Title : Identification of Reversible Small Molecule Inhibitors of Endothelial Lipase (EL) That Demonstrate HDL-C Increase In Vivo - Tora_2020_J.Med.Chem_63_1660 |
Author(s) : Tora G , Kim SH , Pi Z , Johnson JA , Jiang J , Phillips M , Lloyd J , Abell LM , Lu H , Locke G , Adam LP , Taylor DS , Yin X , Behnia K , Zhao L , Yang R , Basso M , Caporuscio C , Chen AY , Liu E , Kirshgessner T , Onorato JM , Ryan C , Traeger SC , Gordon D , Wexler RR , Finlay HJ |
Ref : Journal of Medicinal Chemistry , 63 :1660 , 2020 |
Abstract : |
PubMedSearch : Tora_2020_J.Med.Chem_63_1660 |
PubMedID: 31990537 |
Title : Identification of substituted benzothiazole sulfones as potent and selective inhibitors of endothelial lipase - Kim_2019_Bioorg.Med.Chem.Lett_29_1918 |
Author(s) : Kim SH , Johnson JA , Jiang J , Parkhurst B , Phillips M , Pi Z , Qiao JX , Tora G , Ye Chen A , Liu E , Yin X , Yang R , Zhao L , Taylor DS , Basso M , Behnia K , Onorato J , Chen XQ , Abell LM , Lu H , Locke G , Caporuscio C , Adam LP , Gordon D , Wexler RR , Finlay HJ |
Ref : Bioorganic & Medicinal Chemistry Lett , 29 :1918 , 2019 |
Abstract : |
PubMedSearch : Kim_2019_Bioorg.Med.Chem.Lett_29_1918 |
PubMedID: 31176700 |
Gene_locus related to this paper: human-LIPG |
Title : Sulfonylated Benzothiazoles as Inhibitors of Endothelial Lipase - Johnson_2018_ACS.Med.Chem.Lett_9_1263 |
Author(s) : Johnson JA , Tora G , Pi Z , Phillips M , Yin X , Yang R , Zhao L , Chen AY , Taylor DS , Basso M , Rose A , Behnia K , Onorato J , Chen XQ , Abell LM , Lu H , Locke G , Caporuscio C , Galella M , Adam LP , Gordon D , Wexler RR , Finlay HJ |
Ref : ACS Med Chem Lett , 9 :1263 , 2018 |
Abstract : |
PubMedSearch : Johnson_2018_ACS.Med.Chem.Lett_9_1263 |
PubMedID: 30613337 |
Gene_locus related to this paper: human-LIPG |
Title : Discovery and synthesis of tetrahydropyrimidinedione-4-carboxamides as endothelial lipase inhibitors - Hu_2018_Bioorg.Med.Chem.Lett_28_3721 |
Author(s) : Hu CH , Wang TC , Qiao JX , Haque L , Chen AYA , Taylor DS , Ying X , Onorato JM , Galella M , Shen H , Huang CS , Toussaint N , Li YX , Abell L , Adam LP , Gordon D , Wexler RR , Finlay HJ |
Ref : Bioorganic & Medicinal Chemistry Lett , 28 :3721 , 2018 |
Abstract : |
PubMedSearch : Hu_2018_Bioorg.Med.Chem.Lett_28_3721 |
PubMedID: 30348490 |
Title : Autonomic remodeling in the left atrium and pulmonary veins in heart failure: creation of a dynamic substrate for atrial fibrillation - Ng_2011_Circ.Arrhythm.Electrophysiol_4_388 |
Author(s) : Ng J , Villuendas R , Cokic I , Schliamser JE , Gordon D , Koduri H , Benefield B , Simon J , Murthy SN , Lomasney JW , Wasserstrom JA , Goldberger JJ , Aistrup GL , Arora R |
Ref : Circ Arrhythm Electrophysiol , 4 :388 , 2011 |
Abstract : |
PubMedSearch : Ng_2011_Circ.Arrhythm.Electrophysiol_4_388 |
PubMedID: 21421805 |
Title : Quantitative analysis of parasympathetic innervation of the porcine heart - Ulphani_2010_Heart.Rhythm_7_1113 |
Author(s) : Ulphani JS , Cain JH , Inderyas F , Gordon D , Gikas PV , Shade G , Mayor D , Arora R , Kadish AH , Goldberger JJ |
Ref : Heart Rhythm , 7 :1113 , 2010 |
Abstract : |
PubMedSearch : Ulphani_2010_Heart.Rhythm_7_1113 |
PubMedID: 20381645 |
Title : The ligament of Marshall as a parasympathetic conduit - Ulphani_2007_Am.J.Physiol.Heart.Circ.Physiol_293_H1629 |
Author(s) : Ulphani JS , Arora R , Cain JH , Villuendas R , Shen S , Gordon D , Inderyas F , Harvey LA , Morris A , Goldberger JJ , Kadish AH |
Ref : American Journal of Physiology Heart Circ Physiol , 293 :H1629 , 2007 |
Abstract : |
PubMedSearch : Ulphani_2007_Am.J.Physiol.Heart.Circ.Physiol_293_H1629 |
PubMedID: 17545480 |
Title : d-Conopeptide EVIA isolated from Conus ermineus is a new pharmacological tool for discriminating sodium channel subtypes - |
Author(s) : Barbier J , Lamthanh H , Gall FL , Favreau P , Benoit E , Chen H , Gilles N , Ilan N , Heinemann SH , Gordon D , Menez A , Molgo J |
Ref : Journal de Physiologie (Paris) , 99 :247 , 2006 |
PubMedID: |
Title : Analysis of nicotinic acetylcholine receptor subunits in the cochlea of the mouse - Drescher_1995_Comp.Biochem.Physiol.C.Pharmacol.Toxicol.Endocrinol_112_267 |
Author(s) : Drescher DG , Khan KM , Green GE , Morley BJ , Beisel KW , Kaul H , Gordon D , Gupta AK , Drescher MJ , Barretto RL |
Ref : Comparative Biochemistry & Physiology C Pharmacol Toxicol Endocrinol , 112 :267 , 1995 |
Abstract : |
PubMedSearch : Drescher_1995_Comp.Biochem.Physiol.C.Pharmacol.Toxicol.Endocrinol_112_267 |
PubMedID: 8838678 |
Title : Localization of receptor sites for insect-selective toxins on sodium channels by site-directed antibodies - Gordon_1992_Biochemistry_31_7622 |
Author(s) : Gordon D , Moskowitz H , Eitan M , Warner C , Catterall WA , Zlotkin E |
Ref : Biochemistry , 31 :7622 , 1992 |
Abstract : |
PubMedSearch : Gordon_1992_Biochemistry_31_7622 |
PubMedID: 1324719 |