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Type Inhibitor
Isoindole
Isoindole
General
Fusion of benzene and pyrazole. Building block for many inhibitors of enzymes. Indole is an analog with only one nitrogen atom in position 1. Building block for many inhibitors of enzymes
Inhibitor
Main targeted enzyme familyes
Type
Structure
SCHEMBL1532301
ACHE
Indole
Isoindole
Acridine
Alkyl linked bis-ligand
Derivative of Tacrine
Derivative of Donepezil
Allo-Ile-isoindoline
DPP4N_Peptidase_S9
Isoindole
6H12-(R)2
ACHE
Derivative of Tacrine
Derivative of Valmerin
Urea derivative
GSK-3 kinase inhibitor
Multitarget
Isoindole
Indole
Triazol
6H13-(R)3
ACHE
Derivative of Tacrine
Derivative of Valmerin
Urea derivative
GSK-3 kinase inhibitor
Multitarget
Isoindole
Indole
Triazol
6H14-(S)6
ACHE
Derivative of Tacrine
Derivative of Valmerin
Urea derivative
GSK-3 kinase inhibitor
Multitarget
Isoindole
Indole
Triazol
R-Pro-(decarboxy-Pro)-X99
S9N_PPCE_Peptidase_S9
Pyrrolidine
Isoindole
Indole
Nijmegen-1
RsbQ-like
Cotylimide
Strigolactone receptors ligand
Isoindole
Indole
Butenolide
Phthalimido
isoquinolinederivative18
DPP4N_Peptidase_S9
Piperazine
Isoindole
Indole
1G244
DPP4N_Peptidase_S9
Piperazine
Isoindole
Indole
Phthalimido-Galanthaminium-4d
ACHE
Derivative of Galanthamine
Alkaloid
Natural_modified
Alkyl linked bis-ligand
Isoindole
Phthalimido
Benzazepin
Azepine
Phthalimido-Galanthaminium-8d
ACHE
Derivative of Galanthamine
Alkaloid
Natural_modified
Alkyl linked bis-ligand
Isoindole
Indole
Phthalimido
Benzazepin
Azepine
Dialifor-oxon
ACHE
Organophosphate
Insecticide
Isoindole
Indole
Sulfur Compound
Dialifor
ACHE
Organophosphate
Insecticide
Isoindole
Indole
Sulfur Compound
PIMP
ACHE
Organophosphate
Surrogate OP
Nerve Agent G-series
Derivative of Sarin
Phthalimido
Isoindole
Phosmet
ACHE
Organophosphate
Insecticide
Sulfur Compound
Organothiophosphate
Isoindole
Indole
Phosmetoxon
ACHE
Organophosphate
Insecticide
Sulfur Compound
Organothiophosphate
Isoindole
Indole
Phthalimido