[4,7,10-tris(carboxymethyl)-1,4,7,10-tetrazacyclododec-1-yl]) chelating agent for metallic ions (177Lu and 68Ga for example) used in PET imaging. Gallium Ga 68-DOTA-FAPI-04 is a radioconjugate composed of FAPI-04, a quinoline-based fibroblast activation protein (FAP)-targeted tracer belonging to the group of FAP inhibitors (FAPi), conjugated, through the macrocyclic chelator 1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid (DOTA), to the radioisotope gallium Ga 68

General

Type : Piperazine, Quinoline, PET probe, Carboxamide, tert-Butyl, tert-Butyloxycarbonyl, Tetrazacyclododec, Cyanide

Chemical_Nomenclature : DOTA (S)-N-(2-(2-cyano-4,4-difluoropyrrolidin-1-yl)-2-oxoethyl)-6-(3-(4-tertbutoxycarbonyl-piperazin-1-yl)-1-propoxy)quinoline-4-carboxamide || 2-[4,7-bis(carboxymethyl)-10-[2-[4-[3-[4-[[2-[(2S)-2-cyano-4,4-difluoropyrrolidin-1-yl]-2-oxoethyl]carbamoyl]quinolin-6-yl]oxypropyl]piperazin-1-yl]-2-oxoethyl]-1,4,7,10-tetrazacyclododec-1-yl]acetic acid

Canonical SMILES : C1CN(CCN1CCCOC3=CC2=C(C=CN=C2C=C3)C(=O)NCC(=O)N4CC(CC4C#N)(F)F)C(=O)CN5CCN(CCN(CCN(CC5)CC(=O)O)CC(=O)O)CC(=O)O || C1CN(CCN1CCCOC2=CC3=C(C=CN=C3C=C2)C(=O)NCC(=O)N4CC(CC4C#N)(F)F)C(=O)CN5CCN(CCN(CCN(CC5)CC(=O)O)CC(=O)O)CC(=O)O

InChI : InChI=1S\/C40H54F2N10O10\/c41-40(42)21-29(22-43)52(28-40)34(53)23-45-39(61)31-4-5-44-33-3-2-30(20-32(31)33)62-19-1-6-46-15-17-51(18-16-46)35(54)24-47-7-9-48(25-36(55)56)11-13-50(27-38(59)60)14-12-49(10-8-47)26-37(57)58\/h2-5,20,29H,1,6-19,21,23-28H2,(H,45,61)(H,55,56)(H,57,58)(H,59,60) || InChI=1S\/C40H54F2N10O10\/c41-40(42)21-29(22-43)52(28-40)34(53)23-45-39(61)31-4-5-44-33-3-2-30(20-32(31)33)62-19-1-6-46-15-17-51(18-16-46)35(54)24-47-7-9-48(25-36(55)56)11-13-50(27-38(59)60)14-12-49(10-8-47)26-37(57)58\/h2-5,20,29H,1,6-19,21,23-28H2,(H,45,61)(H,55,56)(H,57,58)(H,59,60)\/t29-\/m0\/s1

InChIKey : ICWDAESAANBIGG-UHFFFAOYSA-N || ICWDAESAANBIGG-LJAQVGFWSA-N

Other name(s) : FAPI-4  ||  ZZ7Stn2lbb  ||  Gallium-68-fapi-04  ||  68Ga-Fapi-04  ||  (68Ga)-DOTA-fapi-04  ||  FAPI-04 Ga-68  ||  SCHEMBL21257058


MW : 872.91

Formula : C40H54F2N10O10

CAS_number :

PubChem : 155907829,    138454803

UniChem : ICWDAESAANBIGG-UHFFFAOYSA-N,    ICWDAESAANBIGG-LJAQVGFWSA-N

Target

Families : FAPI-04 ligand of proteins in family
DPP4N_Peptidase_S9

Protein :
human-FAP

References (94)

Title : 68 Ga-FAPI-04 PET\/CT in Assessment of Fibroblast Activation in Keloids : A Prospective Pilot Study - Wang_2024_Clin.Nucl.Med_49_16
Author(s) : Wang J , Yu N , Wang G , Wang R , Li L , Jiang Y , Sui H , Sun Y , Li Z , Long X , Zhu Z
Ref : Clin Nucl Med , 49 :16 , 2024
Abstract :
PubMedSearch : Wang_2024_Clin.Nucl.Med_49_16
PubMedID: 38015039

Title : Non-invasive visualization of liver fibrosis with [(68)Ga]Ga-DOTA-FAPI-04 PET from preclinical insights to clinical translation - Song_2024_Eur.J.Nucl.Med.Mol.Imaging_51_3572
Author(s) : Song Y , Qin C , Chen Y , Ruan W , Gai Y , Song W , Gao Y , Hu W , Qiao P , Song X , Lv X , Zheng D , Chu H , Jiang D , Yang L , Lan X
Ref : Eur J Nucl Med Mol Imaging , 51 :3572 , 2024
Abstract :
PubMedSearch : Song_2024_Eur.J.Nucl.Med.Mol.Imaging_51_3572
PubMedID: 38850311

Title : [(68)Ga]Ga-labeled FAPI Conjugated with Gly-Pro Sequence for PET Imaging of Malignant Tumors - Shang_2024_Mol.Imaging.Biol_26_729
Author(s) : Shang Y , Zhang G , Yao X , Lai C , Wang F , Zeng B , Liu E , Yuan H , Cheng Z , Jiang L
Ref : Mol Imaging Biol , 26 :729 , 2024
Abstract :
PubMedSearch : Shang_2024_Mol.Imaging.Biol_26_729
PubMedID: 38987449

Title : [(68)Ga]Ga-FAP-2286, a novel promising theragnostic approach for PET\/CT imaging in patients with various type of metastatic cancers - Banihashemian_2024_Eur.J.Nucl.Med.Mol.Imaging_51_1981
Author(s) : Banihashemian SS , Divband G , Pirayesh E , Nikkholgh B , Amini H , Shahrnoy AA , Nami R , Akbari ME
Ref : Eur J Nucl Med Mol Imaging , 51 :1981 , 2024
Abstract :
PubMedSearch : Banihashemian_2024_Eur.J.Nucl.Med.Mol.Imaging_51_1981
PubMedID: 38376804

Title : Value of Semi-Quantitative Parameters of (68)Ga-FAPI-04 PET\/CT in Primary Malignant and Benign Diseases: A Comparison with (18)F-FDG - Li_2024_Cancer.Biother.Radiopharm_39_654
Author(s) : Li T , Liu Y , Dai M , Zhao X , Han J , Zhang Z , Jing F , Tian W , Zhang J , Wang J , Hao T , Wang T
Ref : Cancer Biother Radiopharm , 39 :654 , 2024
Abstract :
PubMedSearch : Li_2024_Cancer.Biother.Radiopharm_39_654
PubMedID: 38808470

Title : Development of an FAP-Targeted PET Probe Based on a Novel Quinolinium Molecular Scaffold - Li_2024_Bioconjug.Chem_35_1309
Author(s) : Li L , Cao R , Chen K , Qu C , Qian K , Lin J , Li R , Lai C , Wang X , Han Z , Xu Z , Zhou L , Song S , Zhu W , Cheng Z
Ref : Bioconjug Chem , 35 :1309 , 2024
Abstract :
PubMedSearch : Li_2024_Bioconjug.Chem_35_1309
PubMedID: 38954733

