ABPP-Probe

General

Activity-based protein profiling (ABPP) is a functional proteomic technology that uses chemical probes that react with mechanistically related classes of enzymes. The probe consists of two elements: a reactive group (RG, sometimes called a warhead) and a tag
Inhibitor Main targeted enzyme familyes Type Structure
Desthiobiotin-PEG3-Azide Carbon-carbon_bond_hydrolase Azido ABPP-Probe Biotin derivative
Lalistat-alkyne-probe Acidic_Lipase 6_AlphaBeta_hydrolase Cutinase Hormone-sensitive_lipase_like Monoglyceridelipase_lysophospholip Piperidine Lipase inhibitor Sulfur Compound Thiadiazol Alkyne ABPP-Probe
alkyne-PEG-FP Organophosphate ABPP-Probe Fluorescent Probe Alkyne
PhenylPhosphonateAzidoProbe3 Organophosphate ABPP-Probe Azido
PhenylPhosphonateAzidoProbe5 Organophosphate ABPP-Probe Azido Sulfur Compound
PhenylPhosphonateAzidoProbe4 Organophosphate ABPP-Probe Azido
ABP-C6 Hormone-sensitive_lipase_like Monoglyceridelipase_lysophospholip ABHD11-Acetyl_transferase Carb_B_Chordata A85-EsteraseD-FGH LYsophospholipase_carboxylesterase PPase_methylesterase_euk ACPH_Peptidase_S9 CGI-58_ABHD5_ABHD4 Arylacetamide_deacetylase BCHE Prolylcarboxypeptidase DPP4N_Peptidase_S9 PC-sterol_acyltransferase pNP Organophosphate ABPP-Probe Azido
NBD-CP Organophosphate ABPP-Probe NBD-nitro-benzoxadiazol-fluorescent Benzoxadiazole pNP Phenanthrene
NBD-TG Hormone-sensitive_lipase_like Monoglyceridelipase_lysophospholip ABHD11-Acetyl_transferase Triacylglycerol NBD-nitro-benzoxadiazol-fluorescent ABPP-Probe pNP Benzoxadiazole
NBD-HE-HP Hormone-sensitive_lipase_like Carb_B_Chordata Monoglyceridelipase_lysophospholip A85-EsteraseD-FGH ABHD11-Acetyl_transferase LYsophospholipase_carboxylesterase PPase_methylesterase_euk ACPH_Peptidase_S9 CGI-58_ABHD5_ABHD4 Bacterial_lip_FamI.2 Lipase_3 Carb_B_Arthropoda Juvenile_hormone_esterase S9N_PPCE_Peptidase_S9 Organophosphate ABPP-Probe NBD-nitro-benzoxadiazol-fluorescent pNP Benzoxadiazole
NBD-AE-MPF ACHE Organophosphate ABPP-Probe NBD-nitro-benzoxadiazol-fluorescent Benzoxadiazole
NBD-P-MPF ACHE Organophosphate ABPP-Probe NBD-nitro-benzoxadiazol-fluorescent Benzoxadiazole
NBD-AP-MPF ACHE Organophosphate ABPP-Probe NBD-nitro-benzoxadiazol-fluorescent Benzoxadiazole
FP-Azido Organophosphate ABPP-Probe Azido
VX-Biotin Carboxypeptidase_S10 ACHE BCHE A85-EsteraseD-FGH ACPH_Peptidase_S9 Carb_B_Chordata Hormone-sensitive_lipase_like LYsophospholipase_carboxylesterase Lipase_3 Monoglyceridelipase_lysophospholip Arylacetamide_deacetylase Thioesterase DPP4N_Peptidase_S9 PC-sterol_acyltransferase ABHD6-Lip PAF-Acetylhydrolase S9N_PREPL_Peptidase_S9 PPase_methylesterase_euk Kynurenine-formamidase Organophosphate ABPP-Probe Imidazole Sulfur Compound Biotin derivative Derivative of VX
FP-Biotin Organophosphate ABPP-Probe Imidazole Sulfur Compound Biotin derivative
FP-Desthiobiotin LIDHydrolase Organophosphate ABPP-Probe Biotin derivative
FP-TAMRA Organophosphate ABPP-Probe Benzoate Xanthene
Sal-A-alkyne Plasmodium_subtelomeric_PST-A ABHD13-BEM46 Duf_676 PGAP1 ABHD17-depalmitoylase Organophosphate Cyclic OP Lipase inhibitor ABPP-Probe Alkyne
MB064 Lipase_3 ABPP-Probe