Title : (68)Ga-FAPI-04 PET\/CT in Non-Small Cell Lung Cancer: Accurate Evaluation of Lymph Node Metastasis and Correlation with Fibroblast Activation Protein Expression - Li_2024_J.Nucl.Med_65_527
Author(s) : Li C , Chen Q , Tian Y , Chen J , Xu K , Xiao Z , Zhong J , Wu J , Wen B , He Y
Ref : J Nucl Med , 65 :527 , 2024
Abstract :
PubMedSearch : Li_2024_J.Nucl.Med_65_527
PubMedID: 38453362

Title : (68)Ga\/(177)Lu-Labeled Theranostic Pair for Targeting Fibroblast Activation Protein with Improved Tumor Uptake and Retention - Huang_2024_J.Med.Chem_67_17785
Author(s) : Huang J , Zhang X , Liu Q , Gong F , Huang Y , Huang S , Fu L , Tang G
Ref : Journal of Medicinal Chemistry , 67 :17785 , 2024
Abstract :
PubMedSearch : Huang_2024_J.Med.Chem_67_17785
PubMedID: 39321030

Title : Heterogeneity of fibroblast activation protein expression in the microenvironment of an intracranial tumor cohort: head-to-head comparison of gallium-68 FAP inhibitor-04 ((68)Ga-FAPi-04) and fluoride-18 fluoroethyl-L-tyrosine ((18)F-FET) in positron emission tomography-computed tomography imaging - Hua_2024_Quant.Imaging.Med.Surg_14_4450
Author(s) : Hua T , Chen M , Fu P , Zhou W , Zhao W , Li M , Zuo C , Guan Y , Xu H
Ref : Quant Imaging Med Surg , 14 :4450 , 2024
Abstract :
PubMedSearch : Hua_2024_Quant.Imaging.Med.Surg_14_4450
PubMedID: 39022225

Title : An Automated Radiosynthesis of [68Ga]Ga-FAPI-46 for Routine Clinical Use - Morandeau_2024_J.Vis.Exp__
Author(s) : Morandeau L , Ioppolo JA , Alvarez de Eulate E , Mohamed S , Cullen D , Asad AH , Francis RJ , Atkinson J
Ref : J Vis Exp , : , 2024
Abstract :
PubMedSearch : Morandeau_2024_J.Vis.Exp__
PubMedID: 38856210

Title : Development and Evaluation of DOTA-FAPI-Maleimide as a Novel Radiotracer for Tumor Theranostic with Extended Circulation - Feng_2024_Mol.Pharm_21_4386
Author(s) : Feng L , Hu W , Zeng X , Wei Z , Long Y , Li M , Sun S , Guo Z , Lan X , Zhang X , Zhuang R , Jiang D
Ref : Mol Pharm , 21 :4386 , 2024
Abstract :
PubMedSearch : Feng_2024_Mol.Pharm_21_4386
PubMedID: 39046432

Title : Preclinical Evaluation and a Pilot Clinical Positron Emission Tomography Imaging Study of [(68)Ga]Ga-FAPI-FUSCC-II - Du_2024_Mol.Pharm_21_904
Author(s) : Du X , Gu B , Wang X , Ji M , Zhang J , He S , Xu X , Yang Z , Song S
Ref : Mol Pharm , 21 :904 , 2024
Abstract :
PubMedSearch : Du_2024_Mol.Pharm_21_904
PubMedID: 38179677

Title : Clinical translation of a novel FAPI dimer [(68)Ga]Ga-LNC1013 - Tan_2024_Eur.J.Nucl.Med.Mol.Imaging_51_2761
Author(s) : Tan Y , Li J , Zhao T , Zhou M , Liu K , Xiang S , Tang Y , Jakobsson V , Xu P , Chen X , Zhang J
Ref : Eur J Nucl Med Mol Imaging , 51 :2761 , 2024
Abstract :
PubMedSearch : Tan_2024_Eur.J.Nucl.Med.Mol.Imaging_51_2761
PubMedID: 38561515

Title : Molecular imaging reveals the heterogeneous progression of tumor cells and tumor stroma: a practice of FDG PET and FAPI PET in diagnosing PSMA-negative bone metastases of progressive prostate cancer - Zhu_2024_Am.J.Nucl.Med.Mol.Imaging_14_13
Author(s) : Zhu L , Chen P , Guo Z , Li F , Luo X , Du X , Zhang L , Zuo C , Li X
Ref : Am J Nucl Med Mol Imaging , 14 :13 , 2024
Abstract :
PubMedSearch : Zhu_2024_Am.J.Nucl.Med.Mol.Imaging_14_13
PubMedID: 38500747

Title : The earliest optimal timing for total-body (68)Ga-fibroblast activation protein inhibitor-04 PET scans: an evidence-based single-centre study - Zheng_2024_Eur.Radiol_34_4550
Author(s) : Zheng Z , Gao H , Lin Y , Yu H , Mao W , Yang R , He Y , Chen X , Wu H , Hu P , Shi H
Ref : Eur Radiol , 34 :4550 , 2024
Abstract :
PubMedSearch : Zheng_2024_Eur.Radiol_34_4550
PubMedID: 38110627

Title : Early detection of anthracycline-induced cardiotoxicity using [(68) Ga]Ga-FAPI-04 imaging - Wei_2024_Eur.J.Nucl.Med.Mol.Imaging_51_2204
Author(s) : Wei Z , Xu H , Chen B , Wang J , Yang X , Yang MF , Zhao S
Ref : Eur J Nucl Med Mol Imaging , 51 :2204 , 2024
Abstract :
PubMedSearch : Wei_2024_Eur.J.Nucl.Med.Mol.Imaging_51_2204
PubMedID: 38491214

Title : Molecular imaging of fibroblast activity in pressure overload heart failure using [(68) Ga]Ga-FAPI-04 PET\/CT - Wang_2023_Eur.J.Nucl.Med.Mol.Imaging_50_465
Author(s) : Wang G , Yang Q , Wu S , Xu X , Li X , Liang S , Pan G , Zuo C , Zhao X , Cheng C , Liu S
Ref : Eur J Nucl Med Mol Imaging , 50 :465 , 2023
Abstract :
PubMedSearch : Wang_2023_Eur.J.Nucl.Med.Mol.Imaging_50_465
PubMedID: 36171409

Title : Novel (68)Ga-Labeled Pyridine-Based Fibroblast Activation Protein-Targeted Tracers with High Tumor-to-Background Contrast - Verena_2023_Pharmaceuticals.(Basel)_16_
Author(s) : Verena A , Kuo HT , Merkens H , Zeisler J , Bendre S , Wong A , Benard F , Lin KS
Ref : Pharmaceuticals (Basel) , 16 : , 2023
Abstract :
PubMedSearch : Verena_2023_Pharmaceuticals.(Basel)_16_
PubMedID: 36986548

Title : Fibroblast activation protein-targeted radionuclide therapy: background, opportunities, and challenges of first (pre)clinical studies - Prive_2023_Eur.J.Nucl.Med.Mol.Imaging_50_1906
Author(s) : Prive BM , Boussihmad MA , Timmermans B , van Gemert WA , Peters SMB , Derks YHW , van Lith SAM , Mehra N , Nagarajah J , Heskamp S , Westdorp H
Ref : Eur J Nucl Med Mol Imaging , 50 :1906 , 2023
Abstract :
PubMedSearch : Prive_2023_Eur.J.Nucl.Med.Mol.Imaging_50_1906
PubMedID: 36813980

Title : Utility of [(68)Ga]FAPI-04 and [(18)F]FDG dual-tracer PET\/CT in the initial evaluation of gastric cancer - Miao_2023_Eur.Radiol_33_4355
Author(s) : Miao Y , Feng R , Guo R , Huang X , Hai W , Li J , Yu T , Qu Q , Zhang M , Shangguan C , Mi J , Zhu Z , Li B
Ref : Eur Radiol , 33 :4355 , 2023
Abstract :
PubMedSearch : Miao_2023_Eur.Radiol_33_4355
PubMedID: 36522509

Title : PET Imaging of Fibroblast Activation Protein in Various Types of Cancer Using (68)Ga-FAP-2286: Comparison with (18)F-FDG and (68)Ga-FAPI-46 in a Single-Center, Prospective Study - Pang_2023_J.Nucl.Med_64_386
Author(s) : Pang Y , Zhao L , Meng T , Xu W , Lin Q , Wu H , Zhang J , Chen X , Sun L , Chen H
Ref : J Nucl Med , 64 :386 , 2023
Abstract :
PubMedSearch : Pang_2023_J.Nucl.Med_64_386
PubMedID: 36215571

Title : Noninvasive Assessment of Renal Fibrosis of Chronic Kidney Disease in Rats by [(68)Ga]Ga-FAPI-04 Small Animal PET\/CT and Biomarkers - Mao_2023_Mol.Pharm_20_2714
Author(s) : Mao H , Chen L , Wu W , Zhang L , Li X , Chen Y , Huang Z , Ou S
Ref : Mol Pharm , 20 :2714 , 2023
Abstract :
PubMedSearch : Mao_2023_Mol.Pharm_20_2714
PubMedID: 37010328

Title : Comparison of 18 F-FDG and 68 Ga-FAPI-04 Uptake in Postoperative Re-evaluation of Gastric, Duodenal, and Colorectal Cancers - Liu_2023_Clin.Nucl.Med_48_304
Author(s) : Liu H , Yang X , Liu L , Qu G , Chen Y
Ref : Clin Nucl Med , 48 :304 , 2023
Abstract :
PubMedSearch : Liu_2023_Clin.Nucl.Med_48_304
PubMedID: 36800254

Title : Usefulness of [(68)Ga]FAPI-04 and [(18)F]FDG PET\/CT for the detection of primary tumour and metastatic lesions in gastrointestinal carcinoma: a comparative study - Li_2023_Eur.Radiol_33_2779
Author(s) : Li C , Tian Y , Chen J , Jiang Y , Xue Z , Xing D , Wen B , He Y
Ref : Eur Radiol , 33 :2779 , 2023
Abstract :
PubMedSearch : Li_2023_Eur.Radiol_33_2779
PubMedID: 36394603

Title : Fibroblast Activation Protein Targeting Probe with Gly-Pro Sequence for PET of Glioblastoma - Lai_2023_Mol.Pharm_20_4120
Author(s) : Lai C , Cao R , Li R , He C , Wang X , Shi H , Qu C , Qian K , Song S , Chen WH , Cheng Z
Ref : Mol Pharm , 20 :4120 , 2023
Abstract :
PubMedSearch : Lai_2023_Mol.Pharm_20_4120
PubMedID: 37487027

Title : Impact of 68 Ga-FAPI-04 PET\/CT on Staging and Therapeutic Management in Patients With Digestive System Tumors - Kosmala_2023_Clin.Nucl.Med_48_35
Author(s) : Kosmala A , Serfling SE , Schlotelburg W , Lindner T , Michalski K , Schirbel A , Higuchi T , Hartrampf PE , Buck AK , Weich A , Werner RA
Ref : Clin Nucl Med , 48 :35 , 2023
Abstract :
PubMedSearch : Kosmala_2023_Clin.Nucl.Med_48_35
PubMedID: 36354691

Title : Noninvasive imaging of FAP expression using positron emission tomography: A comparative evaluation of a [(18)F]-labeled glycopeptide-containing FAPI with [(18)F]FAPI-42 - Huang_2023_Eur.J.Nucl.Med.Mol.Imaging_50_3363
Author(s) : Huang J , Fu L , Zhang X , Huang S , Dong Y , Hu K , Han Y , Zhou K , Min C , Huang Y , Tang G
Ref : Eur J Nucl Med Mol Imaging , 50 :3363 , 2023
Abstract :
PubMedSearch : Huang_2023_Eur.J.Nucl.Med.Mol.Imaging_50_3363
PubMedID: 37266596

Title : Fibroblast Activation Protein Inhibitor Theranostics: Early Clinical Translation - Mori_2023_PET.Clin_18_419
Author(s) : Mori Y , Kratochwil C , Haberkorn U , Giesel FL
Ref : PET Clin , 18 :419 , 2023
Abstract :
PubMedSearch : Mori_2023_PET.Clin_18_419
PubMedID: 37030981

Title : Pneumonia with Intense (68)Ga-FAPI Uptake Mimicking Metastasis on (68)Ga-FAPI PET\/CT in a Patient with Rectal Cancer - Erol_2023_Mol.Imaging.Radionucl.Ther_32_237
Author(s) : Erol Fenercioglu O , Beyhan E , Samanci N , Cermik TF , Ergul N
Ref : Mol Imaging Radionucl Ther , 32 :237 , 2023
Abstract :
PubMedSearch : Erol_2023_Mol.Imaging.Radionucl.Ther_32_237
PubMedID: 37870301

Title : Comparison of [(68)Ga]Ga-DOTA-FAPI-04 and [(18)F]FDG PET\/MRI in the Preoperative Diagnosis of Gastric Cancer - Du_2023_Can.J.Gastroenterol.Hepatol_2023_6351330
Author(s) : Du T , Zhang S , Cui XM , Hu RH , Wang HY , Jiang JJ , Zhao J , Zhong L , Jiang XH
Ref : Can J Gastroenterol Hepatol , 2023 :6351330 , 2023
Abstract :
PubMedSearch : Du_2023_Can.J.Gastroenterol.Hepatol_2023_6351330
PubMedID: 37090103

Title : Prognostic value of preoperative [(68) Ga]Ga-FAPI-04 PET\/CT in patients with resectable pancreatic ductal adenocarcinoma in correlation with immunohistological characteristics - Ding_2023_Eur.J.Nucl.Med.Mol.Imaging_50_1780
Author(s) : Ding J , Qiu J , Hao Z , Huang H , Liu Q , Liu W , Ren C , Hacker M , Zhang T , Wu W , Huo L , Li X
Ref : Eur J Nucl Med Mol Imaging , 50 :1780 , 2023
Abstract :
PubMedSearch : Ding_2023_Eur.J.Nucl.Med.Mol.Imaging_50_1780
PubMedID: 36695823

Title : Distinguishing Benign and Malignant Findings on [(68) Ga]-FAPI PET\/CT Based on Quantitative SUV Measurements - Dabir_2023_Mol.Imaging.Biol_25_324
Author(s) : Dabir M , Novruzov E , Mattes-Gyorgy K , Beu M , Dendl K , Antke C , Koerber SA , Rohrich M , Kratochwil C , Debus J , Haberkorn U , Giesel FL
Ref : Mol Imaging Biol , 25 :324 , 2023
Abstract :
PubMedSearch : Dabir_2023_Mol.Imaging.Biol_25_324
PubMedID: 35997853

Title : Feasibility of acquisitions using total-body PET\/CT with a half-dose [(68)Ga]Ga-FAPI-04 activity in oncology patients - Chen_2023_Eur.J.Nucl.Med.Mol.Imaging_50_3961
Author(s) : Chen Z , Wang Y , Yang X , Li L , Huo Y , Yu X , Xiao X , Zhang C , Chen Y , Zhao H , Zhou Y , Huang G , Liu J , Chen R
Ref : Eur J Nucl Med Mol Imaging , 50 :3961 , 2023
Abstract :
PubMedSearch : Chen_2023_Eur.J.Nucl.Med.Mol.Imaging_50_3961
PubMedID: 37535107

Title : Tumor-to-blood ratio for assessment of fibroblast activation protein receptor density in pancreatic cancer using [(68)Ga]Ga-FAPI-04 - Chen_2023_Eur.J.Nucl.Med.Mol.Imaging_50_929
Author(s) : Chen R , Yang X , Yu X , Zhou X , Ng YL , Zhao H , Li L , Huang G , Zhou Y , Liu J
Ref : Eur J Nucl Med Mol Imaging , 50 :929 , 2023
Abstract :
PubMedSearch : Chen_2023_Eur.J.Nucl.Med.Mol.Imaging_50_929
PubMedID: 36334106

Title : The feasibility of ultra-early and fast total-body [(68) Ga]Ga-FAPI-04 PET\/CT scan - Chen_2023_Eur.J.Nucl.Med.Mol.Imaging_50_661
Author(s) : Chen R , Yang X , Yu X , Zhou X , Ng YL , Chen Y , Li L , Zhou Y , Huang G , Liu J
Ref : Eur J Nucl Med Mol Imaging , 50 :661 , 2023
Abstract :
PubMedSearch : Chen_2023_Eur.J.Nucl.Med.Mol.Imaging_50_661
PubMedID: 36308535

Title : First Total-Body Kinetic Modeling and Parametric Imaging of Dynamic (68)Ga-FAPI-04 PET in Pancreatic and Gastric Cancer - Chen_2023_J.Nucl.Med_64_960
Author(s) : Chen R , Yang X , Ng YL , Yu X , Huo Y , Xiao X , Zhang C , Chen Y , Zheng C , Li L , Huang G , Zhou Y , Liu J
Ref : J Nucl Med , 64 :960 , 2023
Abstract :
PubMedSearch : Chen_2023_J.Nucl.Med_64_960
PubMedID: 36604180

Title : 68 Ga-FAPI-04 PET\/CT in Selected Breast Cancer Patients With Low FDG Affinity : A Head-to-Head Comparative Study - Alcin_2023_Clin.Nucl.Med_48_e420
Author(s) : Alcin G , Arslan E , Aksoy T , Cin M , Erol Fenercioglu O , Beyhan E , Ergul N , Cermik TF
Ref : Clin Nucl Med , 48 :e420 , 2023
Abstract :
PubMedSearch : Alcin_2023_Clin.Nucl.Med_48_e420
PubMedID: 37351868

Title : Synthesis and Preclinical Evaluation of a Novel FAPI-04 Dimer for Cancer Theranostics - Zhong_2023_Mol.Pharm_20_2402
Author(s) : Zhong X , Guo J , Han X , Wu W , Yang R , Zhang J , Shao G
Ref : Mol Pharm , 20 :2402 , 2023
Abstract :
PubMedSearch : Zhong_2023_Mol.Pharm_20_2402
PubMedID: 37015025

Title : Physiological Uptake Characteristics of Breast on (68)Ga-FAPI-04 PET\/CT - Zhang_2023_Mol.Imaging.Biol_25_1045
Author(s) : Zhang Y , Zhou Y , Tian R , Su M
Ref : Mol Imaging Biol , 25 :1045 , 2023
Abstract :
PubMedSearch : Zhang_2023_Mol.Imaging.Biol_25_1045
PubMedID: 37945972

Title : Dynamic PET\/CT scan of (68)Ga-FAPI-04 for the optimal acquisition time in suspected malignant hepatic cancer patients - Xing_2023_Abdom.Radiol.(NY)_48_895
Author(s) : Xing H , Hu G , Zhu W , Dong C , Shi X , Li F , Huo L
Ref : Abdom Radiol (NY) , 48 :895 , 2023
Abstract :
PubMedSearch : Xing_2023_Abdom.Radiol.(NY)_48_895
PubMedID: 36583752

Title : Increased uptake of (68)Ga-DOTA-FAPI-04 in bones and joints: metastases and beyond - Qin_2022_Eur.J.Nucl.Med.Mol.Imaging_49_709
Author(s) : Qin C , Song Y , Liu X , Gai Y , Liu Q , Ruan W , Liu F , Hu F , Lan X
Ref : Eur J Nucl Med Mol Imaging , 49 :709 , 2022
Abstract :
PubMedSearch : Qin_2022_Eur.J.Nucl.Med.Mol.Imaging_49_709
PubMedID: 34241652

Title : Noninvasive Monitoring of Reparative Fibrosis after Myocardial Infarction in Rats Using (68)Ga-FAPI-04 PET\/CT - Qiao_2022_Mol.Pharm_19_4171
Author(s) : Qiao P , Wang Y , Zhu K , Zheng D , Song Y , Jiang D , Qin C , Lan X
Ref : Mol Pharm , 19 :4171 , 2022
Abstract :
PubMedSearch : Qiao_2022_Mol.Pharm_19_4171
PubMedID: 35969029

Title : Non-tumoral uptake of (68)Ga-FAPI-04 PET: A retrospective study - Qi_2022_Front.Oncol_12_989595
Author(s) : Qi N , Wang H , Ren S , You Z , Chen X , Guan Y , Xie F , Hua F , Zhao J
Ref : Front Oncol , 12 :989595 , 2022
Abstract :
PubMedSearch : Qi_2022_Front.Oncol_12_989595
PubMedID: 36531015

Title : Imaging of cardiac fibroblast activation in a patient after acute myocardial infarction using (68)Ga-FAPI-04 - Notohamiprodjo_2022_J.Nucl.Cardiol_29_2254
Author(s) : Notohamiprodjo S , Nekolla SG , Robu S , Villagran Asiares A , Kupatt C , Ibrahim T , Laugwitz KL , Makowski MR , Schwaiger M , Weber WA , Varasteh Z
Ref : J Nucl Cardiol , 29 :2254 , 2022
Abstract :
PubMedSearch : Notohamiprodjo_2022_J.Nucl.Cardiol_29_2254
PubMedID: 33860458

Title : Comparison of physiological uptake of normal tissues in patients with cancer using (18)F-FAPI-04 and (18)F-FAPI-42 PET\/CT - Mu_2022_Front.Nucl.Med_2_927843
Author(s) : Mu X , Huang X , Li M , Sun W , Fu W
Ref : Front Nucl Med , 2 :927843 , 2022
Abstract :
PubMedSearch : Mu_2022_Front.Nucl.Med_2_927843
PubMedID: 39354982

Title : Feasibility, Biodistribution, and Preliminary Dosimetry in Peptide-Targeted Radionuclide Therapy of Diverse Adenocarcinomas Using (177)Lu-FAP-2286: First-in-Humans Results - Baum_2022_J.Nucl.Med_63_415
Author(s) : Baum RP , Schuchardt C , Singh A , Chantadisai M , Robiller FC , Zhang J , Mueller D , Eismant A , Almaguel F , Zboralski D , Osterkamp F , Hoehne A , Reineke U , Smerling C , Kulkarni HR
Ref : J Nucl Med , 63 :415 , 2022
Abstract :
PubMedSearch : Baum_2022_J.Nucl.Med_63_415
PubMedID: 34168013

Title : Non-oncologic incidental uptake on FAPI PET\/CT imaging - Hotta_2022_Br.J.Radiol__20220463
Author(s) : Hotta M , Rieger AC , Jafarvand MG , Menon N , Farolfi A , Benz MR , Calais J
Ref : Br J Radiol , :20220463 , 2022
Abstract :
PubMedSearch : Hotta_2022_Br.J.Radiol__20220463
PubMedID: 35776566

Title : Comparison of [(68)Ga]Ga-DOTA-FAPI-04 and [(18)F]FDG Uptake in Esophageal Cancer - Liu_2022_Front.Oncol_12_875081
Author(s) : Liu H , Hu Z , Yang X , Dai T , Chen Y
Ref : Front Oncol , 12 :875081 , 2022
Abstract :
PubMedSearch : Liu_2022_Front.Oncol_12_875081
PubMedID: 35785188

Title : [(68)Ga]Ga-DOTA-FAPI-04 PET\/CT in the evaluation of gastric cancer: comparison with [(18)F]FDG PET\/CT - Lin_2022_Eur.J.Nucl.Med.Mol.Imaging_49_2960
Author(s) : Lin R , Lin Z , Chen Z , Zheng S , Zhang J , Zang J , Miao W
Ref : Eur J Nucl Med Mol Imaging , 49 :2960 , 2022
Abstract :
PubMedSearch : Lin_2022_Eur.J.Nucl.Med.Mol.Imaging_49_2960
PubMedID: 35462566

Title : A systematic review of [(68)Ga]Ga-DOTA-FAPI-04 and [(18)F]FDG PET\/CT in the diagnostic value of malignant tumor bone metastasis - Li_2022_Front.Oncol_12_978506
Author(s) : Li L , Hu X , Ma J , Yang S , Gong W , Zhang C
Ref : Front Oncol , 12 :978506 , 2022
Abstract :
PubMedSearch : Li_2022_Front.Oncol_12_978506
PubMedID: 36439440

Title : The potential utility of [(68) Ga]Ga-DOTA-FAPI-04 as a novel broad-spectrum oncological and non-oncological imaging agent-comparison with [(18)F]FDG - Lan_2022_Eur.J.Nucl.Med.Mol.Imaging_49_963
Author(s) : Lan L , Liu H , Wang Y , Deng J , Peng D , Feng Y , Wang L , Chen Y , Qiu L
Ref : Eur J Nucl Med Mol Imaging , 49 :963 , 2022
Abstract :
PubMedSearch : Lan_2022_Eur.J.Nucl.Med.Mol.Imaging_49_963
PubMedID: 34410435

Title : Pitfalls and Common Findings in (68)Ga-FAPI PET: A Pictorial Analysis - Kessler_2022_J.Nucl.Med_63_890
Author(s) : Kessler L , Ferdinandus J , Hirmas N , Zarrad F , Nader M , Kersting D , Weber M , Kazek S , Sraieb M , Hamacher R , Lueckerath K , Umutlu L , Fendler WP , Rischpler C
Ref : J Nucl Med , 63 :890 , 2022
Abstract :
PubMedSearch : Kessler_2022_J.Nucl.Med_63_890
PubMedID: 34620730

Title : Head-to-head comparison of [(68)Ga]Ga-FAPI-04 and [(18)F]-FDG PET\/CT in evaluating the extent of disease in gastric adenocarcinoma - Kuten_2022_Eur.J.Nucl.Med.Mol.Imaging_49_743
Author(s) : Kuten J , Levine C , Shamni O , Pelles S , Wolf I , Lahat G , Mishani E , Even-Sapir E
Ref : Eur J Nucl Med Mol Imaging , 49 :743 , 2022
Abstract :
PubMedSearch : Kuten_2022_Eur.J.Nucl.Med.Mol.Imaging_49_743
PubMedID: 34302504

Title : Comparison of [(68) Ga]Ga-DOTA-FAPI-04 PET\/CT and [(18)F]FDG PET\/CT in colorectal cancer - Komek_2022_Eur.J.Nucl.Med.Mol.Imaging_49_3898
Author(s) : Komek H , Can C , Kaplan I , Gundogan C , Kepenek F , Karaoglan H , Demirkiran A , Ebinc S , Guzel Y , Gundes E
Ref : Eur J Nucl Med Mol Imaging , 49 :3898 , 2022
Abstract :
PubMedSearch : Komek_2022_Eur.J.Nucl.Med.Mol.Imaging_49_3898
PubMedID: 35578038

Title : Comparison of [(68) Ga]Ga-FAPI-04 and [(18)F]-FDG for the detection of primary and metastatic lesions in patients with gastric cancer: a bicentric retrospective study - Jiang_2022_Eur.J.Nucl.Med.Mol.Imaging_49_732
Author(s) : Jiang D , Chen X , You Z , Wang H , Zhang X , Li X , Ren S , Huang Q , Hua F , Guan Y , Zhao J , Xie F
Ref : Eur J Nucl Med Mol Imaging , 49 :732 , 2022
Abstract :
PubMedSearch : Jiang_2022_Eur.J.Nucl.Med.Mol.Imaging_49_732
PubMedID: 34297193

Title : [(18)F]FAPI-42 PET imaging in cancer patients: optimal acquisition time, biodistribution, and comparison with [(68)Ga]Ga-FAPI-04 - Hu_2022_Eur.J.Nucl.Med.Mol.Imaging_49_2833
Author(s) : Hu K , Wang L , Wu H , Huang S , Tian Y , Wang Q , Xiao C , Han Y , Tang G
Ref : Eur J Nucl Med Mol Imaging , 49 :2833 , 2022
Abstract :
PubMedSearch : Hu_2022_Eur.J.Nucl.Med.Mol.Imaging_49_2833
PubMedID: 34893920

Title : Head-to-head evaluation of [(18)F]FDG and [(68) Ga]Ga-DOTA-FAPI-04 PET\/CT in recurrent soft tissue sarcoma - Gu_2022_Eur.J.Nucl.Med.Mol.Imaging_49_2889
Author(s) : Gu B , Liu X , Wang S , Xu X , Hu S , Yan W , Luo Z , Song S
Ref : Eur J Nucl Med Mol Imaging , 49 :2889 , 2022
Abstract :
PubMedSearch : Gu_2022_Eur.J.Nucl.Med.Mol.Imaging_49_2889
PubMedID: 35113192

Title : 86Y-Labeled Albumin-Binding Fibroblast Activation Protein Inhibitor for Late-Time-Point Cancer Diagnosis - Ding_2022_Mol.Pharm_19_3429
Author(s) : Ding J , Xu M , Chen J , Zhang P , Huo L , Kong Z , Liu Z
Ref : Mol Pharm , 19 :3429 , 2022
Abstract :
PubMedSearch : Ding_2022_Mol.Pharm_19_3429
PubMedID: 35976352

Title : Prospective comparison of (68)Ga-FAPI-04 and (18)F-FDG PET\/CT for tumor staging in nasopharyngeal carcinoma - Ding_2022_Front.Oncol_12_1047010
Author(s) : Ding H , Liang J , Qiu L , Xu T , Cai L , Wan Q , Wang L , Liu Y , Chen Y
Ref : Front Oncol , 12 :1047010 , 2022
Abstract :
PubMedSearch : Ding_2022_Front.Oncol_12_1047010
PubMedID: 36568172

Title : (68)Ga-DOTA-FAPI-04 PET\/CT imaging in radioiodine-refractory differentiated thyroid cancer (RR-DTC) patients - Chen_2022_Ann.Nucl.Med_36_610
Author(s) : Chen Y , Zheng S , Zhang J , Yao S , Miao W
Ref : Ann Nucl Med , 36 :610 , 2022
Abstract :
PubMedSearch : Chen_2022_Ann.Nucl.Med_36_610
PubMedID: 35551610

Title : Radiosynthesis and First Preclinical Evaluation of the Novel (11)C-Labeled FAP Inhibitor (11)C-FAPI: A Comparative Study of (11)C-FAPIs and ((68)Ga) Ga-DOTA-FAPI-04 in a High-FAP-Expression Mouse Model - Wang_2022_Front.Chem_10_939160
Author(s) : Wang C , Hu Z , Ding F , Zhao H , Du F , Lv C , Li L , Huang G , Liu J
Ref : Front Chem , 10 :939160 , 2022
Abstract :
PubMedSearch : Wang_2022_Front.Chem_10_939160
PubMedID: 35991604

Title : Comparison of the diagnostic efficacy of (68) Ga-FAPI-04 PET\/MR and (18)F-FDG PET\/CT in patients with pancreatic cancer - Zhang_2022_Eur.J.Nucl.Med.Mol.Imaging_49_2877
Author(s) : Zhang Z , Jia G , Pan G , Cao K , Yang Q , Meng H , Yang J , Zhang L , Wang T , Cheng C , Zuo C
Ref : Eur J Nucl Med Mol Imaging , 49 :2877 , 2022
Abstract :
PubMedSearch : Zhang_2022_Eur.J.Nucl.Med.Mol.Imaging_49_2877
PubMedID: 35243518

Title : Comparison of Diagnostic Efficacy of [(68)Ga]Ga-FAPI-04 and [(18)F]FDG PET\/CT for Staging and Restaging of Gastric Cancer - Zhang_2022_Front.Oncol_12_925100
Author(s) : Zhang S , Wang W , Xu T , Ding H , Li Y , Liu H , Huang Y , Liu L , Du T , Zhao Y , Chen Y , Qiu L
Ref : Front Oncol , 12 :925100 , 2022
Abstract :
PubMedSearch : Zhang_2022_Front.Oncol_12_925100
PubMedID: 35847877

Title : The Application of [(68)Ga]-Labeled FAPI-04 PET\/CT for Targeting and Early Detection of Pancreatic Carcinoma in Patient-Derived Orthotopic Xenograft Models - Zhang_2022_Contrast.Media.Mol.Imaging_2022_6596702
Author(s) : Zhang H , An J , Wu P , Zhang C , Zhao Y , Tan D , Shi C , Ge X
Ref : Contrast Media Mol Imaging , 2022 :6596702 , 2022
Abstract :
PubMedSearch : Zhang_2022_Contrast.Media.Mol.Imaging_2022_6596702
PubMedID: 36051919

Title : Head-tohead assessment of [(68)Ga]Ga-DOTA-FAPI-04 PET\/CT vs [(18)F]FDG PET\/CT in fibroblastic tumors - Zhang_2022_Eur.J.Radiol_155_110507
Author(s) : Zhang A , Meng X , Yao Y , Zhou X , Zhang Y , Li N
Ref : Eur J Radiol , 155 :110507 , 2022
Abstract :
PubMedSearch : Zhang_2022_Eur.J.Radiol_155_110507
PubMedID: 36075176

Title : Albumin Binder-Conjugated Fibroblast Activation Protein Inhibitor Radiopharmaceuticals for Cancer Therapy - Xu_2022_J.Nucl.Med_63_952
Author(s) : Xu M , Zhang P , Ding J , Chen J , Huo L , Liu Z
Ref : J Nucl Med , 63 :952 , 2022
Abstract :
PubMedSearch : Xu_2022_J.Nucl.Med_63_952
PubMedID: 34593598

Title : [(18)F]AlF-NOTA-FAPI-04: FAP-targeting specificity, biodistribution, and PET\/CT imaging of various cancers - Wei_2022_Eur.J.Nucl.Med.Mol.Imaging_49_2761
Author(s) : Wei Y , Zheng J , Ma L , Liu X , Xu S , Wang S , Pei J , Cheng K , Yuan S , Yu J
Ref : Eur J Nucl Med Mol Imaging , 49 :2761 , 2022
Abstract :
PubMedSearch : Wei_2022_Eur.J.Nucl.Med.Mol.Imaging_49_2761
PubMedID: 35262766

Title : [(18)F]AlF-NOTA-FAPI-04 PET\/CT uptake in metastatic lesions on PET\/CT imaging might distinguish different pathological types of lung cancer - Wei_2022_Eur.J.Nucl.Med.Mol.Imaging_49_1671
Author(s) : Wei Y , Cheng K , Fu Z , Zheng J , Mu Z , Zhao C , Liu X , Wang S , Yu J , Yuan S
Ref : Eur J Nucl Med Mol Imaging , 49 :1671 , 2022
Abstract :
PubMedSearch : Wei_2022_Eur.J.Nucl.Med.Mol.Imaging_49_1671
PubMedID: 34870727

Title : (68)Ga-DOTA-FAPI-04 PET\/CT as a Promising Tool for Differentiating Ovarian Physiological Uptake: Preliminary Experience of Comparative Analysis With (18)F-FDG - Wang_2021_Front.Med.(Lausanne)_8_748683
Author(s) : Wang Q , Yang S , Tang W , Liu L , Chen Y
Ref : Front Med (Lausanne) , 8 :748683 , 2021
Abstract :
PubMedSearch : Wang_2021_Front.Med.(Lausanne)_8_748683
PubMedID: 34671627

Title : (68)Ga-FAPI-04 Versus (18)F-FDG PET\/CT in the Detection of Hepatocellular Carcinoma - Wang_2021_Front.Oncol_11_693640
Author(s) : Wang H , Zhu W , Ren S , Kong Y , Huang Q , Zhao J , Guan Y , Jia H , Chen J , Lu L , Xie F , Qin L
Ref : Front Oncol , 11 :693640 , 2021
Abstract :
PubMedSearch : Wang_2021_Front.Oncol_11_693640
PubMedID: 34249748

Title : Fibroblast imaging of hepatic carcinoma with (68)Ga-FAPI-04 PET\/CT: a pilot study in patients with suspected hepatic nodules - Shi_2021_Eur.J.Nucl.Med.Mol.Imaging_48_196
Author(s) : Shi X , Xing H , Yang X , Li F , Yao S , Zhang H , Zhao H , Hacker M , Huo L , Li X
Ref : Eur J Nucl Med Mol Imaging , 48 :196 , 2021
Abstract :
PubMedSearch : Shi_2021_Eur.J.Nucl.Med.Mol.Imaging_48_196
PubMedID: 32468254

Title : A head-to-head comparison of (68)Ga-DOTA-FAPI-04 and (18)F-FDG PET\/MR in patients with nasopharyngeal carcinoma: a prospective study - Qin_2021_Eur.J.Nucl.Med.Mol.Imaging_48_3228
Author(s) : Qin C , Liu F , Huang J , Ruan W , Liu Q , Gai Y , Hu F , Jiang D , Hu Y , Yang K , Lan X
Ref : Eur J Nucl Med Mol Imaging , 48 :3228 , 2021
Abstract :
PubMedSearch : Qin_2021_Eur.J.Nucl.Med.Mol.Imaging_48_3228
PubMedID: 33609152

Title : High fibroblast-activation-protein expression in castration-resistant prostate cancer supports the use of FAPI-molecular theranostics - Kesch_2021_Eur.J.Nucl.Med.Mol.Imaging_49_385
Author(s) : Kesch C , Yirga L , Dendl K , Handke A , Darr C , Krafft U , Radtke JP , Tschirdewahn S , Szarvas T , Fazli L , Gleave M , Giesel FL , Haberkorn U , Hadaschik B
Ref : Eur J Nucl Med Mol Imaging , 49 :385 , 2021
Abstract :
PubMedSearch : Kesch_2021_Eur.J.Nucl.Med.Mol.Imaging_49_385
PubMedID: 34226953

Title : Imaging fibroblast activation protein in liver cancer: a single-center post hoc retrospective analysis to compare [(68)Ga]Ga-FAPI-04 PET\/CT versus MRI and [(18)F]-FDG PET\/CT - Guo_2021_Eur.J.Nucl.Med.Mol.Imaging_48_1604
Author(s) : Guo W , Pang Y , Yao L , Zhao L , Fan C , Ke J , Guo P , Hao B , Fu H , Xie C , Lin Q , Wu H , Sun L , Chen H
Ref : Eur J Nucl Med Mol Imaging , 48 :1604 , 2021
Abstract :
PubMedSearch : Guo_2021_Eur.J.Nucl.Med.Mol.Imaging_48_1604
PubMedID: 33179149

Title : FAPI-04 Uptake in Healthy Tissues of Cancer Patients in (68)Ga-FAPI-04 PET\/CT Imaging - Gundogan_2021_Contrast.Media.Mol.Imaging_2021_9750080
Author(s) : Gundogan C , Guzel Y , Can C , Kaplan I , Komek H
Ref : Contrast Media Mol Imaging , 2021 :9750080 , 2021
Abstract :
PubMedSearch : Gundogan_2021_Contrast.Media.Mol.Imaging_2021_9750080
PubMedID: 34887714

Title : Usefulness of [(68)Ga]Ga-DOTA-FAPI-04 PET\/CT in patients presenting with inconclusive [(18)F]FDG PET\/CT findings - Chen_2021_Eur.J.Nucl.Med.Mol.Imaging_48_73
Author(s) : Chen H , Zhao L , Ruan D , Pang Y , Hao B , Dai Y , Wu X , Guo W , Fan C , Wu J , Huang W , Lin Q , Sun L , Wu H
Ref : Eur J Nucl Med Mol Imaging , 48 :73 , 2021
Abstract :
PubMedSearch : Chen_2021_Eur.J.Nucl.Med.Mol.Imaging_48_73
PubMedID: 32588089

Title : Rational Design, Pharmacomodulation, and Synthesis of [(68)Ga]Ga-Alb-FAPtp-01, a Selective Tumor-Associated Fibroblast Activation Protein Tracer for PET Imaging of Glioma - Lin_2021_ACS.Sens_6_3424
Author(s) : Lin JJ , Chuang CP , Lin JY , Huang FT , Huang CW
Ref : ACS Sens , 6 :3424 , 2021
Abstract :
PubMedSearch : Lin_2021_ACS.Sens_6_3424
PubMedID: 34415143
Gene_locus related to this paper: human-FAP

Title : Clinical translational evaluation of Al(18)F-NOTA-FAPI for fibroblast activation protein-targeted tumour imaging - Wang_2021_Eur.J.Nucl.Med.Mol.Imaging_48_4259
Author(s) : Wang S , Zhou X , Xu X , Ding J , Liu S , Hou X , Li N , Zhu H , Yang Z
Ref : Eur J Nucl Med Mol Imaging , 48 :4259 , 2021
Abstract :
PubMedSearch : Wang_2021_Eur.J.Nucl.Med.Mol.Imaging_48_4259
PubMedID: 34165601

Title : Dynamic PET\/CT Imaging of (68)Ga-FAPI-04 in Chinese Subjects - Wang_2021_Front.Oncol_11_651005
Author(s) : Wang S , Zhou X , Xu X , Ding J , Liu T , Jiang J , Li N , Zhu H , Yang Z
Ref : Front Oncol , 11 :651005 , 2021
Abstract :
PubMedSearch : Wang_2021_Front.Oncol_11_651005
PubMedID: 33777814
Gene_locus related to this paper: human-FAP

Title : Value of [(68)Ga]Ga-FAPI-04 imaging in the diagnosis of renal fibrosis - Zhou_2021_Eur.J.Nucl.Med.Mol.Imaging_48_3493
Author(s) : Zhou Y , Yang X , Liu H , Luo W , Lv T , Wang J , Qin J , Ou S , Chen Y
Ref : Eur J Nucl Med Mol Imaging , 48 :3493 , 2021
Abstract :
PubMedSearch : Zhou_2021_Eur.J.Nucl.Med.Mol.Imaging_48_3493
PubMedID: 33829416

Title : Characterization of the benign lesions with increased (68)Ga-FAPI-04 uptake in PET\/CT - Zheng_2021_Ann.Nucl.Med_35_1312
Author(s) : Zheng S , Lin R , Chen S , Zheng J , Lin Z , Zhang Y , Xue Q , Chen Y , Zhang J , Lin K , You X , Yao S , Miao W
Ref : Ann Nucl Med , 35 :1312 , 2021
Abstract :
PubMedSearch : Zheng_2021_Ann.Nucl.Med_35_1312
PubMedID: 34424505

Title : Role of [(68)Ga]Ga-DOTA-FAPI-04 PET\/CT in the evaluation of peritoneal carcinomatosis and comparison with [(18)F]-FDG PET\/CT - Zhao_2021_Eur.J.Nucl.Med.Mol.Imaging_48_1944
Author(s) : Zhao L , Pang Y , Luo Z , Fu K , Yang T , Sun L , Wu H , Lin Q , Chen H
Ref : Eur J Nucl Med Mol Imaging , 48 :1944 , 2021
Abstract :
PubMedSearch : Zhao_2021_Eur.J.Nucl.Med.Mol.Imaging_48_1944
PubMedID: 33415432

Title : Non-malignant findings of focal (68)Ga-FAPI-04 uptake in pancreas - Zhang_2021_Eur.J.Nucl.Med.Mol.Imaging_48_2635
Author(s) : Zhang X , Song W , Qin C , Liu F , Lan X
Ref : Eur J Nucl Med Mol Imaging , 48 :2635 , 2021
Abstract :
PubMedSearch : Zhang_2021_Eur.J.Nucl.Med.Mol.Imaging_48_2635
PubMedID: 33452634

Title : Comparison of the Relative Diagnostic Performance of [(68)Ga]Ga-DOTA-FAPI-04 and [(18)F]FDG PET\/CT for the Detection of Bone Metastasis in Patients With Different Cancers - Wu_2021_Front.Oncol_11_737827
Author(s) : Wu J , Wang Y , Liao T , Rao Z , Gong W , Ou L , Chen Y , Zhang C
Ref : Front Oncol , 11 :737827 , 2021
Abstract :
PubMedSearch : Wu_2021_Front.Oncol_11_737827
PubMedID: 34604078

Title : FAP-specific PET signaling shows a moderately positive correlation with relative CBV and no correlation with ADC in 13 IDH wildtype glioblastomas - Rohrich_2020_Eur.J.Radiol_127_109021
Author(s) : Rohrich M , Floca R , Loi L , Adeberg S , Windisch P , Giesel FL , Kratochwil C , Flechsig P , Rathke H , Lindner T , Loktev A , Schlemmer HP , Haberkorn U , Paech D
Ref : Eur J Radiol , 127 :109021 , 2020
Abstract :
PubMedSearch : Rohrich_2020_Eur.J.Radiol_127_109021
PubMedID: 32344293
Gene_locus related to this paper: human-FAP

Title : The Role of (68)Ga-FAPI PET\/CT for Patients with Malignancies of the Lower Gastrointestinal Tract: First Clinical Experience - Koerber_2020_J.Nucl.Med_61_1331
Author(s) : Koerber SA , Staudinger F , Kratochwil C , Adeberg S , Haefner MF , Ungerechts G , Rathke H , Winter E , Lindner T , Syed M , Bhatti IA , Herfarth K , Choyke PL , Jaeger D , Haberkorn U , Debus J , Giesel FL
Ref : J Nucl Med , 61 :1331 , 2020
Abstract :
PubMedSearch : Koerber_2020_J.Nucl.Med_61_1331
PubMedID: 32060216

Title : Radiation Dosimetry and Biodistribution of (68)Ga-FAPI-46 PET Imaging in Cancer Patients - Meyer_2020_J.Nucl.Med_61_1171
Author(s) : Meyer C , Dahlbom M , Lindner T , Vauclin S , Mona C , Slavik R , Czernin J , Haberkorn U , Calais J
Ref : J Nucl Med , 61 :1171 , 2020
Abstract :
PubMedSearch : Meyer_2020_J.Nucl.Med_61_1171
PubMedID: 31836685

Title : Comparison of [(68)Ga]Ga-DOTA-FAPI-04 and [(18)F] FDG PET\/CT for the diagnosis of primary and metastatic lesions in patients with various types of cancer - Chen_2020_Eur.J.Nucl.Med.Mol.Imaging_47_1820
Author(s) : Chen H , Pang Y , Wu J , Zhao L , Hao B , Wei J , Wu S , Luo Z , Lin X , Xie C , Sun L , Lin Q , Wu H
Ref : Eur J Nucl Med Mol Imaging , 47 :1820 , 2020
Abstract :
PubMedSearch : Chen_2020_Eur.J.Nucl.Med.Mol.Imaging_47_1820
PubMedID: 32222810

Title : Theranostics Targeting Fibroblast Activation Protein in the Tumor Stroma: (64)Cu- and (225)Ac-Labeled FAPI-04 in Pancreatic Cancer Xenograft Mouse Models - Watabe_2020_J.Nucl.Med_61_563
Author(s) : Watabe T , Liu Y , Kaneda-Nakashima K , Shirakami Y , Lindner T , Ooe K , Toyoshima A , Nagata K , Shimosegawa E , Haberkorn U , Kratochwil C , Shinohara A , Giesel F , Hatazawa J
Ref : J Nucl Med , 61 :563 , 2020
Abstract :
PubMedSearch : Watabe_2020_J.Nucl.Med_61_563
PubMedID: 31586001

Title : IDH-wildtype glioblastomas and grade III\/IV IDH-mutant gliomas show elevated tracer uptake in fibroblast activation protein-specific PET\/CT - Rohrich_2019_Eur.J.Nucl.Med.Mol.Imaging_46_2569
Author(s) : Rohrich M , Loktev A , Wefers AK , Altmann A , Paech D , Adeberg S , Windisch P , Hielscher T , Flechsig P , Floca R , Leitz D , Schuster JP , Huber PE , Debus J , von Deimling A , Lindner T , Haberkorn U
Ref : Eur J Nucl Med Mol Imaging , 46 :2569 , 2019
Abstract :
PubMedSearch : Rohrich_2019_Eur.J.Nucl.Med.Mol.Imaging_46_2569
PubMedID: 31388723

Title : Molecular Imaging of Fibroblast Activity After Myocardial Infarction Using a (68)Ga-Labeled Fibroblast Activation Protein Inhibitor, FAPI-04 - Varasteh_2019_J.Nucl.Med_60_1743
Author(s) : Varasteh Z , Mohanta S , Robu S , Braeuer M , Li Y , Omidvari N , Topping G , Sun T , Nekolla SG , Richter A , Weber C , Habenicht A , Haberkorn UA , Weber WA
Ref : J Nucl Med , 60 :1743 , 2019
Abstract :
PubMedSearch : Varasteh_2019_J.Nucl.Med_60_1743
PubMedID: 31405922

Title : (68)Ga-FAPI PET\/CT: Tracer Uptake in 28 Different Kinds of Cancer - Kratochwil_2019_J.Nucl.Med_60_801
Author(s) : Kratochwil C , Flechsig P , Lindner T , Abderrahim L , Altmann A , Mier W , Adeberg S , Rathke H , Rohrich M , Winter H , Plinkert PK , Marme F , Lang M , Kauczor HU , Jager D , Debus J , Haberkorn U , Giesel FL
Ref : J Nucl Med , 60 :801 , 2019
Abstract :
PubMedSearch : Kratochwil_2019_J.Nucl.Med_60_801
PubMedID: 30954939

Title : A Tumor-Imaging Method Targeting Cancer-Associated Fibroblasts - Loktev_2018_J.Nucl.Med_59_1423
Author(s) : Loktev A , Lindner T , Mier W , Debus J , Altmann A , Jager D , Giesel F , Kratochwil C , Barthe P , Roumestand C , Haberkorn U
Ref : J Nucl Med , 59 :1423 , 2018
Abstract :
PubMedSearch : Loktev_2018_J.Nucl.Med_59_1423
PubMedID: 29626120
Gene_locus related to this paper: human-FAP

Title : Development of Quinoline-Based Theranostic Ligands for the Targeting of Fibroblast Activation Protein - Lindner_2018_J.Nucl.Med_59_1415
Author(s) : Lindner T , Loktev A , Altmann A , Giesel F , Kratochwil C , Debus J , Jager D , Mier W , Haberkorn U
Ref : J Nucl Med , 59 :1415 , 2018
Abstract :
PubMedSearch : Lindner_2018_J.Nucl.Med_59_1415
PubMedID: 29626119
Gene_locus related to this paper: human-FAP